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Bruno Melillo

Broad Institute

35H-index
114Paper Count
3.4KCitation Count
Published Papers 57
Publication Date
Minimum Inoculum of Resistance Assay for Evaluating Antitoxoplasmosis Compounds That Target Phenylalanine tRNA Synthetase
err2026-06-18
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errOAAI
errTaher Uddin; Payal Mittal; Han Xie; Bruno Melillo; Amit Sharma; Arnab K. Chatterjee; L. David Sibley
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A Global Ligandability Map of Tryptoline Butynamide Stereoprobes Identifies Covalent Inhibitors of the Actin Maturation Protease
err2026-05-20
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PREAI
errYijun Xiong; Christopher J. Reinhardt; Tracey Nguyen; Melissa A. Hoffman; Gabriel M. Simon; Bruno Melillo; Benjamin F. Cravatt
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High-throughput ligand diversification to discover chemical inducers of proximity
err2026-02-16
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errOAAI
errJames B. Shaum; Miquel Muñoz i Ordoño; Erica A. Steen; Daniela V. Wenge; Hakyung Cheong; Jordan Janowski; Moritz Hunkeler; Eric M. Bilotta; Zoe J. Rutter; Paige A. Barta; Abby M. Thornhill; Natalia Milosevich; Lauren M. Hargis; Timothy R. Bishop; Trever R. Carter; Bryce da Camara; Matthias Hinterndorfer; Lucas Dada; Wen-Ji He; Fabian Offensperger; Hirotake Furihata; Sydney R. Schweber; Charlie Hatton; Yanhe Wen; Benjamin F. Cravatt; Keary M. Engle; Katherine A. Donovan; Bruno Melillo; Seiya Kitamura; Alessio Ciulli; Scott A. Armstrong; Eric S. Fischer; Georg E. Winter; Michael A. Erb
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Correction to “Improved Bicyclic Pyrrolidine Analogues Inhibit Toxoplasma gondii Growth In Vitro and Cure Infection In Vivo”
err2026-02-05
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PREAI
errTaher Uddin; Han Xie; Payal Mittal; Chloe Ence; Anil K. Gupta; Shrushti Patil; Christy Cho; Satavisha Banerjee; Amit Sharma; Bruno Melillo; Arnab K. Chatterjee; L. David Sibley
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Targeting extrachromosomal DNA in human cancers
err2026-02-03
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PREAI
errIvy Tsz-Lo Wong; Hyerim Yi; Bruno Melillo; Benjamin F. Cravatt; Howard Y. Chang; Paul S. Mischel
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Cysteine Reactivity Profiling Identifies Host Regulators of Mycobacterium tuberculosis Replication in Human Macrophages
err2026-01-27
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PREAI
errJohn K. Neff; Kristen E. DeMeester; Paola K. Párraga Solórzano; Radu M. Suciu; Melissa M. Dix; Gabriel Simon; Max A. Gianakopoulos; Bruno Melillo; Benjamin F. Cravatt; Michael U. Shiloh
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Structural and mechanistic analysis of covalent ligands targeting the RNA-binding protein NONO
err2026-01-13
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errOAAI
errGarrett L. Lindsey; Thomas K. Hockley; Alejandro Villa Gomez; Andrew C. Marshall; William R. Brothers; Colin T. Finney; Jacob Gross; Archa H. Fox; Gene W. Yeo; Bruno Melillo; Charles S. Bond; Benjamin F. Cravatt
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Complexoform-restricted covalent TRMT112 ligands that allosterically agonize METTL5
err2026-01-08
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errOAAI
errF. Wieland Goetzke; Steffen M. Bernard; Cheng-Wei Ju; Jonathan Pollock; Kristen E. DeMeester; Jacob Gross; Gabriel M. Simon; Chuan He; Bruno Melillo; Benjamin F. Cravatt
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Proteomic Ligandability Maps of Phosphorus(V) Stereoprobes Identify Covalent TLCD1 Inhibitors
err2025-04-23
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PREAI
errSharma, Hayden A.; Bielecki, Michael; Holm, Meredith A.; Thompson, Ty M.; Yin, Yue; Cravatt, Jacob B.; Ware, Timothy B.; Reed, Alex; Nassir, Molhm; Ewing, Tamara El-Hayek; Melillo, Bruno; Bazan, J. Fernando; Baran, Phil S.
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SF3B1 thermostability as an assay for splicing inhibitor interactions
err2025-02-01
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errOAAI
errAmorello, Angela N.; Reddy, Guddeti Chandrashekar; Melillo, Bruno; Cravatt, Benjamin F.; Ghosh, Arun K.; Jurica, Melissa S.
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Covalent targeting of splicing in T cells
err2025-01-01
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PREAI
errScott, Kevin A.; Kojima, Hiroyuki; Ropek, Nathalie; Warren, Charles D.; Zhang, Tiffany L.; Hogg, Simon J.; Sanford, Henry; Webster, Caroline; Zhang, Xiaoyu; Rahman, Jahan; Melillo, Bruno; Cravatt, Benjamin F.; Lyu, Jiankun; Abdel-Wahab, Omar; Vinogradova, Ekaterina V.
