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Alessio Ciulli

University of Dundee

59H-index
305Paper Count
1.4WCitation Count
Published Papers 129
Publication Date
Linkerology in PROTACs: learnings for proximity-inducing therapeutics
err2026-07-31
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errOAAI
errRubén Prieto-Díaz; Aina Urbina; María Rodríguez-Ríos; Alessio Ciulli
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Induced ubiquitination of the partially disordered estrogen receptor alpha via a 14-3-3 directed molecular glue-PROTAC
err2026-07-15
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errOAAI
errCarlo J. A. Verhoef; Charlotte Crowe; Mark A. Nakasone; Aitana DeLaCuadra-Basté; Tessa Harzing; Naomi A. S. Span; Gajanan Sathe; Laura C. Demmers; Kentaro Iso; Christian Ottmann; Luc Brunsveld; Alessio Ciulli; Peter J. Cossar
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Targeted Protein Degradation of NUDT5 Dissociates Catalytic Inhibition from Protein Loss in 6-Thioguanine Response
err2026-06-30
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errOAAI
errAnne-Sophie M. C. Marques; Ludwig G. Bauer; Tuan-Anh Nguyen; Alejandro Gonzalez Orta; Jan-Lennart Venne; Carol Cheng; Esra Balıkçı; Yusi Liu; Barr Tivon; Alena Kroupova; Alessio Ciulli; Nir London; Stefan Kubicek; Kilian V. M. Huber
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The benchmarking and application of tag-degraders in vivo to validate therapeutic targets
err2026-05-29
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errOAAI
errCharlene M. Magtoto; Stephen Mieruszynski; Hao Dong; Ashley P. Ng; Ladina Di Rago; Andrew J. Kueh; Martin Brzozowski; Christoph Grohmann; Joel R. Walker; Ngee Kiat Chua; Laura F. Dagley; Alessio Ciulli; Guillaume Lessene; Marco J. Herold; Joan K. Heath; John Silke; Rebecca Feltham
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BromoCatch: a self-labelling tag platform for protein modification and live cell imaging
err2026-05-13
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errOAAI
errMaria Rodriguez-Rios; Conner Craigon; Mark A. Nakasone; Gajanan Sathe; Adam G. Bond; Mark Dorward; Anthony K. Edmonds; Mark C. Norley; Robert E. Arnold; Paul M. Wood; Stephen J. Reynolds; Joel O. Cresser-Brown; Graham P. Marsh; Hannah J. Maple; Alessio Ciulli
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Dual E3 ligase recruitment by monovalent degraders for tunable SMARCA 2/4 degradation
err2026-05-01
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PREAI
errSpiteri, Valentina A.; Segal, Dmitri; Correa-Saez, Alejandro; Iso, Kentaro; Casement, Ryan; Munoz I Ordono, Miquel; Nakasone, Mark A.; Sathe, Gajanan; Schatz, Caroline; Peters, Hannah E.; Doward, Mark; Kainacher, Lisa; Cowan, Angus D.; Ciulli, Alessio; Winter, Georg E.
