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Paolo Filipponi

University of Pisa

28H-index
123Paper Count
2.1KCitation Count
Published Papers 24
Publication Date
Continuous Flow Synthesis of the PARP-1/2 Inhibitor HYDAMTIQ: Synthetic Strategy, Optimization, and Green Metrics Evaluation
err2023-11-14
err3
errOAAI
errFilipponi, Paolo; Cerra, Bruno; Piccinno, Alessandro; Camaioni, Emidio; Gioiello, Antimo
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Continuous Flow Acylation of (Hetero)aryllithiums with Polyfunctional N,N-Dimethylamides and Tetramethylurea in Toluene
err2021-09-09
err9
errOAAI
errDjukanovic, Dimitrije; Heinz, Benjamin; Mandrelli, Francesca; Mostarda, Serena; Filipponi, Paolo; Martin, Benjamin; Knochel, Paul
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Regioselective difunctionalization of pyridines via 3,4-pyridynes
err2021-01-01
err10
errOAAI
errHeinz, Benjamin; Djukanovic, Dimitrije; Filipponi, Paolo; Martin, Benjamin; Karaghiosoff, Konstantin; Knochel, Paul
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Reaction Calorimetry in Continuous Flow Mode: A New Approach for the Thermal Characterization of High Energetic and Fast Reactions
err2020-07-07
err19
PREAI
errMortzfeld, Frederik; Polenk, Jutta; Guelat, Bertrand; Venturoni, Francesco; Schenkel, Berthold; Filipponi, Paolo
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Application of Transition-Metal Catalysis, Biocatalysis, and Flow Chemistry as State-of-the-Art Technologies in the Synthesis of LCZ696
err2020-05-15
err28
PREAI
errGu, Xingxian; Zhao, Jibin; Chen, Like; Li, Yunzhong; Yu, Bo; Tian, Xiangguang; Min, Zhongcheng; Xu, Su; Gu, Huijuan; Sun, Junjie; Lu, Xiaoquan; Chang, Meng; Wang, Xufan; Zhao, Liqun; Ye, Shengqing; Yang, Hongwei; Tian, Yingtao; Gao, Feng; Gai, Yu; Jia, Guanghua; Wu, Jingjing; Wang, Yan; Zhang, Jianghua; Zhang, Xuesong; Liu, Weichun; Gu, Xin; Luo, Xi; Dong, Hai; Wang, Huaimin; Schenkel, Berthold; Venturoni, Francesco; Filipponi, Paolo; Guelat, Bertrand; Allmendinger, Thomas; Wietfeld, Bernhard; Hoehn, Pascale; Kovacic, Nikola; Hermann, Luca; Schlama, Thierry; Ruch, Thomas; Derrien, Nadine; Piechon, Philippe; Kleinbeck, Florian
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Sustainable Flow Synthesis of a Versatile Cyclopentenone Building Block
err2017-11-15
err11
errOAAI
errBaumann, Marcus; Baxendale, Ian R.; Filipponi, Paolo; Hu, Te
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Discovery of 3α,7α,11β-Trihydroxy-6α-ethyl-5β-cholan-24-oic Acid (TC-100), a Novel Bile Acid as Potent and Highly Selective FXR Agonist for Enterohepatic Disorders
err2016-10-04
err53
PREAI
errPellicciari, Roberto; Passeri, Daniela; De Franco, Francesca; Mostarda, Serena; Filipponi, Paolo; Colliva, Carolina; Gadaleta, Raffaella Maria; Franco, Placido; Carotti, Andrea; Macchiarulo, Antonio; Roda, Aldo; Moschetta, Antonio; Gioiello, Antimo
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A Simple Scale-up Strategy for Organolithium Chemistry in Flow Mode: From Feasibility to Kilogram Quantities
err2016-09-28
err46
PREAI
errHafner, Andreas; Filipponi, Paolo; Piccioni, Lorenzo; Meisenbach, Mark; Schenkel, Berthold; Venturoni, Francesco; Sedelmeier, Joerg
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Controlled Flow Precipitation as a Valuable Tool for Synthesis
err2015-11-20
err38
errOAAI
errFilipponi, Paolo; Gioiello, Antimo; Baxendale, Ian R.
