arrow
Back
V

Vadim Cherezov

university of southern california

81H-index
306Paper Count
3.7WCitation Count
Published Papers 87
Publication Date
Molecular mechanisms for subtype selectivity of kinin receptors’ antagonists
err2026-05-25
err0
errOAAI
errMeng Xia; Aleksey Raskovalov; My V. T. Nguyen; Shiliu Mei; Donggyun Kim; Jayden Salve; Vsevolod Katritch; Vadim Cherezov; Haitao Zhang
errShare
errSave
ABEL-FRET bridges the timescale gap in single-molecule measurements of the structural dynamics in the A2A adenosine receptor
err2026-03-09
err0
errOAAI
errIvan Maslov; Valentin Borshchevskiy; Iván Pérez; Vadim Cherezov; Johan Hofkens; Jelle Hendrix; Michael Börsch; Thomas Gensch
errShare
errSave
Novel fold and wing structure of Forkhead transcription factor facilitate DNA binding
err2025-10-14
err0
errOAAI
errWang, George L.; Jiang, Yibei; Sun, Yuying; Nasertorabi, Fariborz; Weller, Jesse A.; Mitra, Raktim; Batyuk, Alexander; Aparicio, Oscar M.; Cherezov, Vadim; Rohs, Remo
errShare
errSave
Structural insights into the mechanism of activation and inhibition of the prostaglandin D2 receptor 1
err2025-10-08
err0
errOAAI
errBehnaz Davoudinasab; Aleksey Raskovalov; Woojin Lee; Donggyun Kim; Heesoo Kim; Jordy Homing Lam; Gye Won Han; Vsevolod Katritch; Vadim Cherezov
errShare
errSave
In Science Journals
errScience
IF45.8
err2025-08-28
err0
PREAI
errAngela Hessler; Bianca Lopez; Michael A. Funk; Marc S. Lavine; Ian S. Osborne; Vadim Cherezov; Jack Huang; Annalisa VanHook; Jesse Smith; Mattia Maroso; Yevgeniya Nusinovich; Stella M. Hurtley; Sarah H. Ross; Sacha Vignieri; Christiana N. Fogg; John Delaney; Catherine Charneski
errShare
errSave
Unlocking GPCR-ligand interactions: Measuring binding affinities with thermal shift assay
err2025-04-18
err0
PREAI
errDashevskii, Dmitrii; Luginina, Aleksandra; Maslov, Ivan; Shevelyova, Marina; Khorn, Polina; Dmitrieva, Daria; Kapranov, Ivan; Belousov, Anatolii; Permyakov, Sergei; Cherezov, Vadim; Borshchevskiy, Valentin; Mishin, Alexey
errShare
errSave
Structural insights into the high basal activity and inverse agonism of the orphan receptor GPR6 implicated in Parkinson's disease
err2024-12-03
err0
PREAI
errBarekatain, Mahta; Johansson, Linda C.; Lam, Jordy H.; Chang, Hao; Sadybekov, Anastasiia V.; Han, Gye Won; Russo, Joseph; Bliesath, Joshua; Brice, Nicola L.; Carlton, Mark B. L.; Saikatendu, Kumar S.; Sun, Hukai; Murphy, Sean T.; Monenschein, Holger; Schiffer, Hans H.; Popov, Petr; Lutomski, Corinne A.; Robinson, Carol V.; Liu, Zhi-Jie; Hua, Tian; Katritch, Vsevolod; Cherezov, Vadim
errShare
errSave
Structure basis of ligand recognition and activation of GPR55
err2024-10-31
err0
PREAI
errChang, Hao; Li, Xiaoting; Shen, Ling; Ge, Xuanrui; Hao, Shuming; Wu, Lijie; Liu, Shenhui; Liu, Junlin; Cherezov, Vadim; Hua, Tian
errShare
errSave
Nicotinamide Riboside and CD38: Covalent Inhibition and Live-Cell Labeling
errJACS AU
IF8.7
err2024-10-30
err0
errOAAI
errKao, Guoyun; Zhang, Xiao-Nan; Nasertorabi, Fariborz; Katz, Benjamin B.; Li, Zeyang; Dai, Zhefu; Zhang, Zeyu; Zhang, Lei; Louie, Stan G.; Cherezov, Vadim; Zhang, Yong
errShare
errSave
ONE-GO: Direct detection of context-dependent GPCR activity
err2024-04-30
err0
errOAAI
errRaskovalov, Aleksey; Kim, Donggyun; Cherezov, Vadim
errShare
errSave
Structural diversity of leukotriene G-protein coupled receptors
err2023-10-01
err5
errOAAI
errLuginina, Aleksandra; Gusach, Anastasiia; Lyapina, Elizaveta; Khorn, Polina; Safronova, Nadezda; Shevtsov, Mikhail; Dmitirieva, Daria; Dashevskii, Dmitrii; Kotova, Tatiana; Smirnova, Ekaterina; Borshchevskiy, Valentin; Cherezov, Vadim; Mishin, Alexey
errShare
errSave
Structural insights into angiotensin receptor signaling modulation by balanced and biased agonists
