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Michael J. Waring

newcastle university - uk

65H-index
406Paper Count
1.9WCitation Count
Published Papers 83
Publication Date
Covalent Alkynylpyridopyrimidinones Targeting Cysteine 775 of the Epidermal Growth Factor Receptor Overcome Resistance to Current Therapies
err2025-12-01
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PREAI
errStewart, Hannah L.; Bordoni, Cinzia; Jennings, Claire E.; Al-Khawaldeh, Islam; Martin, Mathew P.; Noble, Richard A.; Phillips, Nicole; Pintar, Sara; Prendergast, Lisa; Thomas, Huw D.; Wang, Lan-Z.; Watt, Jessica E.; Wittner, Anita; Bronowska, Agnieszka K.; Cano, Celine; Noble, Martin E. M.; Wedge, Stephen R.; Waring, Michael J.
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Design and synthesis of a chemically diverse; lead-like DNA-encoded library from sequential amide coupling
err2025-08-22
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errOAAI
errCameron E. Taylor; Grace Roper; Rhianna Young; Fredrik Svensson; Andreas Brunschweiger; Sam Butterworth; Andrew G. Leach; Michael J. Waring
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Improvements in micelle promoted DNA-encoded library synthesis by surfactant optimisation
err2025-08-17
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errOAAI
errJake A. Odger; Matthew J. Anderson; Thomas P. Carton; Bao Nguyen; Kevin Foote; Michael J. Waring
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Crystallographic fragment screening of CDK2-cyclin A: FragLites map sites of protein-protein interaction
err2025-08-14
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PREAI
errIan Hope; Mathew P. Martin; Ziwei Jiang; Michael J. Waring; Martin E.M. Noble; Jane A. Endicott; Natalie J. Tatum
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Factors affecting irreversible inhibition of EGFR and influence of chirality on covalent binding (vol 8, 111, 2025)
err2025-05-19
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errOAAI
errMorese, Pasquale A.; Ahmad, Ayaz; Martin, Mathew P.; Noble, Richard A.; Pintar, Sara; Wang, Lan Z.; Xu, Shangze; Lister, Andrew; Ward, Richard A.; Bronowska, Agnieszka K.; Noble, Martin E. M.; Stewart, Hannah L.; Waring, Michael J.
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Factors affecting irreversible inhibition of EGFR and influence of chirality on covalent binding
err2025-04-09
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errOAAI
errMorese, Pasquale A.; Ahmad, Ayaz; Martin, Mathew P.; Noble, Richard A.; Pintar, Sara; Wang, Lan Z.; Xu, Shangze; Lister, Andrew; Ward, Richard A.; Bronowska, Agnieszka K.; Noble, Martin E. M.; Stewart, Hannah L.; Waring, Michael J.
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Micelle-Promoted Reductive Amination of DNA-Conjugated Amines for DNA-Encoded Library Synthesis
err2024-02-21
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errOAAI
errAnderson, Matthew J.; Carton, Thomas P.; Salvini, Catherine L. A.; Crawford, James J.; Pairaudeau, Garry; Waring, Michael J.
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An analysis of the physicochemical properties of oral drugs from 2000 to 2022
err2024-01-01
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errOAAI
errPirie, Rachael; Stanway-Gordon, Harriet A.; Stewart, Hannah L.; Wilson, Kirsty L.; Patton, Summer; Tyerman, Jack; Cole, Daniel J.; Fowler, Katherine; Waring, Michael J.
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Targeting Cytotoxic Agents through EGFR-Mediated Covalent Binding and Release
err2023-08-30
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errOAAI
errMorese, Pasquale A.; Anthony, Nahoum; Bodnarchuk, Michael; Jennings, Claire; Martin, Mathew P.; Noble, Richard A.; Phillips, Nicole; Thomas, Huw D.; Wang, Lan Z.; Lister, Andrew; Noble, Martin E. M.; Ward, Richard A.; Wedge, Stephen R.; Stewart, Hannah L.; Waring, Michael J.
