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J

John H. Bushweller

university of virginia

50H-index
193Paper Count
9.1KCitation Count
Published Papers 48
Publication Date
The MLLT3 YEATS domain binds histone marks (H3K9/18/27ac/cr) and ncRNA (7SK), linking transcription and RNA signaling to regulate hematopoiesis
err2026-06-09
err0
errOAAI
errAdam Boulton; Ashish Kabra; Nicholas Achille; Emmalee R. Adelman; Dimitrios G. Anastasakis; Felipe Beckedorff; Pradeep Kumar Reddy Cingaram; Devin G. Roller; Ying Zhang; Benjamin Leach; Daniel Gioeli; Ramin Shiekhattar; Akihiko Yokoyama; Markus Hafner; Maria Figueroa; Nancy Zeleznik-Le; John H. Bushweller
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FGFR2-RUNX2 activation: An unexplored therapeutic pathway in luminal breast cancer related to tumor progression
err2024-12-28
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PREAI
errRodriguez, Maria S.; Mahmoud, Yamil D.; Vanzulli, Silvia; Giulianelli, Sebastian; Spengler, Eunice; Vazquez, Paula Martinez; Burruchaga, Javier; Bushweller, John; Lamb, Caroline A.; Luthy, Isabel A.; Lanari, Claudia; Pinero, Cecilia Perez
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The co-receptor Neuropilin-1 enhances proliferation in inv(16) acute myeloid leukemia via VEGF signaling
errLEUKEMIA
IF13.4
err2024-11-21
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PREAI
errHegde, Mahesh; Ahmad, Mohd H.; Lazaro, Roger Mulet; Sugita, Mayumi; Li, Rui; Hu, Kai; Gebhard, Claudia; Guzman, Monica L.; Bushweller, John H.; Zhu, Lihua J.; Brehm, Michael; Wolfe, Scot A.; Delwel, Ruud; Castilla, Lucio H.
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RUNX2 inhibition alters PAX3::FOXO1 driven fusion-positive rhabdomyosarcoma cell state and growth
err2024-03-22
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PREAI
errMendes, Elizabeth A.; Chambers, Audrey L.; Weitzel, Samantha J.; Deel, Michael; Munshi, Aanandi; Counter, Christopher M.; Zimmerman, Seth; Bushweller, John; Linardic, Corinne M.
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N-MYC regulates cell survival via eIF4G1 in inv(16) acute myeloid leukemia
err2024-03-01
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errOAAI
errPeramangalam, Philomina Sona; Surapally, Sridevi; Veltri, Anthony J.; Zheng, Shikan; Burns, Robert; Zhu, Nan; Rao, Sridhar; Muller-Tidow, Carsten; Bushweller, John H.; Pulikkan, John A.
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Gene regulatory network analysis predicts cooperating transcription factor regulons required for FLT3-ITD+ AML growth
err2023-12-01
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errOAAI
errColeman, Daniel J. L.; Keane, Peter; Luque-Martin, Rosario; Chin, Paulynn S.; Blair, Helen; Ames, Luke; Kellaway, Sophie G.; Griffin, James; Holmes, Elizabeth; Potluri, Sandeep; Assi, Salam A.; Bushweller, John; Heidenreich, Olaf; Cockerill, Peter N.; Bonifer, Constanze
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Small-Molecule Inhibitors of the MLL1 CXXC Domain, an Epigenetic Reader of DNA Methylation
err2022-07-07
err9
errOAAI
errKalmode, Hanuman P.; Podsiadly, Izabella; Kabra, Ashish; Boulton, Adam; Reddy, Prabhakar; Gao, Yan; Li, Christopher; Bushweller, John H.
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KIX domain determines a selective tumor-promoting role for EP300 and its vulnerability in small cell lung cancer
err2022-02-18
err15
errOAAI
errKim, Kee-Beom; Kabra, Ashish; Kim, Dong-Wook; Xue, Yongming; Huang, Yuanjian; Hou, Pei-Chi; Zhou, Yunpeng; Miranda, Leilani J.; Park, Jae-Il; Shi, Xiaobing; Bender, Timothy P.; Bushweller, John H.; Park, Kwon-Sik
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Structure of the Complex of an Iminopyridinedione Protein Tyrosine Phosphatase 4A3 Phosphatase Inhibitor with Human Serum Albumin
