Harald H. Sitte - Publications, H-index & Citations

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Harald H. Sitte

university of texas medical branch galveston

59H-index

395Paper Count

1.1WCitation Count

Published Papers 151

Publication Date

Structural and functional basis of antinociceptive action of χ-conotoxin AoIA at the noradrenaline transporter

NATURE STRUCTURAL & MOLECULAR BIOLOGY

IF10.1

2026-07-21

OAAI

Oliver J. V. Belleza; Heng Zhang; Helmut Schmidhammer; Tye I. Gonzalez; Cosmin I. Ciotu; Nataša Tomašević; Carlo Martin M. Ocampo; Jomari C. Fernando; Johannes Koehbach; Paula Schwarz; Mounaf Al Makhlouf; Gabor Tajti; Simon Hasinger; Nina Kastner; Orcun Avsar; Bernhard Retzl; Kathrin Jäntsch; Yi Jiang; Roland Hellinger; Michael J. M. Fischer; K. Johan Rosengren; Christian W. Gruber; Aaron Joseph L. Villaraza; Thomas Stockner; Mariana Spetea; H. Eric Xu; Harald H. Sitte

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The Development of Dual-Acting OCT3/SERT Inhibitors to Probe Monoaminergic Regulation in Depression

Journal of Pharmacology and Experimental Therapeutics

IF3.8

2026-05-01

PREAI

Meccia, Salvatore; Chavez, Timothy J.; Skopec, Sophie; Ludwig, Iina; Prajapati, Ritu; Sitte, Harald; Hernandez, Gisela A. Camacho

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The Novel OCT3 Inhibitor Peficitinib Attenuates Doxorubicin-Induced Cardiotoxicity

Journal of Pharmacology and Experimental Therapeutics

IF3.8

2026-05-01

PREAI

Boeckman, Mike; Ahmed, Bagdad; Lin, Zhihong; Kumar, Damu Sunil; Ahmed, Eman; Curry, John; Ham, Alexander; Islam, Mohammad N.; Kooti, Fatemeh; Sitte, Harald; Stockner, Thomas; Corps, Kara; Wu, Meng; Peterson, Blake; Baker, Sharyn; Addison, Daniel; Sparreboom, Alex; Huang, Kevin M.

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Optimizing Cognitive Enhancement through Dopamine Transporter Modulation

Neuropharmacology

IF4.6

2026-04-12

OAAI

Marco Niello; Predrag Kalaba; Anita Cybulska-Klosowicz; Michael Kirchhofer; Iva Spreitzer; Markus Spreitzer; Judith Wackerlig-Damle; Michele Santoni; Claudia Sagheddu; Simone B. Sartori; Karl Ebner; Jana Lubec; Ahmed M. Hussein; Tamara Stojanovic; Nicolas Singewald; Marco Pistis; Gert Lubec; Harald H. Sitte

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Correction to “Next-Generation MDMA Analogue SDMA: Pharmacological and Metabolic Insights”

ACS Chemical Neuroscience

IF3.9

2026-03-04

OAAI

Nina Kastner; Núria Nadal-Gratacós; Selina Hemmer; Leticia Alves da Silva; John L. McKee; Tamara Hell; Giulia Cicalese; Marion Holy; Fatemeh Kooti; Kathrin Jäntsch; Ricarda Baron; Naomi Shacham; Bruna Cuccurazzu; Adam L. Halberstadt; John D. McCorvy; Thomas Stockner; Markus R. Meyer; Raúl López-Arnau; Matthias Grill; Harald H. Sitte

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Trials and tribulations of responsible people trying to uphold scientific standards

Research Integrity and Peer Review

IF10.7

2026-02-16

OAAI

Harald H. Sitte; Jutta Hübner; Norbert Aust; Viktor Weisshäupl; Edzard Ernst

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Next-Generation MDMA Analogue SDMA: Pharmacological and Metabolic Insights

ACS CHEMICAL NEUROSCIENCE

IF3.9

2025-12-01

PREAI

Kastner, Nina; Nadal-Gratacos, Nuria; Hemmer, Selina; da Silva, Leticia Alves; Mckee, John L.; Hell, Tamara; Cicalese, Giulia; Holy, Marion; Kooti, Fatemeh; Jantsch, Kathrin; Baron, Ricarda; Shacham, Naomi; Cuccurazzu, Bruna; Halberstadt, Adam L.; Mccorvy, John D.; Stockner, Thomas; Meyer, Markus R.; Lopez-Arnau, Raul; Grill, Matthias; Sitte, Harald H.

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Health risks of cocaine adulteration: local anesthetics as modulators of monoamine and organic cation transporters

Frontiers in Pharmacology

IF4.8

2025-11-19

OAAI

Oliver Kudlacek †; Niklas Senning †; Alexandra Karden †; Iina Ludwig; Julia Bicher; Fatemeh Kooti; Marion Holy; Thomas Stockner †; Anton Luf †; Harald H. Sitte †

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The psychedelic phenethylamine 25C-NBF, a selective 5-HT2A agonist, shows psychoplastogenic properties and rapid antidepressant effects in male rodents

Molecular Psychiatry

IF10.1

2025-11-14

OAAI

Núria Nadal-Gratacós; Pol Puigseslloses; Laura Guzmán; Nicola Weiss; Eline Pottie; Clara Riera-Colomer; Virginie Lardeux; Nathalie Thiriet; Fu-Hua Wang; Liselott Källsten; Irene Pérez-Esteban; Gabriel Ketsela; Joel Margall; Xavier Berzosa; David Pubill; Marta Rodríguez-Arias; Miren Ettcheto; Jan Kehr; Christophe Stove; Marcello Solinas; Harald H. Sitte; Elena Escubedo; Raul López-Arnau

