Not logged in The Concise Guide to PHARMACOLOGY 2025/26: G protein-coupled receptors Alexander, Stephen P. H.; Davenport, Anthony P.; Kelly, Eamonn; Gibb, Alasdair J.; Mathie, Alistair A.; Peach, Chloe J.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George R.; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bennett, Kirstie A.; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria A.; Bonaventure, Pascal; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Brown, Andrew J.; Burnstock, Geoffrey; Busnelli, Marta; Calo, Girolamo; Caruso, Vanni; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Christopoulos, Arthur; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dautzenberg, Frank M.; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Dubocovich, Margarita L.; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Forsman, Huamei Fu; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gbahou, Florence; Gerard, Craig; Gershengorn, Marvin; Glass, Michelle; Gloriam, David E.; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gruber, Christian; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hartman, Deborah S.; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Heitman, Laura; Herr, Deron R.; Hollenberg, Morley D.; Holliday, Nicholas D.; Holst, Birgitte; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; IJzerman, Adriaan P.; Inagami, Tadashi; Insel, Paul A.; Jacobson, Kenneth A.; Jacobson, Laura H.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kinsolving, Julia; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Laishram, Luxmichan; Langenhan, Tobias; Langmead, Christopher J.; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Leurs, Rob; Li, Xaria X.; Liebscher, Ines; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet J.; Malfacini, Davide; Manning, Maurice; Marangon, Davide; Martemyanov, Kirill; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Neubig, Richard R.; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Perry-Hauser, Nicole; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Qin, Helena Chengxue; Quinn, Mark; Raffaele, Stefano; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Buzon, Alejandro Romeral; Rondard, Philippe; Rosenkilde, Mette M.; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Scholz, Nicole; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Shukla, Arun K.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Smith, Nicola J.; Staeubert, Claudia; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David M.; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Verbalis, Joseph G.; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Wu, Huixian; Yang, Cheng; Yao, Chengcan; Ye, Richard D.; Zaidman, Nathan Share Save
The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors Alexander, Stephen P. H.; Christopoulos, Arthur; Davenport, Anthony P.; Kelly, Eamonn; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Burnstock, Geoffrey; Calo, Girolamo; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gerard, Craig; Gershengorn, Marvin; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Herr, Deron; Hollenberg, Morley D.; Holliday, Nicholas D.; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; Ijzerman, Adriaan P.; Inagami, Tadashi; Jacobson, Kenneth A.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Langenhan, Tobias; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Li, Xaria X.; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet; Malfacini, Davide; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Quinn, Mark; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Rondard, Philippe; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Yao, Chengcan; Ye, Richard D. Share Save
Design, synthesis and biological evaluation of novel orthosteric-allosteric ligands of the cannabinoid receptor type 2 (CB2R) Ferrisi, Rebecca; Gado, Francesca; Polini, Beatrice; Ricardi, Caterina; Mohamed, Kawthar A. A.; Stevenson, Lesley A. A.; Ortore, Gabriella; Rapposelli, Simona; Saccomanni, Giuseppe; Pertwee, Roger G. G.; Laprairie, Robert B. B.; Manera, Clementina; Chiellini, Grazia Share Save
Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: from Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands Gado, Francesca; Ferrisi, Rebecca; Polini, Beatrice; Mohamed, Kawthar A.; Ricardi, Caterina; Lucarini, Elena; Carpi, Sara; Domenichini, Federica; Stevenson, Lesley A.; Rapposelli, Simona; Saccomanni, Giuseppe; Nieri, Paola; Ortore, Gabriella; Pertwee, Roger G.; Ghelardini, Carla; Mannelli, Lorenzo Di Cesare; Chiellini, Grazia; Laprairie, Robert B.; Manera, Clementina Share Save
Osteogenic growth peptide is a potent anti-inflammatory and bone preserving hormone via cannabinoid receptor type 2 Raphael-Mizrahi, Bitya; Attar-Namdar, Malka; Chourasia, Mukesh; Cascio, Maria G.; Shurki, Avital; Tam, Joseph; Neuman, Moshe; Rimmerman, Neta; Vogel, Zvi; Shteyer, Arie; Pertwee, Roger G.; Zimmer, Andreas; Kogan, Natalya M.; Bab, Itai; Gabet, Yankel; Zaidi, Mone Share Save
