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Arthur Christopoulos

universidad de cordoba

95H-index
1.9KPaper Count
4.1WCitation Count
Published Papers 303
Publication Date
The Concise Guide to PHARMACOLOGY 2025/26: G protein-coupled receptors
err2025-12-01
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errAlexander, Stephen P. H.; Davenport, Anthony P.; Kelly, Eamonn; Gibb, Alasdair J.; Mathie, Alistair A.; Peach, Chloe J.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George R.; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bennett, Kirstie A.; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria A.; Bonaventure, Pascal; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Brown, Andrew J.; Burnstock, Geoffrey; Busnelli, Marta; Calo, Girolamo; Caruso, Vanni; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Christopoulos, Arthur; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dautzenberg, Frank M.; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Dubocovich, Margarita L.; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Forsman, Huamei Fu; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gbahou, Florence; Gerard, Craig; Gershengorn, Marvin; Glass, Michelle; Gloriam, David E.; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gruber, Christian; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hartman, Deborah S.; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Heitman, Laura; Herr, Deron R.; Hollenberg, Morley D.; Holliday, Nicholas D.; Holst, Birgitte; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; IJzerman, Adriaan P.; Inagami, Tadashi; Insel, Paul A.; Jacobson, Kenneth A.; Jacobson, Laura H.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kinsolving, Julia; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Laishram, Luxmichan; Langenhan, Tobias; Langmead, Christopher J.; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Leurs, Rob; Li, Xaria X.; Liebscher, Ines; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet J.; Malfacini, Davide; Manning, Maurice; Marangon, Davide; Martemyanov, Kirill; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Neubig, Richard R.; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Perry-Hauser, Nicole; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Qin, Helena Chengxue; Quinn, Mark; Raffaele, Stefano; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Buzon, Alejandro Romeral; Rondard, Philippe; Rosenkilde, Mette M.; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Scholz, Nicole; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Shukla, Arun K.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Smith, Nicola J.; Staeubert, Claudia; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David M.; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Verbalis, Joseph G.; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Wu, Huixian; Yang, Cheng; Yao, Chengcan; Ye, Richard D.; Zaidman, Nathan
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Structure-Activity Relationships of Highly Potent and Selective A2B Adenosine Receptor Agonists
err2025-10-01
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PREAI
errSmedley, Christopher J.; Awalt, Jon Kyle; Nguyen, Anh T. N.; Wang, Bing H.; Christopoulos, Arthur; Jorg, Manuela; May, Lauren T.; Scammells, Peter J.
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682. THE EFFECTS OF MATERNAL IMMUNE ACTIVATION ON THE PHOSPHO-PROTEOME OF THE DEVELOPING ADOLESCENT MOUSE HIPPOCAMPUS
err2025-08-18
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errU Thivisol; L Dwomoh; C Choy; J Cole; A Merritt; S Liong; S Luza; S Selemidis; A Tobin; A Christopoulos; J Nithianantharajah; C Pantelis
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Molecular basis of ligand binding and receptor activation at the human A3 adenosine receptor
err2025-08-18
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errLiudi Zhang; Jesse I. Mobbs; Felix M. Bennetts; Hariprasad Venugopal; Anh T. N. Nguyen; Arthur Christopoulos; Daan van der Es; Laura H. Heitman; Lauren T. May; Alisa Glukhova; David M. Thal
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SEX-DEPENDENT AND DYNAMIC BRAIN STRUCTURAL MRI CHANGES IN MICE FOLLOWING INFLUENZA A VIRUS MATERNAL IMMUNE ACTIVATION
err2025-08-01
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errPeng, D.; Choy, C.; Liong, S.; Brkljaca, R.; Merritt, A.; Wannan, C.; Thivisol, U.; Wright, D.; Christopoulos, A.; Selemidis, S.; Nithianantharajah, J.; Syeda, W.; Pantelis, C.
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Cryo-EM reveals an extrahelical allosteric binding site at the M5 mAChR
err2025-07-31
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errWessel A. C. Burger; Jesse I. Mobbs; Bhavika Rana; Jinan Wang; Keya Joshi; Patrick R. Gentry; Mahmuda Yeasmin; Hariprasad Venugopal; Aaron M. Bender; Craig W. Lindsley; Yinglong Miao; Arthur Christopoulos; Celine Valant; David M. Thal
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A Structure–Activity Relationship Study of Novel Positive Allosteric Modulators for the δ-Opioid Receptor
err2025-07-18
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PREAI
errOwindeep Deo; Vi Pham; Sadia Alvi; Nicholas Barnes; Arisbel B. Gondin; Arthur Christopoulos; Daniel P. Poole; Simona E. Carbone; David M. Thal; Manuela Jörg; Ben Capuano; Celine Valant; Peter J. Scammells
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The Prosperity and Adversity of M4 Muscarinic Acetylcholine Receptor Activators in the Treatment of Neuropsychiatric Disorders
err2025-04-16
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PREAI
errLiu, Boqun; Christopoulos, Arthur; Thal, David M.; Capuano, Ben; Valant, Celine; Scammells, Peter J.
