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Florian Nachon

institut de recherche biomedicale des armees

48H-index
256Paper Count
7.9KCitation Count
Published Papers 93
Publication Date
Rational Design and Evaluation of Rivastigmine-Based Pleiotropic Prodrugs for the Treatment of Alzheimer’s Disease
err2026-04-13
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PREAI
errValentin Travers-Lesage; Marc Since; Alice Wang; Audrey Davis; Dimitri Fayolle; Benoit Bernay; Fabrice Modeste; Florian Nachon; Xavier Brazzalotto; Lucie Crouzier; Jana Sopkova-De Oliveira Santos; Tangui Maurice; Patrick Dallemagne; Christophe Rochais
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Access to novel potent pleiotropic prodrugs, targeting both butyrylcholinesterase and serotonin reuptake, with anti-amnesic activities in Alzheimer’s disease model.
err2026-02-12
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PREAI
errValentin Travers--Lesage; Lucie Crouzier; Mirjana Antonijevic; Alice Wang; François-Xavier Toublet; Audrey Davis; Fabrice Modeste; Xavier Brazzolotto; Florian Nachon; Marc Since; Tangui Maurice; Christophe Rochais; Patrick Dallemagne
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Dual Cholinergic Modulation in Dementia: Quinuclidine Carbamates Targeting Butyrylcholinesterase and α7 Nicotinic Receptor
err2025-11-15
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PREAI
errPeter Mastnak-Sokolov; Damijan Knez; Anže Meden; Nika Strašek Benedik; Svit Ferjančič Benetik; Martina Hrast Rambaher; Maša Zorman; Florian Nachon; Xavier Brazzolotto; Kent Jardemark; Oscar Jungholm; Joseph Bruton; Emilia Strandback; Tomas Nyman; Mohammed Shahid; Stanislav Gobec
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Challenges and advances in the development of antidotes against A-series nerve agents
err2025-10-06
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PREAI
errRajan K. Tripathy; Khushi Goyal; Prakash Y. Khandave; Janek Bzdrenga; Xavier Brazzolotto; Florian Nachon; Abhay H. Pande
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N-Propargylpyrrolidine-based butyrylcholinesterase and monoamine oxidase inhibitors
err2025-07-30
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errUrban Košak; Damijan Knez; Anja Pišlar; Selena Horvat; Simon Žakelj; Alexandre Igert; José Dias; Florian Nachon; Xavier Brazzolotto; Stanislav Gobec
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Chiral switch of a butyrylcholinesterase inhibitor for the treatment of Alzheimer's disease
err2025-07-23
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PREAI
errUrban Košak; Damijan Knez; Svit Ferjančič Benetik; Peter Mastnak Sokolov; Anja Pišlar; Selena Horvat; Jure Stojan; Bingbing Lv; Weiting Zhang; Yuanyuan Wang; Qinjie Wang; Alexandre Igert; José Dias; Florian Nachon; Xavier Brazzolotto; Haopeng Sun; Stanislav Gobec
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Multifunctional, Fluorene-Based Modulator of Cholinergic and GABAergic Neurotransmission as a Novel Drug Candidate for Palliative Treatment of Alzheimer's Disease
err2024-11-22
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errOAAI
errPanek, Dawid; Pasieka, Anna; Jonczyk, Jakub; Gawlinska, Milena; Zareba, Paula; Siwek, Agata; Wolak, Malgorzata; Mordyl, Barbara; Gluch-Lutwin, Monika; Latacz, Gniewomir; Brazzolotto, Xavier; Chantegreil, Fabien; Nachon, Florian; Zdarova Karasova, Jana; Pejchal, Jaroslav; Mzik, Martin; Sestak, Vit; Prchal, Lukas; Odvarkova, Jitka; Soukup, Ondrej; Korabecny, Jan; Sorf, Ales; Hamsikova, Marie; Zemanova, Lucie; Muckova, Lubica; Vanova, Nela; Dryja, Pola; Salat, Kinga; Hoefner, Georg; Wanner, Klaus; Wieckowska, Anna; Malawska, Barbara
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Role of paraoxonase 1 in organophosphate G-series nerve agent poisoning and future therapeutic strategies
err2024-10-02
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PREAI
errTripathy, Rajan K.; Khandave, Prakash Y.; Bzdrenga, Janek; Nachon, Florian; Brazzolotto, Xavier; Pande, Abhay H.
