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Rational In Silico Design of Selective TMPRSS6 Peptidomimetic Inhibitors via Exploitation of the S2 Subpocket Desgagne, Michael; Desilets, Antoine; Ferkova, Sara; Lepage, Matthieu; Perreault, Olivier; Joushomme, Alexandre; Lemieux, Gabriel; Guerrab, Walid; Froehlich, Ulrike; Comeau, Christian; Sarret, Philippe; Leduc, Richard; Boudreault, Pierre-Luc Share Save
Discovery of a CCR2-targeting pepducin therapy for chronic pain Midavaine, Elora; Brouillette, Rebecca L.; Theberge, Elizabeth; Mona, Christine E.; Kashem, Sakeen W.; Cote, Jerome; Zeugin, Vera; Besserer-Offroy, Elie; Longpre, Jean-Michel; Marsault, Eric; Sarret, Philippe Share Save
Dopamine-sensitive neurons in the mesencephalic locomotor region control locomotion initiation, stop, and turns Tello, Andrea Juarez; van der Zouwen, Cornelis Immanuel; Dejas, Leonie; Duque-Yate, Juan; Boutin, Joel; Medina-Ortiz, Katherine; Suresh, Jacinthlyn Sylvia; Swiegers, Jordan; Sarret, Philippe; Ryczko, Dimitri Share Save
Apelin stimulation of the vascular skeletal muscle stem cell niche enhances endogenous repair in dystrophic mice Le Moal, Emmeran; Liu, Yuguo; Collerette-Tremblay, Jasmin; Dumontier, Simon; Fabre, Paul; Molina, Thomas; Dort, Junio; Orfi, Zakaria; Denault, Nicolas; Boutin, Joel; Michaud, Joris; Giguere, Hugo; Desroches, Alexandre; Tran, Kien; Ellezam, Benjamin; Vezina, Francois; Bedard, Sonia; Raynaud, Catherine; Balg, Frederic; Sarret, Philippe; Boudreault, Pierre-Luc; Scott, Michelle S.; Denault, Jean-Bernard; Marsault, Eric; Feige, Jerome N.; Auger-Messier, Mannix; Dumont, Nicolas A.; Bentzinger, C. Florian Share Save
Structural insight into apelin receptor-G protein stoichiometry Yue, Yang; Liu, Lier; Wu, Li-Jie; Wu, Yiran; Wang, Ling; Li, Fei; Liu, Junlin; Han, Gye-Won; Chen, Bo; Lin, Xi; Brouillette, Rebecca L.; Breault, Emile; Longpre, Jean-Michel; Shi, Songting; Lei, Hui; Sarret, Philippe; Stevens, Raymond C.; Hanson, Michael A.; Xu, Fei Share Save
Size-Reduced Macrocyclic Analogues of [Pyr1]-apelin-13 Showing Negative Gα12 Bias Still Produce Prolonged Cardiac Effects Tran, Kien; Sainsily, Xavier; Cote, Jerome; Coquerel, David; Couvineau, Pierre; Saibi, Sabrina; Haroune, Lounes; Besserer-Offroy, Elie; Flynn-Robitaille, Joel; Rojas, Martin Resua; Murza, Alexandre; Longpre, Jean-Michel; Auger-Messier, Mannix; Lesur, Olivier; Bouvier, Michel; Marsault, Eric; Boudreault, Pierre-Luc; Sarret, Philippe Share Save
Apelin-13 in septic shock: effective in supporting hemodynamics in sheep but compromised by enzymatic breakdown in patients Coquerel, David; Lamoureux, Julie; Chagnon, Frederic; Tran, Kien; Sage, Michael; Fortin-Pellerin, Etienne; Delile, Eugenie; Sainsily, Xavier; Fournier, Justin; Dumont, Audrey-Ann; Auger-Messier, Mannix; Sarret, Philippe; Marsault, Eric; Praud, Jean-Paul; Fulop, Tamas; Lesur, Olivier Share Save
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Pharmacodynamic and pharmacokinetic profiles of a neurotensin receptor type 2 (NTS2) analgesic macrocyclic analog Chartier, Magali; Desgagne, Michael; Sousbie, Marc; Rumsby, Charles; Chevillard, Lucie; Theroux, Lea; Haroune, Lounes; Cote, Jerome; Longpre, Jean-Michel; Boudreault, Pierre-Luc; Marsault, Eric; Sarret, Philippe Share Save