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Jelena Konstantinović

helmholtz centre for infection research

11H-index
22Paper Count
292Citation Count
Published Papers 14
Publication Date
Multiparameter Optimization of Pseudomonas aeruginosa Elastase Inhibitors for Systemic Administration
err2026-02-05
err0
errOAAI
errAhmed S. Abdelsamie; Jelena Konstantinović; Andreas M. Kany; Christian Schütz; Dominik Kolling; Samira Speicher; Andreas Klein; Roya Shafiei; Mélodie Bouté; Katharina Mundry; Yu Mi Park; Brigitta Loretz; Rolf Müller; Jean-Michel Sallenave; Claus-Michael Lehr; Jesko Koehnke; Katharina Rox; Jörg Haupenthal; Anna K. H. Hirsch
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Dual inhibitors of Pseudomonas aeruginosa virulence factors LecA and LasB
err2024-01-01
err0
errOAAI
errMetelkina, Olga; Konstantinovic, Jelena; Klein, Andreas; Shafiei, Roya; Fares, Mario; Alhayek, Alaa; Yahiaoui, Samir; Elgaher, Walid A. M.; Haupenthal, Joerg; Titz, Alexander; Hirsch, Anna K. H.
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Inhibitors of the Elastase LasB for the Treatment of Pseudomonas aeruginosa Lung Infections
err2023-10-27
err7
errOAAI
errKonstantinovic, Jelena; Kany, Andreas M.; Alhayek, Alaa; Abdelsamie, Ahmed S.; Sikandar, Asfandyar; Voos, Katrin; Yao, Yiwen; Andreas, Anastasia; Shafiei, Roya; Loretz, Brigitta; Schoenauer, Esther; Bals, Robert; Brandstetter, Hans; Hartmann, Rolf W.; Ducho, Christian; Lehr, Claus-Michael; Beisswenger, Christoph; Mueller, Rolf; Rox, Katharina; Haupenthal, Joerg; Hirsch, Anna K. H.
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Structure-Based Design of α-Substituted Mercaptoacetamides as Inhibitors of the Virulence Factor LasB from Pseudomonas aeruginosa
err2022-04-22
err13
errOAAI
errKaya, Cansu; Walter, Isabell; Alhayek, Alaa; Shafiei, Roya; Jezequel, Gwenaelle; Andreas, Anastasia; Konstantinovic, Jelena; Schoenauer, Esther; Sikandar, Asfandyar; Haupenthal, Joerg; Mueller, Rolf; Brandstetter, Hans; Hartmann, Rolf W.; Hirsch, Anna K. H.
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N-Aryl Mercaptopropionamides as Broad-Spectrum Inhibitors of Metallo-β-Lactamases
err2022-02-21
err11
PREAI
errKaya, Cansu; Konstantinovic, Jelena; Kany, Andreas M.; Andreas, Anastasia; Kramer, Jan S.; Brunst, Steffen; Weizel, Lilia; Rotter, Marco J.; Frank, Denia; Yahiaoui, Samir; Mueller, Rolf; Hartmann, Rolf W.; Haupenthal, Joerg; Proschak, Ewgenij; Wichelhaus, Thomas A.; Hirsch, Anna K. H.
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Substrate-Inspired Fragment Merging and Growing Affords Efficacious LasB Inhibitors
err2021-12-13
err16
errOAAI
errKaya, Cansu; Walter, Isabell; Yahiaoui, Samir; Sikandar, Asfandyar; Alhayek, Alaa; Konstantinovic, Jelena; Kany, Andreas M.; Haupenthal, Jorg; Koehnke, Jesko; Hartmann, Rolf W.; Hirsch, Anna K. H.
