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Philippe Sarret

universite de sherbrooke

50H-index
222Paper Count
6.4KCitation Count
Published Papers 95
Publication Date
Docking of virtual libraries identifies small-molecule agonists of neurotensin receptors with analgesic activity
err2026-07-22
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errOAAI
errNicolas Panel; Duy Duc Vo; Harald Hübner; Mattia Deluigi; Szymon Pach; Félix Bélair; Dorothee Weikert; Christoph Klenk; Mark Hilge; Niharika Shiva; Isabelle Brochu; Jean-Michel Longpré; Frida Bällgren; Aljona Saleh; Huabin Hu; Jon Kapla; Stefanie Kampen; Israel Cabeza de Vaca; Jan Kihlberg; Nina Wettschureck; Philippe Sarret; Andreas Plückthun; Peter Gmeiner; Jens Carlsson
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Improved brain penetration of neurotensin(8–13) via blood-brain barrier shuttle conjugation underlies strong analgesia
err2026-05-23
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errOAAI
errCamille Lagard; Jérôme Côté; Nathan Meneboo; Shauna Barreto; Michael Desgagné; Sabrina Beaulieu; Alain Larocque; Élie Besserer-Offroy; Karine Belleville; Karyn Kirby; Jean-Michel Longpré; Michel Demeule; Philippe Sarret
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Dual-target opioid/neurotensin ligands drive potent and safer analgesia in vivo
err2026-05-11
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errOAAI
errÉmile Breault; Jolien De Neve; Amirmohammad Ranjbaran; Alexandre Tremblay; Ines Robberechts; Frédérique Lussier; Félix Bélair; Victoria Tremblay; Brian J. Holleran; Isabelle Brochu; Nicolò Bisi; Jérôme Côté; Jean-Michel Longpré; Louis Gendron; Steven Ballet; Philippe Sarret
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A neurotensin receptor type 1-derived pepducin acts as a biased allosteric modulator to regulate target receptor function
err2025-12-30
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errOAAI
errRebecca L. Brouillette; Frédérique Lussier; Émile Breault; Nathan Meneboo; Malihe Hassanzadeh; Victoria Tremblay; Magali Chartier; Élora Midavaine; Laurence Ulrich; Jérôme Côté; Véronique Blais; Christine E. Mona; Jean-Michel Longpré; Michel Grandbois; Pierre-Luc Boudreault; Martin Audet; Élie Besserer-Offroy; Philippe Sarret
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Structure-based design of macrocyclic peptides to generate functional antibodies against G protein-coupled receptors
err2025-12-12
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errOAAI
errMarie-Edith Nepveu-Traversy; Malihe Hassanzadeh; Laurent Bruneau-Cossette; Élie Besserer-Offroy; Rebecca Brouillette; Sandra Morissette; Hassan Traboulsi; Karyn Kirby; Alexandre Murza; Jean-Michel Longpré; Billy Breton; Fernand-Pierre Gendron; Simon Gaudreau; Pierre-Luc Boudreault; Philippe Sarret
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Spotlight on Endocannabinoids in Healthy Individuals Using Volumetric Absorptive Microsampling Combined with LC-MS/MS Analysis
err2025-11-06
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errOAAI
errLounes Haroune; Sabrina Saibi; Jean-Philippe Bellenger; Matthieu Vincenot; Guillaume Léonard; Louis Gendron; Philippe Sarret
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Structure-activity relationships of contulakin-G: Design, synthesis, and characterization of Thr10 analogs for pain modulation
err2025-10-22
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errOAAI
errAnnik Lanoie; Sára Ferková; Édouard Caron-Duval; Juliana C.C. Dallagnol; Sitan Diarra; Alexandre Murza; Alexandre Tremblay; Léa Théroux; Émile Breault; Amirmohammad Ranjbaran; Léa Landry; Jérôme Côté; Jean-Michel Longpré; Pierre-Luc Boudreault; David Chatenet; Philippe Sarret
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Opioid Analgesics: Rise and Fall of Ligand Biased Signaling and Future Perspectives in the Quest for the Holy Grail
err2025-04-01
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PREAI
errBreault, Emile; Brouillette, Rebecca L.; Hebert, Terence E.; Sarret, Philippe; Besserer-Offroy, Elie
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Multitarget ligands that comprise opioid/nonopioid pharmacophores for pain management: Current state of the science
err2024-11-01
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errOAAI
errBreault, Emile; Desgagne, Michael; De Neve, Jolien; Cote, Jerome; Barlow, Thomas M. A.; Ballet, Steven; Sarret, Philippe
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Development of Macrocyclic Neurotensin Receptor Type 2 (NTS2) Opioid-Free Analgesics
err2024-10-14
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PREAI
errDesgagne, Michael; Chartier, Magali; Lagard, Camille; Ferkova, Sara; Choquette, Mathieu; Longpre, Jean-Michel; Cote, Jerome; Boudreault, Pierre-Luc; Sarret, Philippe
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Plasma Endocannabinoids Are Independently Associated With the Metabolic Function of White Adipose Tissue
err2024-09-19
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errOAAI
errDion, Dany; Noll, Christophe; Fortin, Melanie; Haroune, Lounes; Saibi, Sabrina; Sarret, Philippe; Carpentier, Andre C.