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Conformational study into N-alkyl-N0.625pt′-aryl ureas to inform drug discovery
err2023-08-01
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errOAAI
errStewart, Hannah L.; Bon, Marta; Wills, Corinne; Martin, Mathew P.; Wang, Lan Z.; Mackenzie, Eilidh S.; Waddell, Paul G.; Waring, Michael J.
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Micelle-Mediated Sonogashira Coupling for DNA-Encoded Library Synthesis
err2023-06-16
err3
errOAAI
errGraham, Jessica S.; Stanway-Gordon, Harriet A.; Waring, Michael J.
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Development of a Micellar-Promoted Heck Reaction for the Synthesis of DNA-Encoded Libraries
err2023-03-08
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errOAAI
errStanway-Gordon, Harriet A.; Odger, Jake A.; Waring, Michael J.
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Fragment expansion with NUDELs - poised DNA-encoded libraries
err2023-01-01
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errOAAI
errSalvini, Catherine L. A.; Darlot, Benoit; Davison, Jack; Martin, Mathew P.; Tudhope, Susan J.; Turberville, Shannon; Kawamura, Akane; Noble, Martin E. M.; Wedge, Stephen R.; Crawford, James J.; Waring, Michael J.
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Mapping Ligand Interactions of Bromodomains BRD4 and ATAD2 with FragLites and PepLites_ Halogenated Probes of Druglike and Peptide-like Molecular Interactions
err2022-11-11
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errOAAI
errDavison, Gemma; Martin, Mathew P.; Turberville, Shannon; Dormen, Selma; Heath, Richard; Heptinstall, Amy B.; Lawson, Marie; Miller, Duncan C.; Ng, Yi Min; Sanderson, James N.; Hope, Ian; Wood, Daniel J.; Cano, Celine; Endicott, Jane A.; Hardcastle, Ian R.; Noble, Martin E. M.; Waring, Michael J.
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Build-Couple-Transform: A Paradigm for Lead-like Library Synthesis with Scaffold Diversity
err2022-08-09
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errOAAI
errUguen, Melanie; Davison, Gemma; Sprenger, Lukas J.; Hunter, James H.; Martin, Mathew P.; Turberville, Shannon; Watt, Jessica E.; Golding, Bernard T.; Noble, Martin E. M.; Stewart, Hannah L.; Waring, Michael J.
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Parallel Optimization of Potency and Pharmacokinetics Leading to the Discovery of a Pyrrole Carboxamide ERK5 Kinase Domain Inhibitor
err2022-04-25
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errOAAI
errMiller, Duncan C.; Reuillon, Tristan; Molyneux, Lauren; Blackburn, Timothy; Cook, Simon J.; Edwards, Noel; Endicott, Jane A.; Golding, Bernard T.; Griffin, Roger J.; Hardcastle, Ian; Harnor, Suzannah J.; Heptinstall, Amy; Lochhead, Pamela; Martin, Mathew P.; Martin, Nick C.; Myers, Stephanie; Newell, David R.; Noble, Richard A.; Phillips, Nicole; Rigoreau, Laurent; Thomas, Huw; Tucker, Julie A.; Wang, Lan-Zhen; Waring, Michael J.; Wong, Ai-Ching; Wedge, Stephen R.; Noble, Martin E. M.; Cano, Celine
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Identification and optimization of a novel series of selective PIP5K inhibitors
err2022-01-01
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errOAAI
errAndrews, David M.; Cartic, Sharon; Cosulich, Sabina; Divecha, Nullin; Faulder, Paul; Flemington, Vikki; Kern, Oliver; Kettle, Jason G.; MacDonald, Ellen; McKelvie, Jennifer; Pike, Kurt G.; Roberts, Bryan; Rowlinson, Rachel; Smith, James M.; Stockley, Martin; Swarbrick, Martin E.; Treinies, Iris; Waring, Michael J.
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Functional Group Tolerance of a Micellar on-DNA Suzuki-Miyaura Cross-Coupling Reaction for DNA-Encoded Library Design
err2021-11-24
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errOAAI
errHunter, James H.; Potowski, Marco; Stanway-Gordon, Harriet A.; Madin, Andrew; Pairaudeau, Garry; Brunschweiger, Andreas; Waring, Michael J.
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