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N-Aryl-3-mercaptosuccinimides as Antivirulence Agents Targeting Pseudomonas aeruginosa Elastase and Clostridium Collagenases
err2020-05-29
err28
errOAAI
errKonstantinovic, Jelena; Yahiaoui, Samir; Alhayek, Alaa; Haupenthal, Joerg; Schoenauer, Esther; Andreas, Anastasia; Kany, Andreas M.; Mueller, Rolf; Koehnke, Jesko; Berger, Fabian K.; Bischoff, Markus; Hartmann, Rolf W.; Brandstetter, Hans; Hirsch, Anna K. H.
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4-Aminoquinoline-based compounds as antileishmanial agents that inhibit the energy metabolism of Leishmania
err2019-10-01
err13
PREAI
errManzano, Jose Ignacio; Konstantinovic, Jelena; Scaccabarozzi, Diletta; Perea, Ana; Pavic, Aleksandar; Cavicchini, Loredana; Basilico, Nicoletta; Gamarro, Francisco; Solaja, Bogdan A.
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Novel Aminoquinoline Derivatives Significantly Reduce Parasite Load in Leishmania infantum Infected Mice
err2018-05-04
err13
errOAAI
errKonstantinovic, Jelena; Videnovic, Milica; Orsini, Stefania; Bogojevic, Katarina; D'Alessandro, Sarah; Scaccabarozzi, Diletta; Jovanovic, Natasa Terzic; Gradoni, Luigi; Basilico, Nicoletta; Solaja, Bogdan A.
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Human serum albumin binding of certain antimalarials
err2018-03-01
err29
errOAAI
errMarkovic, Olivera S.; Cvijetic, Ilija N.; Zlatovic, Mario V.; Opsenica, Igor M.; Konstantinovic, Jelena M.; Jovanovic, Natasa V. Terzic; Solaja, Bogdan A.; Verbic, Tatjana Z.
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New Steroidal 4-Aminoquinolines Antagonize Botulinum Neurotoxin Serotype A in Mouse Embryonic Stem Cell Derived Motor Neurons in Postintoxication Model
err2018-02-06
err11
errOAAI
errKonstantinovic, Jelena; Kiris, Erkan; Kota, Krishna P.; Kugelman-Tonos, Johanny; Videnovic, Milica; Cazares, Lisa H.; Jovanovic, Natasa Terzic; Verbic, Tatjana Z.; Andjelkovic, Boban; Duplantier, Allen J.; Bavari, Sina; Solaja, Bogdan A.
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Antimalarials with Benzothiophene Moieties as Aminoquinoline Partners
err2017-02-24
err20
errOAAI
errKonstantinovic, Jelena; Videnovic, Milica; Srbljanovic, Jelena; Djurkovic-Djakovic, Olgica; Bogojevic, Katarina; Sciotti, Richard; Solaja, Bogdan
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Reinvestigating Old Pharmacophores: Are 4-Aminoquinolines and Tetraoxanes Potential Two-Stage Antimalarials?
err2015-12-18
err30
PREAI
errTerzic, Natasa; Konstantinovic, Jelena; Tot, Miklos; Burojevic, Jovana; Djurkovic-Djakovic, Olgica; Srbljanovic, Jelena; Stajner, Tijana; Verbic, Tatjana; Zlatovic, Mario; Machado, Marta; Albuquerque, Ines S.; Prudencio, Miguel; Sciotii, Richard J.; Pecic, Stevan; D'Alessandro, Sarah; Taramelli, Donatella; Solaja, Bogdan A.
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Second Generation Steroidal 4-Aminoquinolines Are Potent, Dual-Target Inhibitors of the Botulinum Neurotoxin Serotype A Metalloprotease and P. falciparum Malaria
err2014-05-01
err31
errOAAI
errVidenovic, Milica; Opsenica, Dejan M.; Burnett, James C.; Gomba, Laura; Nuss, Jonathan E.; Selakovic, Zivota; Konstantinovic, Jelena; Krstic, Maja; Segan, Sandra; Zlatovic, Mario; Sciotti, Richard J.; Bavari, Sina; Solaja, Bogdan A.
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