Not logged in First Sustainable One-Pot Tandem Hantzsch Multicomponent Reaction/Click Reaction Approach for Novel Multitarget-Directed Ligands in Alzheimer's Disease Bernard, Paul J.; Wieckowska, Anna; Grosjean, Sylvain; Godyn, Justyna; Salat, Kinga; Detka, Jan; Palacz, Natalia; Tyrybon, Weronika; Jonczyk, Jakub; Szalaj, Natalia; Zareba, Paula; Martin, Helene; Maj, Maciej; Jozwiak, Krzysztof; Marco-Contelles, Jose; Ismaili, Lhassane Share Save
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Synthesis, Anticonvulsant, Antinociceptive Activity and Preliminary Safety Evaluations of Novel Hybrid Imidazolidine-2,4-Dione Derivatives with Morpholine Moiety Czopek, Anna; Byrtus, Hanna; Gora, Malgorzata; Rapacz, Anna; Salat, Kinga; Koczurkiewicz-Adamczyk, Paulina; Pekala, Elzbieta; Obniska, Jolanta; Kaminski, Krzysztof Share Save
Multifunctional, Fluorene-Based Modulator of Cholinergic and GABAergic Neurotransmission as a Novel Drug Candidate for Palliative Treatment of Alzheimer's Disease Panek, Dawid; Pasieka, Anna; Jonczyk, Jakub; Gawlinska, Milena; Zareba, Paula; Siwek, Agata; Wolak, Malgorzata; Mordyl, Barbara; Gluch-Lutwin, Monika; Latacz, Gniewomir; Brazzolotto, Xavier; Chantegreil, Fabien; Nachon, Florian; Zdarova Karasova, Jana; Pejchal, Jaroslav; Mzik, Martin; Sestak, Vit; Prchal, Lukas; Odvarkova, Jitka; Soukup, Ondrej; Korabecny, Jan; Sorf, Ales; Hamsikova, Marie; Zemanova, Lucie; Muckova, Lubica; Vanova, Nela; Dryja, Pola; Salat, Kinga; Hoefner, Georg; Wanner, Klaus; Wieckowska, Anna; Malawska, Barbara Share Save
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Discovery of New Highly Potent Histamine H3 Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase Inhibitors Malek, Rim; Salat, Kinga; Totoson, Perle; Karcz, Tadeusz; Refouvelet, Bernard; Skrzypczak-Wiercioch, Anna; Maj, Maciej; Simakov, Alexey; Martin, Helene; Siwek, Agata; Szalaj, Natalia; Godyn, Justyna; Panek, Dawid; Wieckowska, Anna; Jozwiak, Krzysztof; Demougeot, Celine; Kiec-Kononowicz, Katarzyna; Chabchoub, Fakher; Iriepa, Isabel; Marco-Contelles, Jose; Ismaili, Lhassane Share Save
Discovery of novel multifunctional ligands targeting GABA transporters, butyrylcholinesterase, β-secretase, and amyloid β aggregation as potential treatment of Alzheimer's disease Zareba, Paula; Latka, Kamil; Mazur, Gabriela; Gryzlo, Beata; Pasieka, Anna; Godyn, Justyna; Panek, Dawid; Skrzypczak-Wiercioch, Anna; Hoefner, Georg C.; Latacz, Gniewomir; Maj, Maciej; Espargaro, Alba; Sabate, Raimon; Jozwiak, Krzysztof; Wanner, Klaus T.; Salat, Kinga; Malawska, Barbara; Kulig, Katarzyna; Bajda, Marek Share Save
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8-Hydroxyquinolylnitrones as multifunctional ligands for the therapy of neurodegenerative diseases Knez, Damijan; Diez-Iriepa, Daniel; Chioua, Mourad; Gottinger, Andrea; Denic, Milica; Chantegreil, Fabien; Nachon, Florian; Brazzolotto, Xavier; Skrzypczak-Wiercioch, Anna; Meden, Anze; Pislar, Anja; Kos, Janko; Zakelj, Simon; Stojan, Jure; Salat, Kinga; Serrano, Julia; Fernandez, Ana Patricia; Sanchez-Garcia, Aitana; Martinez-Murillo, Ricardo; Binda, Claudia; Lopez-Munoz, Francisco; Gobec, Stanislav; Marco-Contelles, Jose Share Save
Discovery of new, highly potent and selective inhibitors of BuChE- design synthesis, in vitro and in vivo evaluation and crystallography studies Panek, Dawid; Pasieka, Anna; Latacz, Gniewomir; Zareba, Paula; Szczech, Michal; Godyn, Justyna; Chantegreil, Fabien; Nachon, Florian; Brazzolotto, Xavier; Skrzypczak-Wiercioch, Anna; Walczak, Maria; Smolik, Magdalena; Salat, Kinga; Hoefner, Georg; Wanner, Klaus; Wieckowska, Anna; Malawska, Barbara Share Save
KM-408, a novel phenoxyalkyl derivative as a potential anticonvulsant and analgesic compound for the treatment of neuropathic pain Waszkielewicz, Anna; Marona, Henryk; Panczyk-Straszak, Katarzyna; Filipek, Barbara; Rapacz, Anna; Salat, Kinga; Kubacka, Monika; Cios, Agnieszka; Fedak, Filip; Walczak, Maria; Hubicka, Urszula; Kwiecien, Anna; Zuromska-Witek, Barbara; Szafranski, Przemyslaw W.; Koczurkiewicz-Adamczyk, Paulina; Pekala, Elzbieta; Przejczowska-Pomierny, Katarzyna; Pociecha, Krzysztof; Wyska, Elzbieta Share Save
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Development and crystallography-aided SAR studies of multifunctional BuChE inhibitors and 5-HT6R antagonists with β-amyloid anti-aggregation properties Wichur, Tomasz; Godyn, Justyna; Goral, Izabella; Latacz, Gniewomir; Bucki, Adam; Siwek, Agata; Gluch-Lutwin, Monika; Mordyl, Barbara; Sniecikowska, Joanna; Walczak, Maria; Knez, Damijan; Jukic, Marko; Salat, Kinga; Gobec, Stanislav; Kolaczkowski, Marcin; Malawska, Barbara; Brazzolotto, Xavier; Wieckowska, Anna Share Save
Development of tricyclic N-benzyl-4-hydroxybutanamide derivatives as inhibitors of GABA transporters mGAT1-4 with anticonvulsant, antinociceptive, and antidepressant activity Zareba, Paula; Salat, Kinga; Hoefner, Georg C.; Latka, Kamil; Bajda, Marek; Latacz, Gniewomir; Kotniewicz, Krzysztof; Rapacz, Anna; Podkowa, Adrian; Maj, Maciej; Jozwiak, Krzysztof; Filipek, Barbara; Wanner, Klaus T.; Malawska, Barbara; Kulig, Katarzyna Share Save
Novel Functionalized Amino Acids as Inhibitors of GABA Transporters with Analgesic Activity Gryzlo, Beata; Zareba, Paula; Malawska, Katarzyna; Mazur, Gabriela; Rapacz, Anna; Latka, Kamil; Hoefner, Georg C.; Latacz, Gniewomir; Bajda, Marek; Salat, Kinga; Wanner, Klaus T.; Malawska, Barbara; Kulig, Katarzyna Share Save
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