未登录 分享 收藏
Hydrochloride Salt of the GABAkine KRM-II-81 Mian, Md Yeunus; Divovic, Branka; Sharmin, Dishary; Pandey, Kamal P.; Golani, Lalit K. .; Tiruveedhula, V. V. N. Phani Babu; Cerne, Rok; Smith, Jodi L.; Ping, Xingjie; Jin, Xiaoming; Imler, Gregory H.; Deschamps, Jeffrey R.; Lippa, Arnold; Cook, James M.; Savic, Miroslav M.; Rowlett, James; Witkin, Jeffrey M. 分享 收藏
Design, Synthesis, and In Vivo Evaluation of C1-Linked 4,5-Epoxymorphinan Haptens for Heroin Vaccines Sulima, Agnieszka; Li, Fuying; Morgan, Jeffrey Brian; Phong Truong; Antoline, Joshua F. G.; Oertel, Therese; Barrientos, Rodell C.; Torres, Oscar B.; Beck, Zoltan; Imler, Gregory H.; Deschamps, Jeffrey R.; Matyas, Gary R.; Jacobson, Arthur E.; Rice, Kenner C. 分享 收藏
Discovery of a Biased Allosteric Modulator for Cannabinoid 1 Receptor: Preclinical Anti-Glaucoma Efficacy Garai, Sumanta; Leo, Luciana M.; Szczesniak, Anna-Maria; Hurst, Dow P.; Schaffer, Peter C.; Zagzoog, Ayat; Black, Tallan; Deschamps, Jeffrey R.; Miess, Elke; Schulz, Stefan; Janero, David R.; Straiker, Alex; Pertwee, Roger G.; Abood, Mary E.; Kelly, Melanie E. M.; Reggio, Patricia H.; Laprairie, Robert B.; Thakur, Ganesh A. 分享 收藏
分享 收藏
G-Protein biased opioid agonists: 3-hydroxy-N-phenethyl-5-phenylmorphans with three-carbon chain substituents at C9 Gutman, Eugene S.; Bow, Eric; Li, Fuying; Sulima, Agnieszka; Kaska, Sophia; Crowley, Rachel; Prisinzano, Thomas E.; Lee, Yong-Sok; Hassan, Sergio A.; Imler, Gregory H.; Deschamps, Jeffrey R.; Jacobson, Arthur E.; Rice, Kenner C. 分享 收藏
Reply to the 'Comment on Investigation of Zr(iv) and 89Zr(IV) complexation with hydroxamates: progress towards designing a better chelator than desferrioxamine B for immuno-PET imaging' by A. Bianchi and M. Savastano, Chem. Commun., 2020, 56, D0CC01189D Guerard, Francois; Lee, Yong-Sok; Tripier, Raphael; Szajek, Lawrence P.; Deschamps, Jeffrey R.; Brechbiel, Martin W. 分享 收藏
C4-Phenylthio β-lactams: Effect of the chirality of the β-lactam ring on antimicrobial activity Kuskovsky, Rostislav; Lloyd, Dina; Arora, Kriti; Plotkin, Balbina J.; Green, Jacalyn M.; Boshoff, Helena I.; Barry, Clifton, III; Deschamps, Jeffrey; Konaklieva, Monika I. 分享 收藏
A Novel Bromine-Containing Paroxetine Analogue Provides Mechanistic Clues for Binding Ambiguity at the Central Primary Binding Site of the Serotonin Transporter 新型含溴的帕罗西汀类似物为5-羟色胺转运蛋白的中央主要结合位点的结合歧义提供了机理线索 Slack, Rachel D.; Abramyan, Ara M.; Tang, Helen; Meena, Sitaram; Davis, Bruce A.; Bonifazi, Alessandro; Giancola, JoLynn B.; Deschamps, Jeffrey R.; Naing, Sett; Yano, Hideaki; Singh, Satinder K.; Newman, Amy Hauck; Shi, Lei 分享 收藏
The Significance of Chirality in Drug Design and Synthesis of Bitopic Ligands as D3 Receptor (D3R) Selective Agonists Battiti, Francisco O.; Cemaj, Sophie L.; Guerrero, Adrian M.; Shaik, Anver Basha; Lam, Jenny; Rais, Rana; Slusher, Barbara S.; Deschamps, Jeffery R.; Imler, Greg H.; Newman, Amy Hauck; Bonifazi, Alessandro 分享 收藏
分享 收藏
分享 收藏
Synthesis and Characterization of the Selective, Reversible PKCβ Inhibitor (9S)-9-[(Dimethylamino)methyl]-6,7,10,11-tetrahydro-9H,18H-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexade cine-18,20(19H)-dione, Ruboxistaurin (LY333531) Lewin, Anita H.; Brieaddy, Larry; Deschamps, Jeffrey R.; Imler, Gregory H.; Mascarella, S. Wayne; Reddy, P. Anantha; Carroll, F. Ivy 分享 收藏
分享 收藏
分享 收藏
分享 收藏
分享 收藏
A Stable Heroin Analogue That Can Serve as a Vaccine Hapten to Induce Antibodies That Block the Effects of Heroin and Its Metabolites in Rodents and That Cross-React Immunologically with Related Drugs of Abuse Sulima, Agnieszka; Jalah, Rashmi; Antoline, Joshua F. G.; Torres, Oscar B.; Imler, Gregory H.; Deschamps, Jeffrey R.; Beck, Zoltan; Alving, Carl R.; Jacobson, Arthur E.; Rice, Kenner C.; Matyas, Gary R. 分享 收藏
Concise Total Synthesis of (-)-Affinisine Oxindole, (+)-Isoalstonisine, (+)-Alstofoline, (-)-Macrogentine, (+)-Na-Demethylalstonisine, (-)-AlstonoxineA, and (+)-Alstonisine Stephen, Michael Rajesh; Rahman, M. Toufiqur; Tiruveedhula, V. V. N. Phani Babu; Fonseca, German O.; Deschamps, Jeffrey R.; Cook, James M. 分享 收藏
Elucidating Surface Ligand-Dependent Kinetic Enhancement of Proteolytic Activity at Surface-Modified Quantum Dots Diaz, Sebastian A.; Sen, Soumyo; Gemmill, Kelly Boeneman; Brown, Carl W., III; Oh, Eunkeu; Susumu, Kimihiro; Stewart, Michael H.; Breger, Joyce C.; Aragones, Guillermo Lasarte; Field, Lauren D.; Deschamps, Jeffrey R.; Kral, Petr; Medintz, Igor L. 分享 收藏
.png){kind=icon}
未登录.png){kind=icon}
.png){kind=icon}
.png){kind=icon}
.png){kind=icon}
.png){kind=icon}