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Proximity Binding Assay for PROTAC Ternary Complex Analysis
err2026-04-21
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errOAAI
errIrene Ponzo; Alice Soldà; Charlotte Crowe; Göran Dahl; Tereza Jahodová; Andreas Heerwig; Stefan Geschwindner; Alessio Ciulli; Ulrich Rant
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High-throughput ligand diversification to discover chemical inducers of proximity
err2026-02-16
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errOAAI
errJames B. Shaum; Miquel Muñoz i Ordoño; Erica A. Steen; Daniela V. Wenge; Hakyung Cheong; Jordan Janowski; Moritz Hunkeler; Eric M. Bilotta; Zoe J. Rutter; Paige A. Barta; Abby M. Thornhill; Natalia Milosevich; Lauren M. Hargis; Timothy R. Bishop; Trever R. Carter; Bryce da Camara; Matthias Hinterndorfer; Lucas Dada; Wen-Ji He; Fabian Offensperger; Hirotake Furihata; Sydney R. Schweber; Charlie Hatton; Yanhe Wen; Benjamin F. Cravatt; Keary M. Engle; Katherine A. Donovan; Bruno Melillo; Seiya Kitamura; Alessio Ciulli; Scott A. Armstrong; Eric S. Fischer; Georg E. Winter; Michael A. Erb
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Identification of a Highly Cooperative PROTAC Degrader Targeting GTP-Loaded KRAS(On) Alleles
err2025-10-30
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errOAAI
errVesna Vetma; Ilaria Puoti; Natalia K. Karolak; Sohini Chakraborti; Emelyne Diers; Enrico Girardi; Shakil Khan; Giorgia Kidd; Katrin G. Kropatsch; Ross Mclennan; Suzanne O’Connor; Matthias Samwer; Nicole Trainor; Claire Whitworth; Andre J. Wijaya; Jeff Y. F. Wong; David Zollman; William Farnaby; Johannes Popow; Alessio Ciulli; Peter Ettmayer; Kirsten McAulay
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Mode of action of a DCAF16-recruiting targeted glue that can selectively degrade BRD9
err2025-10-27
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errOAAI
errScott J. Hughes; Wojciech J. Stec; Colin T. R. Davies; David McGarry; Alicia Williams; Marta Carrara; Ivan Del Barco Barrantes; Rebecca Harris; Anna Tasegian; Dominic D. G. Owens; Alexander Fawcett; John Hellicar; Aleksandra Azevedo; Gregor P. Meier; Andrew C. Runcie; Liliana Greger; Martin O’Rourke; Ian Churcher; Martin Pass; Giles A. Brown; Alessio Ciulli; Louise K. Modis; Andrea Testa
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Opportunities in proximity modulation: Bridging academia and industry
err2025-08-21
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errOAAI
errIvan Dikic; Cristina Mayor-Ruiz; Georg E. Winter; Kerstin Koch; Alessio Ciulli; Nicolas H. Thomä
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A method for the detection and enrichment of endogenous cereblon substrates
err2025-08-08
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errOAAI
errHannah C. Lloyd; Yuli Li; N. Connor Payne; Zhenguang Zhao; Wenqing Xu; Alena Kroupova; David Zollman; Tengfang Long; Farah Kabir; Mei Chen; Rebecca Freeman; Ethan Yang Feng; Sarah Y. Xi; Ya-Chieh Hsu; Alessio Ciulli; Ralph Mazitschek; Christina M. Woo
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Targeted protein degradation for cancer therapy
err2025-04-25
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PREAI
errHinterndorfer, Matthias; Spiteri, Valentina A.; Ciulli, Alessio; Winter, Georg E.
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Loss of Socs2 improves molecular responses to IFNα in a mouse model of myeloproliferative neoplasms driven by JAK2-V617F
errLEUKEMIA
IF13.4
err2025-03-11
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PREAI
errUsart, Marc; Kimmerlin, Quentin; Stetka, Jan; Stoll, Cedric; Rai, Shivam; Fonseca, Tiago Almeida; Karjalainen, Riikka; Hao-Shen, Hui; Roux, Julien; El Taher, Athimed; Lynch, Dylan; Makukhin, Nikolai; Ciulli, Alessio; Skoda, Radek C.
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The efflux pump ABCC1/MRP1 constitutively restricts PROTAC sensitivity in cancer cells
err2025-02-01
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errOAAI
errWolf, Gernot; Craigon, Conner; Teoh, Shao Thing; Essletzbichler, Patrick; Onstein, Svenja; Cassidy, Diane; Uijttewaal, Esther C. H.; Dvorak, Vojtech; Cao, Yuting; Bensimon, Ariel; Elling, Ulrich; Ciulli, Alessio; Superti-Furga, Giulio
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Use of Aldehyde-Alkyne-Amine Couplings to Generate Medicinal Chemistry-Relevant Linkers
err2025-01-25
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errOAAI
errMcgown, Andrew; Vetma, Vesna; Crepin, Damien; Lin, Yan; Adcock, Claire; Craigon, Conner; Nafie, Jordan; von Emloh, Daniel; Sutton, Lea; Bailey, Kiera; Edmunds, Lewis; Sharma, Manvendra; Wilden, Jonathan D.; Coles, Simon J.; Tizzard, Graham J.; Farnaby, William; Ciulli, Alessio; Kostakis, George E.; Spencer, John
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