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DIFFUSE MIDLINE GLIOMA, H3 K27 AND BRAF/FGFR1 CO-ALTERED: DISTINCT BIOLOGY AND THERAPEUTIC OPPORTUNITIES Auffret, L.; Barry, C.; Ajlil, Y.; Tauziede-Espariat, A.; Simbozel, M.; Mayr, L.; Kergorhen, T.; Puiseux, C.; Riffaud, L.; Blouin, P.; Bertozzi, A.; Leblond, P.; Blomgren, K.; Froelich, S.; Picca, A.; Touat, M.; Sanson, M.; Beccaria, K.; Blauwblomme, T.; Dangouloff-Ros, V; Boddaert, N.; Gojo, J.; Filbin, M.; Varlet, P.; Debily, M.; Grill, J.; Castel, D. Share Save
The Kinetics of Bedaquiline Diffusion in Tuberculous Cavities Open a Window for the Emergence of Resistance Bustion, Annamarie E.; Ernest, Jacqueline P.; Kaya, Firat; Silva, Connie; Sarathy, Jansy; Blanc, Landry; Imperial, Marjorie; Gengenbacher, Martin; Xie, Min; Zimmerman, Matthew D.; Robertson, Gregory T.; Weiner, Danielle; Via, Laura E.; Barry, Clifton E.; Savic, Radojka M.; Dartois, Veronique Share Save
Identification of a Series Containing a Pentafluorophenyl Moiety That Targets Pks13 to Inhibit Growth of Mycobacterium tuberculosis Green, SR; Harrison, JR; Thompson, S; Murugesan, D; Libardo, MDJ; Engelhart, CA; Meshanni, J; Fletcher, D; Scullion, P; Edwards, D; Epemolu, O; Mutter, N; Shishikura, Y; Riley, J; Ioerger, TR; Guillén, JJR; López, LG; Read, KD; Barry, CE III; Schnappinger, D; Wyatt, PG; Boshoff, HIM; Cleghorn, LAT Share Save
Distributable, metabolic PET reporting of tuberculosis Khan, R. M. Naseer; Ahn, Yong-Mo; Marriner, Gwendolyn A.; Via, Laura E.; D'Hooge, Francois; Lee, Seung Seo; Yang, Nan; Basuli, Falguni; White, Alexander G.; Tomko, Jaime A.; Frye, L. James; Scanga, Charles A.; Weiner, Danielle M.; Sutphen, Michelle L.; Schimel, Daniel M.; Dayao, Emmanuel; Piazza, Michaela K.; Gomez, Felipe; Dieckmann, William; Herscovitch, Peter; Mason, N. Scott; Swenson, Rolf; Kiesewetter, Dale O.; Backus, Keriann M.; Geng, Yiqun; Raj, Ritu; Anthony, Daniel C.; Flynn, JoAnne L.; Barry III, Clifton E.; Davis, Benjamin G. Share Save
Mtb-Selective 5-Aminomethyl Oxazolidinone Prodrugs: Robust Potency and Potential Liabilities Boshoff, Helena I. M.; Young, Katherine; Ahn, Yong-Mo; Yadav, Veena D.; Crowley, Brendan M.; Yang, Lihu; Su, Jing; Oh, Sangmi; Arora, Kriti; Andrews, Jenna; Manikkam, Michelle; Sutphin, Michelle; Smith, Anthony J.; Weiner, Danielle M.; Piazza, Michaela K.; Fleegle, Joel D.; Gomez, Felipe; Dayao, Emmannual K.; Prideaux, Brendan; Zimmerman, Matthew; Kaya, Firat; Sarathy, Jansy; Tan, Vee Yang; Via, Laura E.; Tschirret-Guth, Richard; Lenaerts, Anne J.; Robertson, Gregory T.; Dartois, Veronique; Olsen, David B.; Barry III, Clifton E. Share Save
Normalizing granuloma vasculature and matrix improves drug delivery and reduces bacterial burden in tuberculosis- infected rabbits Datta, Meenal; Via, Laura E.; Dartois, Veronique; Weiner, Danielle M.; Zimmerman, Matthew; Kaya, Firat; Walker, April M.; Fleegle, Joel D.; Raplee, Isaac D.; Mcninch, Colton; Zarodniuk, Maksym; Kamoun, Walid S.; Yue, Changli; Kumar, Ashwin S.; Subudhi, Sonu; Xu, Lei; Barry, Clifton E.; Jain, Rakesh K. Share Save