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Rational In Silico Design of Selective TMPRSS6 Peptidomimetic Inhibitors via Exploitation of the S2 Subpocket
err2024-07-19
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PREAI
errDesgagne, Michael; Desilets, Antoine; Ferkova, Sara; Lepage, Matthieu; Perreault, Olivier; Joushomme, Alexandre; Lemieux, Gabriel; Guerrab, Walid; Froehlich, Ulrike; Comeau, Christian; Sarret, Philippe; Leduc, Richard; Boudreault, Pierre-Luc
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Discovery of a CCR2-targeting pepducin therapy for chronic pain
err2024-07-01
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errOAAI
errMidavaine, Elora; Brouillette, Rebecca L.; Theberge, Elizabeth; Mona, Christine E.; Kashem, Sakeen W.; Cote, Jerome; Zeugin, Vera; Besserer-Offroy, Elie; Longpre, Jean-Michel; Marsault, Eric; Sarret, Philippe
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Dopamine-sensitive neurons in the mesencephalic locomotor region control locomotion initiation, stop, and turns
err2024-05-01
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errOAAI
errTello, Andrea Juarez; van der Zouwen, Cornelis Immanuel; Dejas, Leonie; Duque-Yate, Juan; Boutin, Joel; Medina-Ortiz, Katherine; Suresh, Jacinthlyn Sylvia; Swiegers, Jordan; Sarret, Philippe; Ryczko, Dimitri
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Apelin stimulation of the vascular skeletal muscle stem cell niche enhances endogenous repair in dystrophic mice
err2024-03-20
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PREAI
errLe Moal, Emmeran; Liu, Yuguo; Collerette-Tremblay, Jasmin; Dumontier, Simon; Fabre, Paul; Molina, Thomas; Dort, Junio; Orfi, Zakaria; Denault, Nicolas; Boutin, Joel; Michaud, Joris; Giguere, Hugo; Desroches, Alexandre; Tran, Kien; Ellezam, Benjamin; Vezina, Francois; Bedard, Sonia; Raynaud, Catherine; Balg, Frederic; Sarret, Philippe; Boudreault, Pierre-Luc; Scott, Michelle S.; Denault, Jean-Bernard; Marsault, Eric; Feige, Jerome N.; Auger-Messier, Mannix; Dumont, Nicolas A.; Bentzinger, C. Florian
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Structural insight into apelin receptor-G protein stoichiometry
err2022-07-11
err24
PREAI
errYue, Yang; Liu, Lier; Wu, Li-Jie; Wu, Yiran; Wang, Ling; Li, Fei; Liu, Junlin; Han, Gye-Won; Chen, Bo; Lin, Xi; Brouillette, Rebecca L.; Breault, Emile; Longpre, Jean-Michel; Shi, Songting; Lei, Hui; Sarret, Philippe; Stevens, Raymond C.; Hanson, Michael A.; Xu, Fei
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Size-Reduced Macrocyclic Analogues of [Pyr1]-apelin-13 Showing Negative Gα12 Bias Still Produce Prolonged Cardiac Effects
err2022-01-04
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PREAI
errTran, Kien; Sainsily, Xavier; Cote, Jerome; Coquerel, David; Couvineau, Pierre; Saibi, Sabrina; Haroune, Lounes; Besserer-Offroy, Elie; Flynn-Robitaille, Joel; Rojas, Martin Resua; Murza, Alexandre; Longpre, Jean-Michel; Auger-Messier, Mannix; Lesur, Olivier; Bouvier, Michel; Marsault, Eric; Boudreault, Pierre-Luc; Sarret, Philippe
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Apelin-13 in septic shock: effective in supporting hemodynamics in sheep but compromised by enzymatic breakdown in patients
err2021-11-23
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errOAAI
errCoquerel, David; Lamoureux, Julie; Chagnon, Frederic; Tran, Kien; Sage, Michael; Fortin-Pellerin, Etienne; Delile, Eugenie; Sainsily, Xavier; Fournier, Justin; Dumont, Audrey-Ann; Auger-Messier, Mannix; Sarret, Philippe; Marsault, Eric; Praud, Jean-Paul; Fulop, Tamas; Lesur, Olivier
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Pharmacodynamic and pharmacokinetic profiles of a neurotensin receptor type 2 (NTS2) analgesic macrocyclic analog
err2021-09-01
err8
errOAAI
errChartier, Magali; Desgagne, Michael; Sousbie, Marc; Rumsby, Charles; Chevillard, Lucie; Theroux, Lea; Haroune, Lounes; Cote, Jerome; Longpre, Jean-Michel; Boudreault, Pierre-Luc; Marsault, Eric; Sarret, Philippe
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