Synthesis and In Vitro Characterization of Selective Cannabinoid CB2 Receptor Agonists: Biological Evaluation against Neuroblastoma Cancer Cells Gado, Francesca; Ferrisi, Rebecca; Di Somma, Sarah; Napolitano, Fabiana; Mohamed, Kawthar A.; Stevenson, Lesley A.; Rapposelli, Simona; Saccomanni, Giuseppe; Portella, Giuseppe; Pertwee, Roger G.; Laprairie, Robert B.; Malfitano, Anna Maria; Manera, Clementina Share Save
CB1 receptor binding sites for NAM and PAM: A first approach for studying, new n-butyl-diphenylcarboxamides as allosteric modulators Gado, Francesca; Ceni, Costanza; Ferrisi, Rebecca; Sbrana, Giulia; Stevenson, Lesley A.; Macchia, Marco; Pertwee, Roger G.; Bertini, Simone; Manera, Clementina; Ortore, Gabriella Share Save
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THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein-coupled receptors Alexander, Stephen P. H.; Christopoulos, Arthur; Davenport, Anthony P.; Kelly, Eamonn; Mathie, Alistair; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Pawson, Adam J.; Southan, Christopher; Davies, Jamie A.; Abbracchio, Maria Pia; Alexander, Wayne; Al-hosaini, Khaled; Baeck, Magnus; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria; Boulay, Francois; Bousquet, Corinne; Braeuner-Osborne, Hans; Burnstock, Geoffrey; Calo, Girolamo; Castano, Justo P.; Catt, KevinJ; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Csaba, Zsolt; Dahlgren, Claes; Dent, Gordon; Singh, Khuraijam Dhanachandra; Douglas, Steven D.; Dournaud, Pascal; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Fumagalli, Marta; Gainetdinov, Raul R.; de Gasparo, Marc; Gerard, Craig; Gershengorn, Marvin; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gregory, Karen J.; Gundlach, Andrew L.; Hamann, Joerg; Hanson, Julien; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Hollenberg, Morley D.; Holliday, Nicholas D.; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; IJzerman, Adriaan P.; Inagami, Tadashi; Jacobson, Kenneth A.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Langenhan, Tobias; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Li, Xaria X.; Williams, Tom Lloyd; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip; Nahon, Jean-Louis; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; Ocarroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Quinn, Mark; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Rondard, Philippe; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David; Thomas, Walter (Wally); Timmermans, PieterB M. W. M.; Tirupula, Kalyan; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Woodruff, Trent M.; Yao, Chengcan; Ye, Richard D. Share Save
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Discovery of a Biased Allosteric Modulator for Cannabinoid 1 Receptor: Preclinical Anti-Glaucoma Efficacy Garai, Sumanta; Leo, Luciana M.; Szczesniak, Anna-Maria; Hurst, Dow P.; Schaffer, Peter C.; Zagzoog, Ayat; Black, Tallan; Deschamps, Jeffrey R.; Miess, Elke; Schulz, Stefan; Janero, David R.; Straiker, Alex; Pertwee, Roger G.; Abood, Mary E.; Kelly, Melanie E. M.; Reggio, Patricia H.; Laprairie, Robert B.; Thakur, Ganesh A. Share Save
Variously substituted 2-oxopyridine derivatives: Extending the structure-activity relationships for allosteric modulation of the cannabinoid CB2 receptor Gado, Francesca; Mohamed, Kawthar A.; Meini, Serena; Ferrisi, Rebecca; Bertini, Simone; Digiacomo, Maria; D'Andrea, Felicia; Stevenson, Lesley A.; Laprairie, Robert B.; Pertwee, Roger G.; Manera, Clementina Share Save
PSNCBAM-1 analogs: Structural evolutions and allosteric properties at cannabinoid CB1 receptor Meini, Serena; Gado, Francesca; Stevenson, Lesley A.; Digiacomo, Maria; Saba, Alessandro; Codini, Simone; Macchia, Marco; Pertwee, Roger G.; Bertini, Simone; Manera, Clementina Share Save
Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activity Brizzi, Antonella; Aiello, Francesca; Boccella, Serena; Cascio, Maria Grazia; De Petrocellis, Luciano; Frosini, Maria; Gado, Francesca; Ligresti, Alessia; Luongo, Livio; Marini, Pietro; Mugnaini, Claudia; Pessina, Federica; Corelli, Federico; Maione, Sabatino; Manera, Clementina; Pertwee, Roger G.; Di Marzo, Vincenzo Share Save
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Application of Fluorine- and Nitrogen-Walk Approaches: Defining the Structural and Functional Diversity of 2-Phenylindole Class of Cannabinoid 1 Receptor Positive Allosteric Modulators Garai, Sumanta; Kulkarni, Pushkar M.; Schaffer, Peter C.; Leo, Luciana M.; Brandt, Asher L.; Zagzoog, Ayat; Black, Tallan; Lin, Xiaoyan; Hurst, Dow P.; Janero, David R.; Abood, Mary E.; Zimmowitch, Anaelle; Straiker, Alex; Pertwee, Roger G.; Kelly, Melanie; Szczesniak, Anna-Maria; Denovan-Wright, Eileen M.; Mackie, Ken; Hohmann, Andrea G.; Reggio, Patricia H.; Laprairie, Robert B.; Thakur, Ganesh A. Share Save
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