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Continuous Flow Synthesis of Thieno[2,3-disoquinolin-5(4H)-one Scaffold: A Valuable Source of PARP-1 Inhibitors
err2014-05-27
err41
PREAI
errFilipponi, Paolo; Ostacolo, Carmine; Novellino, Ettore; Pellicciari, Roberto; Gioiello, Antimo
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Synthesis and Quantitative Structure-Property Relationships of Side Chain-Modified Hyodeoxycholic Acid Derivatives
err2013-08-30
err10
errOAAI
errSabbatini, Paola; Filipponi, Paolo; Sardella, Roccaldo; Natalini, Benedetto; Nuti, Roberto; Macchiarulo, Antonio; Pellicciari, Roberto; Gioiello, Antimo
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Extending SAR of bile acids as FXR ligands: Discovery of 23-N-(carbocinnamyloxy)-3α,7α-dihydroxy-6α-ethyl-24-nor-5β-cholan-23-amine
err2011-04-01
err72
PREAI
errGioiello, Antimo; Macchiarulo, Antonio; Carotti, Andrea; Filipponi, Paolo; Costantino, Gabriele; Rizzo, Giovanni; Adorini, Luciano; Pellicciari, Roberto
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Intramuscular Neridronate in Postmenopausal Women with Low Bone Mineral Density
err2008-10-23
err19
PREAI
errAdami, Silvano; Gatti, Davide; Bertoldo, Francesco; Sartori, Leonardo; Di Munno, Ombretta; Filipponi, Paolo; Marcocci, Claudio; Frediani, Bruno; Palummeri, Ernesto; Fiore, Carmelo Erio; Costi, Daniele; Rossini, Maurizio
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Quantitative heel ultrasound in a population-based study in Italy and its relationship with fracture history: the ESOPO study
err2005-09-02
err74
PREAI
errMaggi, S; Noale, M; Giannini, S; Adami, S; Defeo, D; Isaia, G; Sinigaglia, L; Filipponi, P; Crepaldi, G
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Association of quantitative heel ultrasound with history of osteoporotic fractures in elderly men: The ESOPO study
err2005-06-24
err36
PREAI
errVarenna, M; Sinigaglia, L; Adami, S; Giannini, S; Isaia, G; Maggi, S; Filipponi, P; Di Munno, O; Maugeri, D; de Feo, D; Crepaldi, G
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Effect of age, weight and lifestyle factors on calcaneal quantitative ultrasound in premenopausal women: The ESOPO study
err2004-04-01
err34
PREAI
errAdami, S; Giannini, S; Giorgino, R; Isaia, GC; Maggi, S; Sinigaglia, L; Filipponi, P; Crepaldi, G
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The effect of age, weight, and lifestyle factors on calcaneal quantitative ultrasound: the ESOPO study
err2003-04-11
err98
PREAI
errAdami, S; Giannini, S; Giorgino, R; Isaia, G; Maggi, S; Sinigaglia, L; Filipponi, P; Crepaldi, G; Di Munno, O
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Poorly controlled elderly Type 2 diabetic patients: the effects of increasing sulphonylurea dosages or adding metformin
err2001-12-24
err40
PREAI
errGregorio, F; Ambrosi, F; Manfrini, S; Velussi, M; Carle, F; Testa, R; Merante, D; Filipponi, P
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Paget's disease of bone: Benefits of neridronate as a first treatment and in cases of relapse after clodronate
errBONE
IF3.6
err1998-12-01
err26
PREAI
errFilipponi, P; Cristallini, S; Policani, G; Casciari, C; Gregorio, F
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