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Michel O. Steinmetz

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82H-index
388Paper Count
2.3WCitation Count
Published Papers 156
Publication Date
An integrated experimental and computational pipeline for crystallographic fragment screening of membrane protein in the lipid cubic phase
err2026-05-13
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errOAAI
errChia-Ying Huang; Robert Cheng; Alexander Metz; Denis Bucher; Fabio Andres; Arianna Bacchin; Hannah Glover; Christoph P. Sager; Meitian Wang; Michel O. Steinmetz; Michael Hennig; May Sharpe
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Structural basis of microtubule-mediated signal transduction
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IF42.5
err2025-12-08
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errOAAI
errSung Ryul Choi; Thorsten B. Blum; Matteo Giono; Bibhas Roy; Ioannis Vakonakis; Dominic Schmid; Nicole Oelgarth; Apisha Ranganathan; Alvar D. Gossert; G.V. Shivashankar; Alfred Zippelius; Michel O. Steinmetz
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Asymmetric Total Synthesis of (−)-Glycybridin B, a Pharmacophore Screened Candidate for Tubulin Binding
err2025-08-06
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errOAAI
errDr. Alice Maiocchi; Dr. Maxim Shevelev; Dr. Zlata Boiarska; Dr. Juan Estévez-Gallego; Dr. Francesca Bonato; Dr. Paolo Orlando; Alessandra Chinosi; Emanuele Marcone; Dr. Andrea Citarella; Dr. Dragos Horvath; Prof. Dr. Michel O. Steinmetz; Dr. Andrea E. Prota; Dr. Alexandre Varnek; Dr. Valerio Fasano; Prof. Dr. Daniele Passarella
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Hydrolysis-deficient mosaic microtubules as faithful mimics of the GTP cap
err2025-03-10
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errOAAI
errEstevez-Gallego, Juan; Blum, Thorsten B.; Ruhnow, Felix; Gili, Maria; Speroni, Silvia; Garcia-Castellanos, Raquel; Steinmetz, Michel O.
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Centriolar cap proteins CP110 and CPAP control slow elongation of microtubule plus ends
err2025-01-23
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errOAAI
errIyer, Saishree S.; Chen, Fangrui; Ogunmolu, Funso E.; Moradi, Shoeib; Volkov, Vladimir A.; van Grinsven, Emma J.; van Hoorn, Chris; Wu, Jingchao; Andrea, Nemo; Hua, Shasha; Jiang, Kai; Vakonakis, Ioannis; Potocnjak, Mia; Herzog, Franz; Gigant, Benoit; Gudimchuk, Nikita; Stecker, Kelly E.; Dogterom, Marileen; Steinmetz, Michel O.; Akhmanova, Anna
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Bridging the maytansine and vinca sites: Cryptophycins target β-tubulin ' s T5-loop
err2024-06-01
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errOAAI
errAbel, Anne-Catherine; Muhlethaler, Tobias; Dessin, Cedric; Schachtsiek, Thomas; Sammet, Benedikt; Sharpe, Timothy; Steinmetz, Michel O.; Sewald, Norbert; Prota, Andrea E.
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The novel microtubule-destabilizing compound AUS_001 maintains unique binding to the colchicine site of tubulin and elicits reversible cellular effects relative to other anti-tubulin agents
err2024-03-22
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PREAI
errLelie, Herman; Chou, Yao-Chieh; King, Alastair J.; Boiarska, Zlata; Prota, Andrea E.; Steinmetz, Michel O.; Koutsioumpa, Marina
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Modular synthesis of functional libraries by accelerated SuFEx click chemistry
err2024-01-01
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errHomer, Joshua A.; Koelln, Rebecca A.; Barrow, Andrew S.; Gialelis, Timothy L.; Boiarska, Zlata; Steinohrt, Nikita S.; Lee, Erinna F.; Yang, Wen-Hsuan; Johnson, Robert M.; Chung, Taemoon; Habowski, Amber N.; Vishwakarma, Dharmendra S.; Bhunia, Debmalya; Avanzi, Charlotte; Moorhouse, Adam D.; Jackson, Mary; Tuveson, David A.; Lyons, Scott K.; Lukey, Michael J.; Fairlie, W. Douglas; Haider, Shozeb M.; Steinmetz, Michel O.; Prota, Andrea E.; Moses, John E.
