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Ross McGuire

Radboud University Nijmegen

30H-index
90Paper Count
3.5KCitation Count
Published Papers 19
Publication Date
3D-e-Chem: Structural Cheminformatics Workflows for Computer-Aided Drug Discovery
err2018-02-14
err13
errOAAI
errKooistra, Albert J.; Vass, Marton; McGuire, Ross; Leurs, Rob; de Esch, Iwan J. P.; Vriend, Gert; Verhoeven, Stefan; de Graaf, Chris
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3D-e-Chem-VM: Structural Cheminformatics Research Infrastructure in a Freely Available Virtual Machine
err2017-02-14
err24
errOAAI
errMcGuire, Ross; Verhoeven, Stefan; Vass, Marton; Vriend, Gerrit; de Esch, Iwan J. P.; Lusher, Scott J.; Leurs, Rob; Ridder, Lars; Kooistra, Albert J.; Ritschel, Tina; de Graaf, Chris
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Discovery of Glycine Sulfonamides as Dual Inhibitors of sn-1-Diacylglycerol Lipase α and α/β-Hydrolase Domain 6
err2014-07-23
err35
PREAI
errJanssen, Freek J.; Deng, Hui; Baggelaar, Marc P.; Allara, Marco; van der Wel, Tom; den Dulk, Hans; Ligresti, Alessia; van Esbroeck, Annelot C. M.; McGuire, Ross; Di Marzo, Vincenzo; Overkleeft, Herman S.; van der Stelt, Mario
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Data-driven medicinal chemistry in the era of big data
err2014-07-01
err100
PREAI
errLusher, Scott J.; McGuire, Ross; van Schaik, Rene C.; Nicholson, C. David; de Vlieg, Jacob
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X-ray Structures of Progesterone Receptor Ligand Binding Domain in Its Agonist State Reveal Differing Mechanisms for Mixed Profiles of 11β-Substituted Steroids
err2012-06-01
err32
errOAAI
errLusher, Scott J.; Raaijmakers, Hans C. A.; Vu-Pham, Diep; Kazemier, Bert; Bosch, Rolien; McGuire, Ross; Azevedo, Rita; Hamersma, Hans; Dechering, Koen; Oubrie, Arthur; van Duin, Marcel; de Vlieg, Jacob
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A Prospective Cross-Screening Study on G-Protein-Coupled Receptors: Lessons Learned in Virtual Compound Library Design
err2012-05-23
err33
PREAI
errSanders, Marijn P. A.; Roumen, Luc; van der Horst, Eelke; Lane, J. Robert; Vischer, Henry F.; van Offenbeek, Jody; de Vries, Henk; Verhoeven, Stefan; Chow, Ken Y.; Verkaar, Folkert; Beukers, Margot W.; McGuire, Ross; Leurs, Rob; IJzerman, Adriaan P.; de Vlieg, Jacob; de Esch, Iwan J. P.; Zaman, Guido J. R.; Klomp, Jan P. G.; Bender, Andreas; de Graaf, Chris
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Drug design for ever, from hype to hope
err2012-01-18
err38
errOAAI
errSeddon, G.; Lounnas, V.; McGuire, R.; van den Bergh, T.; Bywater, R. P.; Oliveira, L.; Vriend, G.
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Structural Basis for Agonism and Antagonism for a Set of Chemically Related Progesterone Receptor Modulators
err2011-10-01
err38
errOAAI
errLusher, Scott J.; Raaijmakers, Hans C. A.; Vu-Pham, Diep; Dechering, Koen; Lam, Tsang Wai; Brown, Angus R.; Hamilton, Niall M.; Nimz, Olaf; Bosch, Rolien; McGuire, Ross; Oubrie, Arthur; de Vlieg, Jacob
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A molecular informatics view on best practice in multi-parameter compound optimization
err2011-07-01
err14
PREAI
errLusher, Scott J.; McGuire, Ross; Azevedo, Rita; Boiten, Jan-Willem; van Schaik, Rene C.; de Vlieg, Jacob
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α-amino acid phenolic ester derivatives:: Novel water-soluble general anesthetic agents which allosterically modulate GABAA receptors
err2001-09-14
err36
PREAI
errAnderson, A; Belelli, D; Bennett, DJ; Buchanan, KI; Casula, A; Cooke, A; Feilden, H; Gemmell, DK; Hamilton, NM; Hutchinson, EJ; Lambert, JJ; Maidment, MS; McGuire, R; McPhail, P; Miller, S; Muntoni, A; Peters, JA; Sansbury, FH; Stevenson, D; Sundaram, H
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The first potent and selective inhibitors of the glycine transporter type 2
err2001-07-25
err110
PREAI
errCaulfield, WL; Collie, IT; Dickins, RS; Epemolu, O; McGuire, R; Hill, DR; McVey, G; Morphy, JR; Rankovic, Z; Sundaram, H
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Non-depolarizing neuromuscular blocking activity of bisquaternary amino di- and tripeptide derivatives
err2000-11-08
err9
PREAI
errBooij, LHDJ; van der Broek, LAGM; Caulfield, W; Dommerholt-Caris, BMG; Clark, JK; van Egmond, J; McGuire, R; Muir, AW; Ottenheijm, HCJ; Rees, DC
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Conformationally constrained anesthetic steroids that modulate GABAA receptors
err2000-10-19
err71
PREAI
errAnderson, A; Boyd, AC; Clark, JK; Fielding, L; Gemmell, DK; Hamilton, NM; Maidment, MS; May, V; McGuire, R; McPhail, P; Sansbury, FH; Sundaram, H; Taylor, R
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