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Prolintane analogs as hybrid monoamine transporter ligands: structural determinants and species differences

Journal of Biological Chemistry

IF3.9

2025-11-04

OAAI

Nina Kastner; Mohammad N. Islam; Michael Dybek; Evelyn Roth; Simon Heisinger; Marion Holy; Kathrin Jäntsch; Donna Walther; Thomas Stockner; Michael H. Baumann; Simon D. Brandt; Jason Wallach; Harald H. Sitte; Oliver Kudlacek

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Neurotransmitter Transporters—Unraveling Molecular Mechanisms and Therapeutic Opportunities

Journal of Neurochemistry

IF4

2025-09-22

PREAI

Harald H. Sitte; Ulrik Gether; Eurico Cabrita; Thomas Stockner

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Cell membrane cholesterol affects serotonin transporter efflux due to altered transporter oligomerization

Molecular Psychiatry

IF10.1

2025-09-02

OAAI

Deborah Rudin; Dino Luethi; Marco Niello; Jae-Won Yang; Isabella Burger; Walter Sandtner; Ruth Birner-Gruenberger; Gerhard J. Schütz; Harald H. Sitte

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A transporter's doom or destiny: SLC6A1 in health and disease, novel molecular targets and emerging therapeutic prospects

FRONTIERS IN MOLECULAR NEUROSCIENCE

IF3.8

2024-08-29

OAAI

Shah, Nikita; Kasture, Ameya S.; Fischer, Florian P.; Sitte, Harald H.; Hummel, Thomas; Sucic, Sonja

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Unveiling the crucial role of betaine: modulation of GABA homeostasis via SLC6A1 transporter (GAT1)

CELLULAR AND MOLECULAR LIFE SCIENCES

IF6.2

2024-06-17

OAAI

Bhatt, Manan; Lazzarin, Erika; Alberto-Silva, Ana Sofia; Domingo, Guido; Zerlotti, Rocco; Gradisch, Ralph; Bazzone, Andre; Sitte, Harald H.; Stockner, Thomas; Bossi, Elena

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PyrAtes: Modular Organic Salts with Large Stokes Shifts for Fluo-rescence Microscopy

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

IF16.9

2024-04-03

OAAI

Saridakis, Iakovos; Riomet, Margaux; Belleza, Oliver J. V.; Coussanes, Guilhem; Singer, Nadja K.; Kastner, Nina; Xiao, Yi; Smith, Elliot; Tona, Veronica; de la Torre, Aurelien; Lopes, Eric F.; Sanchez-Murcia, Pedro A.; Gonzalez, Leticia; Sitte, Harald H.; Maulide, Nuno

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Orphan lysosomal solute carrier MFSD1 facilitates highly selective dipeptide transport

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

IF9.1

2024-03-20

OAAI

Boytsov, Danila; Madej, Gregor M.; Horn, Georg; Blaha, Nadine; Koecher, Thomas; Sitte, Harald H.; Siekhaus, Daria; Ziegler, Christine; Sandtner, Walter; Roblek, Marko

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Structure-activity relationships of serotonergic 5-MeO-DMT derivatives: insights into psychoactive and thermoregulatory properties

MOLECULAR PSYCHIATRY

IF10.1

2024-03-14

OAAI

Puigseslloses, Pol; Nadal-Gratacos, Nuria; Ketsela, Gabriel; Weiss, Nicola; Berzosa, Xavier; Estrada-Tejedor, Roger; Islam, Mohammad Nazmul; Holy, Marion; Niello, Marco; Pubill, David; Camarasa, Jordi; Escubedo, Elena; Sitte, Harald H.; Lopez-Arnau, Raul

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Ligand coupling mechanism of the human serotonin transporter differentiates substrates from inhibitors

NATURE COMMUNICATIONS

IF15.7

2024-01-10

OAAI

Gradisch, Ralph; Schlogl, Katharina; Lazzarin, Erika; Niello, Marco; Maier, Julian; Mayer, Felix P.; da Silva, Leticia Alves; Skopec, Sophie M. C.; Blakely, Randy D.; Sitte, Harald H.; Mihovilovic, Marko D.; Stockner, Thomas

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Interactions of calmodulin kinase II with the dopamine transporter facilitate cocaine-induced enhancement of evoked dopamine release

TRANSLATIONAL PSYCHIATRY

IF6.2

2023-06-13

OAAI

Keighron, Jacqueline D.; Bonaventura, Jordi; Li, Yang; Yang, Jae-Won; DeMarco, Emily M. M.; Hersey, Melinda; Cao, Jianjing; Sandtner, Walter; Michaelides, Michael; Sitte, Harald H. H.; Newman, Amy Hauck; Tanda, Gianluigi

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Ethanol inhibits dopamine uptake via organic cation transporter 3: Implications for ethanol and cocaine co-abuse

MOLECULAR PSYCHIATRY

IF10.1

2023-06-13

OAAI

Clauss, N. J.; Mayer, F. P.; Owens, W. A.; Vitela, M.; Clarke, K. M.; Bowman, M. A.; Horton, R. E.; Gruendemann, D.; Schmid, D.; Holy, M.; Gould, G. G.; Koek, W.; Sitte, H. H.; Daws, L. C.

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Research Directions