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Dual inhibitors of Pseudomonas aeruginosa virulence factors LecA and LasB Metelkina, Olga; Konstantinovic, Jelena; Klein, Andreas; Shafiei, Roya; Fares, Mario; Alhayek, Alaa; Yahiaoui, Samir; Elgaher, Walid A. M.; Haupenthal, Joerg; Titz, Alexander; Hirsch, Anna K. H. Share Save
Inhibitors of the Elastase LasB for the Treatment of Pseudomonas aeruginosa Lung Infections Konstantinovic, Jelena; Kany, Andreas M.; Alhayek, Alaa; Abdelsamie, Ahmed S.; Sikandar, Asfandyar; Voos, Katrin; Yao, Yiwen; Andreas, Anastasia; Shafiei, Roya; Loretz, Brigitta; Schoenauer, Esther; Bals, Robert; Brandstetter, Hans; Hartmann, Rolf W.; Ducho, Christian; Lehr, Claus-Michael; Beisswenger, Christoph; Mueller, Rolf; Rox, Katharina; Haupenthal, Joerg; Hirsch, Anna K. H. Share Save
Structure-Based Design of α-Substituted Mercaptoacetamides as Inhibitors of the Virulence Factor LasB from Pseudomonas aeruginosa Kaya, Cansu; Walter, Isabell; Alhayek, Alaa; Shafiei, Roya; Jezequel, Gwenaelle; Andreas, Anastasia; Konstantinovic, Jelena; Schoenauer, Esther; Sikandar, Asfandyar; Haupenthal, Joerg; Mueller, Rolf; Brandstetter, Hans; Hartmann, Rolf W.; Hirsch, Anna K. H. Share Save
N-Aryl Mercaptopropionamides as Broad-Spectrum Inhibitors of Metallo-β-Lactamases Kaya, Cansu; Konstantinovic, Jelena; Kany, Andreas M.; Andreas, Anastasia; Kramer, Jan S.; Brunst, Steffen; Weizel, Lilia; Rotter, Marco J.; Frank, Denia; Yahiaoui, Samir; Mueller, Rolf; Hartmann, Rolf W.; Haupenthal, Joerg; Proschak, Ewgenij; Wichelhaus, Thomas A.; Hirsch, Anna K. H. Share Save
Substrate-Inspired Fragment Merging and Growing Affords Efficacious LasB Inhibitors Kaya, Cansu; Walter, Isabell; Yahiaoui, Samir; Sikandar, Asfandyar; Alhayek, Alaa; Konstantinovic, Jelena; Kany, Andreas M.; Haupenthal, Jorg; Koehnke, Jesko; Hartmann, Rolf W.; Hirsch, Anna K. H. Share Save
N-Aryl-3-mercaptosuccinimides as Antivirulence Agents Targeting Pseudomonas aeruginosa Elastase and Clostridium Collagenases Konstantinovic, Jelena; Yahiaoui, Samir; Alhayek, Alaa; Haupenthal, Joerg; Schoenauer, Esther; Andreas, Anastasia; Kany, Andreas M.; Mueller, Rolf; Koehnke, Jesko; Berger, Fabian K.; Bischoff, Markus; Hartmann, Rolf W.; Brandstetter, Hans; Hirsch, Anna K. H. Share Save
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Novel Aminoquinoline Derivatives Significantly Reduce Parasite Load in Leishmania infantum Infected Mice Konstantinovic, Jelena; Videnovic, Milica; Orsini, Stefania; Bogojevic, Katarina; D'Alessandro, Sarah; Scaccabarozzi, Diletta; Jovanovic, Natasa Terzic; Gradoni, Luigi; Basilico, Nicoletta; Solaja, Bogdan A. Share Save
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New Steroidal 4-Aminoquinolines Antagonize Botulinum Neurotoxin Serotype A in Mouse Embryonic Stem Cell Derived Motor Neurons in Postintoxication Model Konstantinovic, Jelena; Kiris, Erkan; Kota, Krishna P.; Kugelman-Tonos, Johanny; Videnovic, Milica; Cazares, Lisa H.; Jovanovic, Natasa Terzic; Verbic, Tatjana Z.; Andjelkovic, Boban; Duplantier, Allen J.; Bavari, Sina; Solaja, Bogdan A. Share Save
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Reinvestigating Old Pharmacophores: Are 4-Aminoquinolines and Tetraoxanes Potential Two-Stage Antimalarials? Terzic, Natasa; Konstantinovic, Jelena; Tot, Miklos; Burojevic, Jovana; Djurkovic-Djakovic, Olgica; Srbljanovic, Jelena; Stajner, Tijana; Verbic, Tatjana; Zlatovic, Mario; Machado, Marta; Albuquerque, Ines S.; Prudencio, Miguel; Sciotii, Richard J.; Pecic, Stevan; D'Alessandro, Sarah; Taramelli, Donatella; Solaja, Bogdan A. Share Save
Second Generation Steroidal 4-Aminoquinolines Are Potent, Dual-Target Inhibitors of the Botulinum Neurotoxin Serotype A Metalloprotease and P. falciparum Malaria Videnovic, Milica; Opsenica, Dejan M.; Burnett, James C.; Gomba, Laura; Nuss, Jonathan E.; Selakovic, Zivota; Konstantinovic, Jelena; Krstic, Maja; Segan, Sandra; Zlatovic, Mario; Sciotti, Richard J.; Bavari, Sina; Solaja, Bogdan A. Share Save