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Isoquinoline small molecule ligands are agonists and probe-dependent allosteric modulators of the glucagon subfamily of GPCRs
err2024-11-01
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errYuliantie, Elita; Trinh, Phuc N. H.; Hick, Caroline; Ebenhoch, Rebecca; Nar, Herbert; Weichert, Dietmar; Christopoulos, Arthur; Sexton, Patrick M.; Wootten, Denise
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Ligand-directed biased agonism at human histamine H3 receptor isoforms across Gαi/o- and β-arrestin2-mediated pathways
err2024-10-01
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errRahman, Sabrina N.; Imhaouran, Faissal; Leurs, Rob; Christopoulos, Arthur; Valant, Celine; Langmead, Christopher J.
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Positive allosteric modulation of a GPCR ternary complex
err2024-09-13
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errBurger, Wessel A. C.; Draper-Joyce, Christopher J.; Valant, Celine; Christopoulos, Arthur; Thal, David M.
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Brain region-specific alterations in gene expression trajectories in the offspring born from influenza A virus infected mice
err2024-08-01
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errLiong, Stella; Choy, K. H. Christopher; De Luca, Simone N.; Liong, Felicia; Coward-Smith, Madison; Oseghale, Osezua; Miles, Mark A.; Vlahos, Ross; Valant, Celine; Nithianantharajah, Jess; Pantelis, Christos; Christopoulos, Arthur; Selemidis, Stavros
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Discovery of 2-Methyl-5-(1H-pyrazol-4-yl)pyridines and Related Heterocycles as Promising M4 mAChR Positive Allosteric Modulators for the Treatment of Neurocognitive Disorders
err2024-07-18
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PREAI
errLiu, Boqun; Thompson, Geoff; Jorg, Manuela; Barnes, Nicholas; Thal, David M.; Christopoulos, Arthur; Capuano, Ben; Valant, Celine; Scammells, Peter J.
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Impact of secretin receptor homo-dimerization on natural ligand binding
err2024-05-23
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errHarikumar, Kaleeckal G.; Piper, Sarah J.; Christopoulos, Arthur; Wootten, Denise; Sexton, Patrick M.; Miller, Laurence J.
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The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors
err2023-12-20
err149
errOAAI
errAlexander, Stephen P. H.; Christopoulos, Arthur; Davenport, Anthony P.; Kelly, Eamonn; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Burnstock, Geoffrey; Calo, Girolamo; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gerard, Craig; Gershengorn, Marvin; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Herr, Deron; Hollenberg, Morley D.; Holliday, Nicholas D.; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; Ijzerman, Adriaan P.; Inagami, Tadashi; Jacobson, Kenneth A.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Langenhan, Tobias; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Li, Xaria X.; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet; Malfacini, Davide; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Quinn, Mark; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Rondard, Philippe; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Yao, Chengcan; Ye, Richard D.
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Design, synthesis and evaluation of novel 2-phenyl-3-(1H-pyrazol-4-yl) pyridine positive allosteric modulators for the M4 mAChR
err2023-10-01
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PREAI
errJorg, Manuela; van der Westhuizen, Emma T.; Lu, Yao; Choy, K. H. Christopher; Shackleford, David M.; Khajehali, Elham; Tobin, Andrew B.; Thal, David M.; Capuano, Ben; Christopoulos, Arthur; Valant, Celine; Scammells, Peter J.
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Xanomeline displays concomitant orthosteric and allosteric binding modes at the M4 mAChR
err2023-09-06
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errBurger, Wessel A. C.; Pham, Vi; Vuckovic, Ziva; Powers, Alexander S.; Mobbs, Jesse I.; Laloudakis, Yianni; Glukhova, Alisa; Wootten, Denise; Tobin, Andrew B.; Sexton, Patrick M.; Paul, Steven M.; Felder, Christian C.; Danev, Radostin; Dror, Ron O.; Christopoulos, Arthur; Valant, Celine; Thal, David M.
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Role of Conserved Tyrosine Lid Residues in the Activation of the M2 Muscarinic Acetylcholine ReceptorS
err2023-09-01
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errPham, Vi; Jansen, Maria Clazina Cornelia Habben; Thompson, Geoff; Heitman, Laura H.; Christopoulos, Arthur; Thal, David M.; Valant, Celine
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Structure-based virtual screening discovers potent and selective adenosine A1 receptor antagonists
err2023-09-01
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errMatricon, Pierre; Nguyen, Anh T. N.; Vo, Duc Duy; Baltos, Jo-Anne; Jaiteh, Mariama; Luttens, Andreas; Kampen, Stefanie; Christopoulos, Arthur; Kihlberg, Jan; May, Lauren Therese; Carlsson, Jens
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