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A photo-SAR study of photoswitchable azobenzene tubulin-inhibiting antimitotics identifying a general method for near-quantitative photocontrol
err2024-01-01
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errOAAI
errReynders, Martin; Garscia, Malgorzata; Mueller-Deku, Adrian; Wranik, Maximilian; Krauskopf, Kristina; de la Rosa, Luis de la Osa; Schaffer, Konstantin; Joetten, Anna; Rode, Alexander; Stierle, Valentin; Kraus, Yvonne; Baumgartner, Benedikt; Ali, Ahmed; Bubeneck, Andrei; Seal, Trina; Steinmetz, Michel O.; Paulitschke, Philipp; Thorn-Seshold, Oliver
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A multi-reservoir extruder for time-resolved serial protein crystallography and compound screening at X-ray free-electron lasers
err2023-12-02
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errWranik, Maximilian; Kepa, Michal W.; Beale, Emma V.; James, Daniel; Bertrand, Quentin; Weinert, Tobias; Furrer, Antonia; Glover, Hannah; Gashi, Dardan; Carrillo, Melissa; Kondo, Yasushi; Stipp, Robin T.; Khusainov, Georgii; Nass, Karol; Ozerov, Dmitry; Cirelli, Claudio; Johnson, Philip J. M.; Dworkowski, Florian; Beale, John H.; Stubbs, Scott; Zamofing, Thierry; Schneider, Marco; Krauskopf, Kristina; Gao, Li; Thorn-Seshold, Oliver; Bostedt, Christoph; Bacellar, Camila; Steinmetz, Michel O.; Milne, Christopher; Standfuss, Jorg
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The motor domain of the kinesin Kip2 promotes microtubule polymerization at microtubule tips
err2023-04-24
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errChen, Xiuzhen; Portran, Didier; Widmer, Lukas A. A.; Stangier, Marcel M. M.; Czub, Mateusz P. P.; Liakopoulos, Dimitris; Stelling, Jorg; Steinmetz, Michel O. O.; Barral, Yves
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Structural insight into the stabilization of microtubules by taxanes
err2023-03-06
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errProta, Andrea E.; Lucena-Agell, Daniel; Ma, Yuntao; Estevez-Gallego, Juan; Li, Shuo; Bargsten, Katja; Josa-Prado, Fernando; Altmann, Karl-Heinz; Gaillard, Natacha; Kamimura, Shinji; Muhlethaler, Tobias; Gago, Federico; Oliva, Maria A.; Steinmetz, Michel O.; Fang, Wei-Shuo; Diaz, J. Fernando
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Watching the release of a photopharmacological drug from tubulin using time-resolved serial crystallography
err2023-02-17
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errOAAI
errWranik, Maximilian; Weinert, Tobias; Slavov, Chavdar; Masini, Tiziana; Furrer, Antonia; Gaillard, Natacha; Gioia, Dario; Ferrarotti, Marco; James, Daniel; Glover, Hannah; Carrillo, Melissa; Kekilli, Demet; Stipp, Robin; Skopintsev, Petr; Brunle, Steffen; Muhlethaler, Tobias; Beale, John; Gashi, Dardan; Nass, Karol; Ozerov, Dmitry; Johnson, Philip J. M.; Cirelli, Claudio; Bacellar, Camila; Braun, Markus; Wang, Meitian; Dworkowski, Florian; Milne, Chris; Cavalli, Andrea; Wachtveitl, Josef; Steinmetz, Michel O. O.; Standfuss, Jorg
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Multivalency ensures persistence of a plus TIP body at specialized microtubule ends
err2022-12-19
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errMeier, Sandro M.; Farcas, Ana-Maria; Kumar, Anil; Ijavi, Mahdiye; Bill, Robert T.; Stelling, Joerg; Dufresne, Eric R.; Steinmetz, Michel O.; Barral, Yves
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VASH1-SVBP and VASH2-SVBP generate different detyrosination profiles on microtubules
err2022-12-13
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errOAAI
errRamirez-Rios, Sacnicte; Choi, Sung Ryul; Sanyal, Chadni; Blum, Thorsten B. B.; Bosc, Christophe; Krichen, Fatma; Denarier, Eric; Soleilhac, Jean-Marc; Blot, Beatrice; Janke, Carsten; Stoppin-Mellet, Virginie; Magiera, Maria M. M.; Arnal, Isabelle; Steinmetz, Michel O. O.; Moutin, Marie-Jo
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Changes in seam number and location induce holes within microtubules assembled from porcine brain tubulin and in Xenopus egg cytoplasmic extracts
err2022-12-12
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errOAAI
errGuyomar, Charlotte; Bousquet, Clement; Ku, Siou; Heumann, John M.; Guilloux, Gabriel; Gaillard, Natacha; Heichette, Claire; Duchesne, Laurence; Steinmetz, Michel O.; Gibeaux, Romain; Chretien, Denis; Welburn, Julie P., I
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Development of [1,2]oxazoloisoindoles tubulin polymerization inhibitors: Further chemical modifications and potential therapeutic effects against lymphomas
err2022-12-01
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PREAI
errBarreca, Marilia; Span, Virginia; Rocca, Roberta; Bivacqua, Roberta; Abel, Anne -Catherine; Maruca, Annalisa; Montalbano, Alessandra; Raimondi, Maria Valeria; Tarantelli, Chiara; Gaudio, Eugenio; Cascione, Luciano; Rinaldi, Andrea; Bai, Ruoli; Steinmetz, Michel O.; Prota, Andrea E.; Alcaro, Stefano; Hamel, Ernest; Bertoni, Francesco; Barraja, Paola
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Novel fragment-derived colchicine-site binders as microtubule-destabilizing agents
err2022-11-01
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errde la Roche, Noelia Montel; Muehlethaler, Tobias; Di Martino, Rita Maria Concetta; Ortega, Jose Antonio; Gioia, Dario; Roy, Bibhas; Prota, Andrea E.; Steinmetz, Michel O.; Cavalli, Andrea
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Rational Design of a Novel Tubulin Inhibitor with a Unique Mechanism of Action
err2022-04-25
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errOAAI
errMuhlethaler, Tobias; Milanos, Lampros; Ortega, Jose Antonio; Blum, Thorsten B.; Gioia, Dario; Roy, Bibhas; Prota, Andrea E.; Cavalli, Andrea; Steinmetz, Michel O.
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