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A first-in-class leucyl-tRNA synthetase inhibitor, ganfeborole, for rifampicin-susceptible tuberculosis: a phase 2a open-label, randomized trial Diacon, Andreas H.; Barry, Clifton E., III; Carlton, Alex; Chen, Ray Y.; Davies, Matt; de Jager, Veronique; Fletcher, Kim; Koh, Gavin C. K. W.; Kontsevaya, Irina; Heyckendorf, Jan; Lange, Christoph; Reimann, Maja; Penman, Sophie L.; Scott, Rhona; Maher-Edwards, Gareth; Tiberi, Simon; Vlasakakis, Georgios; Upton, Caryn M.; Aguirre, David Barros Share Save
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A Novel Tool to Identify Bactericidal Compounds against Vulnerable Targets in Drug-Tolerant M. tuberculosis found in Caseum Sarathy, Jansy P.; Xie, Min; Jones, Richard M.; Chang, Adrienne; Osiecki, Paulina; Weiner, Danielle; Tsao, Wen-Shan; Dougher, Maureen; Blanc, Landry; Fotouhi, Nader; Via, Laura E.; Barry III, Clifton E.; De Vlaminck, Iwijn; Sherman, David R.; Dartois, Veronique A. Share Save
The Myxobacterial Antibiotic Myxovalargin: Biosynthesis, Structural Revision, Total Synthesis, and Molecular Characterization of Ribosomal Inhibition Koller, Timm O.; Scheid, Ullrich; Koesel, Teresa; Herrmann, Jennifer; Krug, Daniel; Boshoff, Helena I. M.; Beckert, Bertrand; Evans, Joanna C.; Schlemmer, Jan; Sloan, Becky; Weiner, Danielle M.; Via, Laura E.; Moosa, Atica; Ioerger, Thomas R.; Graf, Michael; Zinshteyn, Boris; Abdelshahid, Maha; Nguyen, Fabian; Arenz, Stefan; Gille, Franziska; Siebke, Maik; Seedorf, Tim; Plettenburg, Oliver; Green, Rachel; Warnke, Anna-Luisa; Ullrich, Joachim; Warrass, Ralf; Barry, Clifton E., III; Warner, Digby F.; Mizrahi, Valerie; Kirschning, Andreas; Wilson, Daniel N.; Mueller, Rolf Share Save
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Phylogenomic analysis of the diversity of graspetides and proteins involved in their biosynthesis Makarova, Kira S.; Blackburne, Brittney; Wolf, Yuri, I; Nikolskaya, Anastasia; Karamycheva, Svetlana; Espinoza, Marlene; Barry, Clifton E., III; Bewley, Carole A.; Koonin, Eugene, V Share Save
A Rabbit Model to Study Antibiotic Penetration at the Site of Infection for Nontuberculous Mycobacterial Lung Disease: Macrolide Case Study Kaya, Firat; Ernest, Jacqueline P.; LoMauro, Katherine; Gengenbacher, Martin; Madani, Abdeldjalil; Aragaw, Wassihun Wedajo; Zimmerman, Matthew D.; Sarathy, Jansy P.; Alvarez, Nadine; Daudelin, Isaac; Wang, Han; Lanni, Faye; Weiner, Danielle M.; Via, Laura E.; Barry, Clifton E.; Olivier, Kenneth N.; Dick, Thomas; Podell, Brendan K.; Savic, Radojka M.; Dartois, Veronique Share Save
Identification of β-Lactams Active against Mycobacterium tuberculosis by a Consortium of Pharmaceutical Companies and Academic Institutions Gold, Ben; Zhang, Jun; Quezada, Landys Lopez; Roberts, Julia; Ling, Yan; Wood, Madeleine; Shinwari, Wasima; Goullieux, Laurent; Roubert, Christine; Fraisse, Laurent; Bacque, Eric; Lagrange, Sophie; Filoche-Romme, Bruno; Vieth, Michal; Hipskind, Philip A.; Jungheim, Louis N.; Aube, Jeffrey; Scarry, Sarah M.; McDonald, Stacey L.; Li, Kelin; Perkowski, Andrew; Nguyen, Quyen; Dartois, Veronique; Zimmerman, Matthew; Olsen, David B.; Young, Katherine; Bonnett, Shilah; Joerss, Douglas; Parish, Tanya; Boshoff, Helena, I; Arora, Kriti; Barry, Clifton E., III; Guijarro, Laura; Anca, Sara; Rullas, Joaquin; Rodriguez-Salguero, Beatriz; Martinez-Martinez, Maria S.; Porras-De Francisco, Esther; Cacho, Monica; Barros-Aguirre, David; Smith, Paul; Berthel, Steven J.; Nathan, Carl; Bates, Robert H. Share Save