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Multifunctional, Fluorene-Based Modulator of Cholinergic and GABAergic Neurotransmission as a Novel Drug Candidate for Palliative Treatment of Alzheimer's Disease Panek, Dawid; Pasieka, Anna; Jonczyk, Jakub; Gawlinska, Milena; Zareba, Paula; Siwek, Agata; Wolak, Malgorzata; Mordyl, Barbara; Gluch-Lutwin, Monika; Latacz, Gniewomir; Brazzolotto, Xavier; Chantegreil, Fabien; Nachon, Florian; Zdarova Karasova, Jana; Pejchal, Jaroslav; Mzik, Martin; Sestak, Vit; Prchal, Lukas; Odvarkova, Jitka; Soukup, Ondrej; Korabecny, Jan; Sorf, Ales; Hamsikova, Marie; Zemanova, Lucie; Muckova, Lubica; Vanova, Nela; Dryja, Pola; Salat, Kinga; Hoefner, Georg; Wanner, Klaus; Wieckowska, Anna; Malawska, Barbara Share Save
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8-Hydroxyquinolylnitrones as multifunctional ligands for the therapy of neurodegenerative diseases Knez, Damijan; Diez-Iriepa, Daniel; Chioua, Mourad; Gottinger, Andrea; Denic, Milica; Chantegreil, Fabien; Nachon, Florian; Brazzolotto, Xavier; Skrzypczak-Wiercioch, Anna; Meden, Anze; Pislar, Anja; Kos, Janko; Zakelj, Simon; Stojan, Jure; Salat, Kinga; Serrano, Julia; Fernandez, Ana Patricia; Sanchez-Garcia, Aitana; Martinez-Murillo, Ricardo; Binda, Claudia; Lopez-Munoz, Francisco; Gobec, Stanislav; Marco-Contelles, Jose Share Save
Highly selective butyrylcholinesterase inhibitors related to Amaryllidaceae alkaloids- Design, synthesis, and biological evaluation Pidany, Filip; Kroustkova, Jana; Al Mamun, Abdullah; Suchankova, Daniela; Brazzolotto, Xavier; Nachon, Florian; Chantegreil, Fabien; Dolezal, Rafael; Pulkrabkova, Lenka; Muckova, Lubica; Hrabinova, Martina; Finger, Vladimir; Kufa, Martin; Soukup, Ondrej; Jun, Daniel; Jenco, Jaroslav; Kunes, Jiri; Novakova, Lucie; Korabecny, Jan; Cahlikova, Lucie Share Save
Discovery of new, highly potent and selective inhibitors of BuChE- design synthesis, in vitro and in vivo evaluation and crystallography studies Panek, Dawid; Pasieka, Anna; Latacz, Gniewomir; Zareba, Paula; Szczech, Michal; Godyn, Justyna; Chantegreil, Fabien; Nachon, Florian; Brazzolotto, Xavier; Skrzypczak-Wiercioch, Anna; Walczak, Maria; Smolik, Magdalena; Salat, Kinga; Hoefner, Georg; Wanner, Klaus; Wieckowska, Anna; Malawska, Barbara Share Save
Pseudo-irreversible butyrylcholinesterase inhibitors: Structure-activity relationships, computational and crystallographic study of the N-dialkyl O-arylcarbamate warhead Meden, Anze; Knez, Damijan; Brazzolotto, Xavier; Modeste, Fabrice; Perdih, Andrej; Pislar, Anja; Zorman, Masa; Zorovic, Maja; Denic, Milica; Pajk, Stane; Zivin, Marko; Nachon, Florian; Gobec, Stanislav Share Save
Toxicokinetics of plasmatic VX in a swine model: comparison of a simple enzymatic titration method with a mass spectrometry method Femy, F.; Meesemaecker, G.; Belverge, N.; Courageux, C.; Nervo, A.; Goulay, R.; Reymond, C.; Chantegreil, F.; Madi, M.; Nachon, F.; Taudon, N.; Jaffre, N. Share Save
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A New Class of Bi- and Trifunctional Sugar Oximes as Antidotes against Organophosphorus Poisoning Da Silva, Ophelie; Probst, Nicolas; Landry, Christophe; Hanak, Anne-Sophie; Warnault, Pierre; Coisne, Caroline; Calas, Andre-Guilhem; Gosselet, Fabien; Courageux, Charlotte; Gastellier, Anne-Julie; Trancart, Marilene; Baati, Rachid; Dehouck, Marie-Pierre; Jean, Ludovic; Nachon, Florian; Renard, Pierre-Yves; Dias, Jose Share Save
An Antidote Screening System for Organophosphorus Poisoning Using Zebrafish Larvae Dubrana, Leslie E.; Knoll-Gellida, Anja; Bourcier, Laure M.; Merce, Theo; Pedemay, Sandra; Nachon, Florian; Calas, Andre-Guilhem; Baati, Rachid; Soares, Magalie; Babin, Patrick J. Share Save
Diisopropylfluorophosphate-induced status epilepticus drives complex glial cell phenotypes in adult male mice Maupu, Clemence; Enderlin, Julie; Igert, Alexandre; Oger, Myriam; Auvin, Stephane; Hassan-Abdi, Rahma; Soussi-Yanicostas, Nadia; Brazzolotto, Xavier; Nachon, Florian; Dal Bo, Gregory; Dupuis, Nina Share Save
Sustainable Drug Discovery of Multi-Target-Directed Ligands for Alzheimer's Disease Rossi, Michele; Freschi, Michela; Nascente, Luciana de Camargo; Salerno, Alessandra; Viana Teixeira, Sarah de Melo; Nachon, Florian; Chantegreil, Fabien; Soukup, Ondrej; Prchal, Lukas; Malaguti, Marco; Bergamini, Christian; Bartolini, Manuela; Angeloni, Cristina; Hrelia, Silvana; Soares Romeiro, Luiz Antonio; Bolognesi, Maria Laura Share Save