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Unveiling the Full Dynamical and Reactivity Profiles of Acetylcholinesterase: A Comprehensive All-Atom Investigation
err2024-01-19
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PREAI
errCelerse, Frederic; Lagardere, Louis; Bouchibti, Yasmine; Nachon, Florian; Verdier, Laurent; Piquemal, Jean-Philip; Derat, Etienne
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8-Hydroxyquinolylnitrones as multifunctional ligands for the therapy of neurodegenerative diseases
err2023-05-01
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errOAAI
errKnez, Damijan; Diez-Iriepa, Daniel; Chioua, Mourad; Gottinger, Andrea; Denic, Milica; Chantegreil, Fabien; Nachon, Florian; Brazzolotto, Xavier; Skrzypczak-Wiercioch, Anna; Meden, Anze; Pislar, Anja; Kos, Janko; Zakelj, Simon; Stojan, Jure; Salat, Kinga; Serrano, Julia; Fernandez, Ana Patricia; Sanchez-Garcia, Aitana; Martinez-Murillo, Ricardo; Binda, Claudia; Lopez-Munoz, Francisco; Gobec, Stanislav; Marco-Contelles, Jose
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Highly selective butyrylcholinesterase inhibitors related to Amaryllidaceae alkaloids- Design, synthesis, and biological evaluation
err2023-04-01
err6
PREAI
errPidany, Filip; Kroustkova, Jana; Al Mamun, Abdullah; Suchankova, Daniela; Brazzolotto, Xavier; Nachon, Florian; Chantegreil, Fabien; Dolezal, Rafael; Pulkrabkova, Lenka; Muckova, Lubica; Hrabinova, Martina; Finger, Vladimir; Kufa, Martin; Soukup, Ondrej; Jun, Daniel; Jenco, Jaroslav; Kunes, Jiri; Novakova, Lucie; Korabecny, Jan; Cahlikova, Lucie
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Discovery of new, highly potent and selective inhibitors of BuChE- design synthesis, in vitro and in vivo evaluation and crystallography studies
err2023-03-01
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PREAI
errPanek, Dawid; Pasieka, Anna; Latacz, Gniewomir; Zareba, Paula; Szczech, Michal; Godyn, Justyna; Chantegreil, Fabien; Nachon, Florian; Brazzolotto, Xavier; Skrzypczak-Wiercioch, Anna; Walczak, Maria; Smolik, Magdalena; Salat, Kinga; Hoefner, Georg; Wanner, Klaus; Wieckowska, Anna; Malawska, Barbara
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Pseudo-irreversible butyrylcholinesterase inhibitors: Structure-activity relationships, computational and crystallographic study of the N-dialkyl O-arylcarbamate warhead
err2023-02-01
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PREAI
errMeden, Anze; Knez, Damijan; Brazzolotto, Xavier; Modeste, Fabrice; Perdih, Andrej; Pislar, Anja; Zorman, Masa; Zorovic, Maja; Denic, Milica; Pajk, Stane; Zivin, Marko; Nachon, Florian; Gobec, Stanislav
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Toxicokinetics of plasmatic VX in a swine model: comparison of a simple enzymatic titration method with a mass spectrometry method
err2022-11-03
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PREAI
errFemy, F.; Meesemaecker, G.; Belverge, N.; Courageux, C.; Nervo, A.; Goulay, R.; Reymond, C.; Chantegreil, F.; Madi, M.; Nachon, F.; Taudon, N.; Jaffre, N.
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From tryptophan-based amides to tertiary amines: Optimization of a butyrylcholinesterase inhibitor series
err2022-04-01
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errOAAI
errMeden, Anze; Knez, Damijan; Brazzolotto, Xavier; Nachon, Florian; Dias, Jose; Svete, Jurij; Stojan, Jure; Groselj, Uros; Gobec, Stanislav
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A New Class of Bi- and Trifunctional Sugar Oximes as Antidotes against Organophosphorus Poisoning
err2022-03-07
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errOAAI
errDa Silva, Ophelie; Probst, Nicolas; Landry, Christophe; Hanak, Anne-Sophie; Warnault, Pierre; Coisne, Caroline; Calas, Andre-Guilhem; Gosselet, Fabien; Courageux, Charlotte; Gastellier, Anne-Julie; Trancart, Marilene; Baati, Rachid; Dehouck, Marie-Pierre; Jean, Ludovic; Nachon, Florian; Renard, Pierre-Yves; Dias, Jose
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An Antidote Screening System for Organophosphorus Poisoning Using Zebrafish Larvae
err2021-07-21
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PREAI
errDubrana, Leslie E.; Knoll-Gellida, Anja; Bourcier, Laure M.; Merce, Theo; Pedemay, Sandra; Nachon, Florian; Calas, Andre-Guilhem; Baati, Rachid; Soares, Magalie; Babin, Patrick J.
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Diisopropylfluorophosphate-induced status epilepticus drives complex glial cell phenotypes in adult male mice
err2021-05-01
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errOAAI
errMaupu, Clemence; Enderlin, Julie; Igert, Alexandre; Oger, Myriam; Auvin, Stephane; Hassan-Abdi, Rahma; Soussi-Yanicostas, Nadia; Brazzolotto, Xavier; Nachon, Florian; Dal Bo, Gregory; Dupuis, Nina
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Sustainable Drug Discovery of Multi-Target-Directed Ligands for Alzheimer's Disease
err2021-04-08
err72
errOAAI
errRossi, Michele; Freschi, Michela; Nascente, Luciana de Camargo; Salerno, Alessandra; Viana Teixeira, Sarah de Melo; Nachon, Florian; Chantegreil, Fabien; Soukup, Ondrej; Prchal, Lukas; Malaguti, Marco; Bergamini, Christian; Bartolini, Manuela; Angeloni, Cristina; Hrelia, Silvana; Soares Romeiro, Luiz Antonio; Bolognesi, Maria Laura
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