err2023-04-11
err12
errOAAI
errZhang, Dongqi; Liu, Yongfeng; Zaidi, Saheem A.; Xu, Lingyi; Zhan, Yuting; Chen, Anqi; Guo, Jiangtao; Huang, Xi-Ping; Roth, Bryan L.; Katritch, Vsevolod; Cherezov, Vadim; Zhang, Haitao
errShare
errSave
Sub-millisecond conformational dynamics of the A2A adenosine receptor revealed by single-molecule FRET
err2023-04-03
err13
errOAAI
errMaslov, Ivan; Volkov, Oleksandr; Khorn, Polina; Orekhov, Philipp; Gusach, Anastasiia; Kuzmichev, Pavel; Gerasimov, Andrey; Luginina, Aleksandra; Coucke, Quinten; Bogorodskiy, Andrey; Gordeliy, Valentin; Wanninger, Simon; Barth, Anders; Mishin, Alexey; Hofkens, Johan; Cherezov, Vadim; Gensch, Thomas; Hendrix, Jelle; Borshchevskiy, Valentin
errShare
errSave
The activation mechanism and antibody binding mode for orphan GPR20
err2023-02-28
err7
errOAAI
errLin, Xi; Jiang, Shan; Wu, Yiran; Wei, Xiaohu; Han, Gye-Won; Wu, Lijie; Liu, Junlin; Chen, Bo; Zhang, Zhibin; Zhao, Suwen; Cherezov, Vadim; Xu, Fei
errShare
errSave
High ligand efficiency quinazoline compounds as novel A2A adenosine receptor antagonists
err2022-11-01
err8
errOAAI
errBolteau, Raphael; Duroux, Romain; Laversin, Amelie; Vreulz, Brandon; Shiriaeva, Anna; Stauch, Benjamin; Han, Gye Won; Cherezov, Vadim; Renault, Nicolas; Barczyk, Amelie; Ravez, Severine; Coevoet, Mathilde; Melnyk, Patricia; Liberelle, Maxime; Yous, Said
errShare
errSave
GPCR Agonist-to-Antagonist Conversion: Enabling the Design of Nucleoside Functional Switches for the A2A Adenosine Receptor
err2022-08-17
err13
errOAAI
errShiriaeva, Anna; Park, Daejin; Kim, Gyudong; Lee, Yoonji; Hou, Xiyan; Jarhad, Dnyandev B.; Kim, Gibae; Yu, Jinha; Hyun, Young Eum; Kim, Woomi; Gao, Zhan-Guo; Jacobson, Kenneth A.; Han, Gye Won; Stevens, Raymond C.; Jeong, Lak Shin; Choi, Sun; Cherezov, Vadim
errShare
errSave
Structural basis for receptor selectivity and inverse agonism in S1P5 receptors
err2022-08-12
err8
errOAAI
errLyapina, Elizaveta; Marin, Egor; Gusach, Anastasiia; Orekhov, Philipp; Gerasimov, Andrey; Luginina, Aleksandra; Vakhrameev, Daniil; Ergasheva, Margarita; Kovaleva, Margarita; Khusainov, Georgii; Khorn, Polina; Shevtsov, Mikhail; Kovalev, Kirill; Bukhdruker, Sergey; Okhrimenko, Ivan; Popov, Petr; Hu, Hao; Weierstall, Uwe; Liu, Wei; Cho, Yunje; Gushchin, Ivan; Rogachev, Andrey; Bourenkov, Gleb; Park, Sehan; Park, Gisu; Hyun, Hyo Jung; Park, Jaehyun; Gordeliy, Valentin; Borshchevskiy, Valentin; Mishin, Alexey; Cherezov, Vadim
errShare
errSave
Inhibition of the angiotensin II type 2 receptor AT2R is a novel therapeutic strategy for glioblastoma
err2022-08-02
err7
errOAAI
errPerryman, Richard; Renziehausen, Alexander; Shaye, Hamidreza; Kostagianni, Androniki D.; Tsiailanis, Antonis D.; Thorne, Thomas; Chatziathanasiadou, Maria, V; Sivolapenko, Gregory B.; El Mubarak, Mohamed Ahmed; Han, Gye Won; Zarzycka, Barbara; Katritch, Vsevolod; Lebon, Guillaume; Lo Nigro, Cristiana; Lattanzio, Laura; Morse, Sophie, V; Choi, James J.; O'Neill, Kevin; Kanaki, Zoi; Klinakis, Apostolos; Crook, Tim; Cherezov, Vadim; Tzakos, Andreas G.; Syed, Nelofer
errShare
errSave
MicroED structure of the human adenosine receptor determined from a single nanocrystal in LCP
err2021-09-07
err38
PREAI
errMartynowycz, Michael W.; Shiriaeva, Anna; Ge, Xuanrui; Hattne, Johan; Nannenga, Brent L.; Cherezov, Vadim; Gonen, Tamir
errShare
errSave
Molecular basis for lipid recognition by the prostaglandin D2 receptor CRTH2
err2021-08-02
err13
errOAAI
errLiu, Heng; Deepak, R. N. V. Krishna; Shiriaeva, Anna; Gati, Cornelius; Batyuk, Alexander; Hu, Hao; Weierstall, Uwe; Liu, Wei; Wang, Lei; Cherezov, Vadim; Fan, Hao; Zhang, Cheng
errShare
errSave