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SaveSynthesis, SAR and docking studies of substituted aryl phenylthiazolyl phenylcarboxamide as potential protein tyrosine phosphatase 1B (PTP1B) inhibitors
Varshney, Kanika; Gupta, Amit K.; Rawat, Arun; Srivastava, Rohit; Mishra, Akansha; Saxena, Mridula; Srivastava, Arvind K.; Jain, Sudha; Saxena, Anil K.
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SaveDesign, synthesis and biological evaluation of new substituted 5-benzylideno-2-adamantylthiazol[3,2-b][1,2,4]triazol-6(5H)ones. Pharmacophore models for antifungal activity
Tratrat, C.; Haroun, M.; Paparisva, A.; Geronikaki, A.; Kamoutsis, Ch.; Ciric, A.; Glamoclija, J.; Sokovic, M.; Fotakis, Ch.; Zoumpoulakis, P.; Bhunia, Shome S.; Saxena, Anil K.
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SaveNovel Glycoprotein VI Antagonists as Antithrombotics: Synthesis, Biological Evaluation, and Molecular Modeling Studies on 2,3-Disubstituted Tetrahydropyrido(3,4-b)indoles
Bhunia, Shome S.; Misra, Ankita; Khan, Imran A.; Gaur, Stuti; Jain, Manish; Singh, Surendra; Saxena, Aaruni; Hohlfield, Thomas; Dikshit, Madhu; Saxena, Anil K.
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SaveDesigning, synthesis of selective and high-affinity chalcone-benzothiazole hybrids as Brugia malayi thymidylate kinase inhibitors: In vitro validation and docking studies
Sashidhara, Koneni V.; Avula, Srinivasa Rao; Doharey, Pawan Kumar; Singh, L. Ravithej; Balaramnavar, Vishal M.; Gupta, Jyoti; Misra-Bhattacharya, Shailja; Rathaur, Sushma; Saxena, Anil K.; Saxena, Jitendra Kumar
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SaveNovel, potent, orally bioavailable and selective mycobacterial ATP synthase inhibitors that demonstrated activity against both replicating and non-replicating M. tuberculosis (vol 23, pg 742, 2015)
Singh, Supriya; Roy, Kuldeep K.; Khan, Shaheb R.; Kashyap, Vivek Kr; Sharma, Abhisheak; Jaiswal, Swati; Sharma, Sandeep K.; Krishnan, Manju Yasoda; Chaturvedi, Vineeta; Lal, Jawahar; Sinha, Sudhir; Dasgupta, Arunava; Srivastava, Ranjana; Saxena, Anil K.
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SaveNovel, potent, orally bioavailable and selective mycobacterial ATP synthase inhibitors that demonstrated activity against both replicating and non-replicating M. tuberculosis
Singh, Supriya; Roy, Kuldeep K.; Khan, Shaheb R.; Kashyap, Vivek Kr.; Sharma, Abhisheak; Jaiswal, Swati; Sharma, Sandeep K.; Krishnan, Manju Yasoda; Chaturvedi, Vineeta; Lal, Jawahar; Sinha, Sudhir; Gupta, Arnab D.; Srivastava, Ranjana; Saxena, Anil K.
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SaveIdentification of novel PTP1B inhibitors by pharmacophore based virtual screening, scaffold hopping and docking
Balaramnavar, Vishal M.; Srivastava, Rohit; Rahuja, Neha; Gupta, Swati; Rawat, Arun K.; Varshney, Salil; Chandasana, Hardik; Chhonker, Yashpal S.; Doharey, Pawan Kumar; Kumar, Santosh; Gautam, Sudeep; Srivastava, Swayam Prakash; Bhatta, Rabi Sankar; Saxena, Jitendra Kumar; Gaikwad, Anil Nilkanth; Srivastava, Arvind K.; Saxena, Anil K.
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SaveRohitukine inhibits in vitro adipogenesis arresting mitotic clonal expansion and improves dyslipidemia in vivo
Varshney, Salil; Shankar, Kripa; Beg, Muheeb; Balaramnavar, Vishal M.; Mishra, Sunil Kumar; Jagdale, Pankaj; Srivastava, Shishir; Chhonker, Yashpal S.; Lakshmi, Vijai; Chaudhari, Bhushan P.; Bhatta, Rabi Shankar; Saxena, Anil Kumar; Gaikwad, Anil Nilkanth
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SaveIdentification of Novel Amino Acid Derived CCK-2R Antagonists As Potential Antiulcer Agent: Homology Modeling, Design, Synthesis, and Pharmacology
Gupta, Amit K.; Varshney, Kanika; Singh, Neetu; Mishra, Vaibhav; Saxena, Mridula; Palit, Gautam; Saxena, Anil K.
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