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Novel fold and wing structure of Forkhead transcription factor facilitate DNA binding Wang, George L.; Jiang, Yibei; Sun, Yuying; Nasertorabi, Fariborz; Weller, Jesse A.; Mitra, Raktim; Batyuk, Alexander; Aparicio, Oscar M.; Cherezov, Vadim; Rohs, Remo Share Save
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Unlocking GPCR-ligand interactions: Measuring binding affinities with thermal shift assay Dashevskii, Dmitrii; Luginina, Aleksandra; Maslov, Ivan; Shevelyova, Marina; Khorn, Polina; Dmitrieva, Daria; Kapranov, Ivan; Belousov, Anatolii; Permyakov, Sergei; Cherezov, Vadim; Borshchevskiy, Valentin; Mishin, Alexey Share Save
Structural insights into the high basal activity and inverse agonism of the orphan receptor GPR6 implicated in Parkinson's disease Barekatain, Mahta; Johansson, Linda C.; Lam, Jordy H.; Chang, Hao; Sadybekov, Anastasiia V.; Han, Gye Won; Russo, Joseph; Bliesath, Joshua; Brice, Nicola L.; Carlton, Mark B. L.; Saikatendu, Kumar S.; Sun, Hukai; Murphy, Sean T.; Monenschein, Holger; Schiffer, Hans H.; Popov, Petr; Lutomski, Corinne A.; Robinson, Carol V.; Liu, Zhi-Jie; Hua, Tian; Katritch, Vsevolod; Cherezov, Vadim Share Save
Structure basis of ligand recognition and activation of GPR55 Chang, Hao; Li, Xiaoting; Shen, Ling; Ge, Xuanrui; Hao, Shuming; Wu, Lijie; Liu, Shenhui; Liu, Junlin; Cherezov, Vadim; Hua, Tian Share Save
Nicotinamide Riboside and CD38: Covalent Inhibition and Live-Cell Labeling Kao, Guoyun; Zhang, Xiao-Nan; Nasertorabi, Fariborz; Katz, Benjamin B.; Li, Zeyang; Dai, Zhefu; Zhang, Zeyu; Zhang, Lei; Louie, Stan G.; Cherezov, Vadim; Zhang, Yong Share Save
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Structural diversity of leukotriene G-protein coupled receptors Luginina, Aleksandra; Gusach, Anastasiia; Lyapina, Elizaveta; Khorn, Polina; Safronova, Nadezda; Shevtsov, Mikhail; Dmitirieva, Daria; Dashevskii, Dmitrii; Kotova, Tatiana; Smirnova, Ekaterina; Borshchevskiy, Valentin; Cherezov, Vadim; Mishin, Alexey Share Save
Structural insights into angiotensin receptor signaling modulation by balanced and biased agonists Zhang, Dongqi; Liu, Yongfeng; Zaidi, Saheem A.; Xu, Lingyi; Zhan, Yuting; Chen, Anqi; Guo, Jiangtao; Huang, Xi-Ping; Roth, Bryan L.; Katritch, Vsevolod; Cherezov, Vadim; Zhang, Haitao Share Save
Sub-millisecond conformational dynamics of the A2A adenosine receptor revealed by single-molecule FRET Maslov, Ivan; Volkov, Oleksandr; Khorn, Polina; Orekhov, Philipp; Gusach, Anastasiia; Kuzmichev, Pavel; Gerasimov, Andrey; Luginina, Aleksandra; Coucke, Quinten; Bogorodskiy, Andrey; Gordeliy, Valentin; Wanninger, Simon; Barth, Anders; Mishin, Alexey; Hofkens, Johan; Cherezov, Vadim; Gensch, Thomas; Hendrix, Jelle; Borshchevskiy, Valentin Share Save
The activation mechanism and antibody binding mode for orphan GPR20 Lin, Xi; Jiang, Shan; Wu, Yiran; Wei, Xiaohu; Han, Gye-Won; Wu, Lijie; Liu, Junlin; Chen, Bo; Zhang, Zhibin; Zhao, Suwen; Cherezov, Vadim; Xu, Fei Share Save
High ligand efficiency quinazoline compounds as novel A2A adenosine receptor antagonists Bolteau, Raphael; Duroux, Romain; Laversin, Amelie; Vreulz, Brandon; Shiriaeva, Anna; Stauch, Benjamin; Han, Gye Won; Cherezov, Vadim; Renault, Nicolas; Barczyk, Amelie; Ravez, Severine; Coevoet, Mathilde; Melnyk, Patricia; Liberelle, Maxime; Yous, Said Share Save
GPCR Agonist-to-Antagonist Conversion: Enabling the Design of Nucleoside Functional Switches for the A2A Adenosine Receptor Shiriaeva, Anna; Park, Daejin; Kim, Gyudong; Lee, Yoonji; Hou, Xiyan; Jarhad, Dnyandev B.; Kim, Gibae; Yu, Jinha; Hyun, Young Eum; Kim, Woomi; Gao, Zhan-Guo; Jacobson, Kenneth A.; Han, Gye Won; Stevens, Raymond C.; Jeong, Lak Shin; Choi, Sun; Cherezov, Vadim Share Save
Structural basis for receptor selectivity and inverse agonism in S1P5 receptors Lyapina, Elizaveta; Marin, Egor; Gusach, Anastasiia; Orekhov, Philipp; Gerasimov, Andrey; Luginina, Aleksandra; Vakhrameev, Daniil; Ergasheva, Margarita; Kovaleva, Margarita; Khusainov, Georgii; Khorn, Polina; Shevtsov, Mikhail; Kovalev, Kirill; Bukhdruker, Sergey; Okhrimenko, Ivan; Popov, Petr; Hu, Hao; Weierstall, Uwe; Liu, Wei; Cho, Yunje; Gushchin, Ivan; Rogachev, Andrey; Bourenkov, Gleb; Park, Sehan; Park, Gisu; Hyun, Hyo Jung; Park, Jaehyun; Gordeliy, Valentin; Borshchevskiy, Valentin; Mishin, Alexey; Cherezov, Vadim Share Save
Inhibition of the angiotensin II type 2 receptor AT2R is a novel therapeutic strategy for glioblastoma Perryman, Richard; Renziehausen, Alexander; Shaye, Hamidreza; Kostagianni, Androniki D.; Tsiailanis, Antonis D.; Thorne, Thomas; Chatziathanasiadou, Maria, V; Sivolapenko, Gregory B.; El Mubarak, Mohamed Ahmed; Han, Gye Won; Zarzycka, Barbara; Katritch, Vsevolod; Lebon, Guillaume; Lo Nigro, Cristiana; Lattanzio, Laura; Morse, Sophie, V; Choi, James J.; O'Neill, Kevin; Kanaki, Zoi; Klinakis, Apostolos; Crook, Tim; Cherezov, Vadim; Tzakos, Andreas G.; Syed, Nelofer Share Save
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Molecular basis for lipid recognition by the prostaglandin D2 receptor CRTH2 Liu, Heng; Deepak, R. N. V. Krishna; Shiriaeva, Anna; Gati, Cornelius; Batyuk, Alexander; Hu, Hao; Weierstall, Uwe; Liu, Wei; Wang, Lei; Cherezov, Vadim; Fan, Hao; Zhang, Cheng Share Save