err2020-12-01
err10
errOAAI
errCzub, Mateusz P.; Boulton, Adam M.; Rastelli, Ettore J.; Tasker, Nikhil R.; Maskrey, Taber S.; Blanco, Isabella K.; McQueeney, Kelley E.; Bushweller, John H.; Minor, Wladek; Wipf, Peter; Sharlow, Elizabeth R.; Lazo, John S.
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TNF-α signaling regulates RUNX1 function in endothelial cells
err2020-11-02
err35
errOAAI
errWhitmore, Hannah A. B.; Amarnani, Dhanesh; O'Hare, Michael; Delgado-Tirado, Santiago; Gonzalez-Buendia, Lucia; An, Miranda; Pedron, Julien; Bushweller, John H.; Arboleda-Velasquez, Joseph F.; Kim, Leo A.
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BCOR Binding to MLL-AF9 Is Essential for Leukemia via Altered EYA1, SIX, and MYC Activity
err2020-07-07
err17
errOAAI
errSchmidt, Charles R.; Achille, Nicholas J.; Kuntimaddi, Aravinda; Boulton, Adam M.; Leach, Benjamin, I; Zhang, Shubin; Zeleznik-Le, Nancy J.; Bushweller, John H.
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RUNX proteins desensitize multiple myeloma to lenalidomide via protecting IKZFs from degradation
errLEUKEMIA
IF13.4
err2019-02-13
err44
errOAAI
errZhou, Nan; Gutierrez-Uzquiza, Alvaro; Zheng, Xiang Yu; Chang, Renxu; Vogl, Dan T.; Garfall, Alfred L.; Bernabei, Luca; Saraf, Anita; Florens, Laurence; Washburn, Michael P.; Illendula, Anuradha; Bushweller, John H.; Busino, Luca
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Small Molecule Inhibitor of CBFβ-RUNX Binding for RUNX Transcription Factor Driven Cancers (vol 8, pg 117, 2016)
err2017-11-01
err0
errOAAI
errIllendula, Anuradha; Gilmour, Jane; Grembecka, Jolanta; Tirumala, Venkata Sesha Srimath; Boulton, Adam; Kuntimaddi, Aravinda; Schmidt, Charles; Wang, Lixin; Pulikkan, John A.; Zong, Hongliang; Parlak, Mahmut; Kuscu, Cem; Pickin, Anna; Zhou, Yunpeng; Gao, Yan; Mishra, Lauren; Adli, Mazhar; Castilla, Lucio H.; Rajewski, Roger A.; Janes, Kevin A.; Guzman, Monica L.; Bonifer, Constanze; Bushweller, John H.
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Bacillus anthracis Peptidoglycan Integrity Is Disrupted by the Chemokine CXCL10 through the FtsE/X Complex
err2017-04-27
err10
errOAAI
errMargulieux, Katie R.; Liebov, Benjamin K.; Tirumala, Venkata S. K. K. S.; Singh, Arpita; Bushweller, John H.; Nakamoto, Robert K.; Hughes, Molly A.
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Small Molecule Inhibitor of CBFβ-RUNX Binding for RUNX Transcription Factor Driven Cancers
err2016-06-01
err93
errOAAI
errIllendula, Anuradha; Gilmour, Jane; Grembecka, Jolanta; Tirumala, Venkata Sesha Srimath; Boulton, Adam; Kuntimaddi, Aravinda; Schmidt, Charles; Wang, Lixin; Pulikkan, John A.; Zong, Hongliang; Parlak, Mahmut; Kuscu, Cem; Pickin, Anna; Zhou, Yunpeng; Gao, Yan; Mishra, Lauren; Adli, Mazhar; Castilla, Lucio H.; Rajewski, Roger A.; Janes, Kevin A.; Guzman, Monica L.; Bonifer, Constanze; Bushweller, John H.
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MAPK/ERK2 phosphorylates ERG at serine 283 in leukemic cells and promotes stem cell signatures and cell proliferation
errLEUKEMIA
IF13.4
err2016-03-08
err20
errOAAI
errHuang, Y.; Thoms, J. A. I.; Tursky, M. L.; Knezevic, K.; Beck, D.; Chandrakanthan, V.; Suryani, S.; Olivier, J.; Boulton, A.; Glaros, E. N.; Thomas, S. R.; Lock, R. B.; MacKenzie, K. L.; Bushweller, J. H.; Wong, J. W. H.; Pimanda, J. E.
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Structural and Functional Basis of Alternative ESCRT-0 Protein Complexes
err2016-02-01
err0
errOAAI
errXiao, Shuyan; Zhao, Xiaolin; Xiong, Wen; Brannon, Mary K.; Fread, Kristen; Ellena, Jeffrey; Bushweller, John; Finkielstein, Carla V.; Armstrong, Geoffrey; Capelluto, Daniel G.
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