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Chemical tools to expand the ligandable proteome: Diversity-oriented synthesis-based photoreactive stereoprobes
err2024-12-01
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errOAAI
errOgasawara, Daisuke; Konrad, David B.; Tan, Zher Yin; Carey, Kimberly L.; Luo, Jessica; Won, Sang Joon; Li, Haoxin; Carter, Trever R.; DeMeester, Kristen E.; Njomen, Evert; Schreiber, Stuart L.; Xavier, Ramnik J.; Melillo, Bruno; Cravatt, Benjamin F.
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Redirecting the pioneering function of FOXA1 with covalent small molecules
err2024-11-01
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PREAI
errWon, Sang Joon; Zhang, Yuxiang; Reinhardt, Christopher J.; Hargis, Lauren M.; MacRae, Nicole S.; DeMeester, Kristen E.; Njomen, Evert; Remsberg, Jarrett R.; Melillo, Bruno; Cravatt, Benjamin F.; Erb, Michael A.
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An allosteric cyclin E-CDK2 site mapped by paralog hopping with covalent probes
err2024-09-18
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PREAI
errZhang, Yuanjin; Liu, Zhonglin; Hirschi, Marscha; Brodsky, Oleg; Johnson, Eric; Won, Sang Joon; Nagata, Asako; Bezwada, Divya; Petroski, Matthew D.; Majmudar, Jaimeen D.; Niessen, Sherry; Vanarsdale, Todd; Gilbert, Adam M.; Hayward, Matthew M.; Stewart, Al E.; Nager, Andrew R.; Melillo, Bruno; Cravatt, Benjamin F.
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Bicyclic Pyrrolidine Inhibitors of Toxoplasma gondii Phenylalanine t-RNA Synthetase with Antiparasitic Potency In Vitro and Brain Exposure
err2024-05-14
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PREAI
errEnce, Chloe C.; Uddin, Taher; Borrel, Julien; Mittal, Payal; Xie, Han; Zoller, Jochen; Sharma, Amit; Comer, Eamon; Schreiber, Stuart L.; Melillo, Bruno; Sibley, L. David; Chatterjee, Arnab K.
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Proteomic Ligandability Maps of Spirocycle Acrylamide Stereoprobes Identify Covalent ERCC3 Degraders
err2024-04-03
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PREAI
errLiu, Zhonglin; Remsberg, Jarrett R.; Li, Haoxin; Njomen, Evert; Demeester, Kristen E.; Tao, Yongfeng; Xia, Guoqin; Hayward, Rachel E.; Yoo, Minjin; Nguyen, Tracey; Simon, Gabriel M.; Schreiber, Stuart L.; Melillo, Bruno; Cravatt, Benjamin F.
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Covalent Targeting As a Common Mechanism for Inhibiting NLRP3 Inflammasome Assembly
err2024-01-10
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errOAAI
errStanton, Caroline; Sun, Jie; Nutsch, Kayla; Rosarda, Jessica D.; Nguyen, Thu; Li-Ma, Chloris; Njomen, Evert; Melillo, Bruno; Kutseikin, Sergei; Saez, Enrique; Cravatt, Benjamin F.; Teijaro, John R.; Wiseman, R. Luke; Bollong, Michael J.
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Genetic crosses within and between species of Cryptosporidium
err2023-12-26
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errOAAI
errShaw, Sebastian; Cohn, Ian S.; Baptista, Rodrigo P.; Xia, Guoqin; Melillo, Bruno; Agyabeng-Dadzie, Fiifi; Kissinger, Jessica C.; Striepen, Boris
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Diversity-oriented synthesis encoded by deoxyoligonucleotides (vol 14, 4930, 2023)
err2023-11-21
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errHudson, Liam; Mason, Jeremy W.; Westphal, Matthias V.; Richter, Matthieu J. R.; Thielman, Jonathan R.; Hua, Bruce K.; Gerry, Christopher J.; Xia, Guoqin; Osswald, Heather L.; Knapp, John M.; Tan, Zher Yin; Kokkonda, Praveen; Tresco, Ben I. C.; Liu, Shuang; Reidenbach, Andrew G.; Lim, Katherine S.; Poirier, Jennifer; Capece, John; Bonazzi, Simone; Gampe, Christian M.; Smith, Nichola J.; Bradner, James E.; Coley, Connor W.; Clemons, Paul A.; Melillo, Bruno; Hon, C. Suk-Yee; Ottl, Johannes; Dumelin, Christoph E.; Schaefer, Jonas V.; Faust, Ann Marie E.; Berst, Frederic; Schreiber, Stuart L.; Zecri, Frederic J.; Briner, Karin
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Diversity-oriented synthesis encoded by deoxyoligonucleotides
err2023-08-15
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errOAAI
errHudson, Liam; Mason, Jeremy W.; Westphal, Matthias V.; Richter, Matthieu J. R.; Thielman, Jonathan R.; Hua, Bruce K.; Gerry, Christopher J.; Xia, Guoqin; Osswald, Heather L.; Knapp, John M.; Tan, Zher Yin; Kokkonda, Praveen; Tresco, Ben I. C.; Liu, Shuang; Reidenbach, Andrew G.; Lim, Katherine S.; Poirier, Jennifer; Capece, John; Bonazzi, Simone; Gampe, Christian M.; Smith, Nichola J.; Bradner, James E.; Coley, Connor W.; Clemons, Paul A.; Melillo, Bruno; Hon, C. Suk-Yee; Ottl, Johannes; Dumelin, Christoph E.; Schaefer, Jonas V.; Faust, Ann Marie E.; Berst, Frederic; Schreiber, Stuart L.; Zecri, Frederic J.; Briner, Karin
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