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J

Jana Selent

pompeu fabra university

33H指数
143论文数
3.6K被引数
收录论文 71
发表时间
The GPCRVP score reliably predicts the impact of GLP1R human variants on receptor functionGPCRVP评分可靠地预测GLP1R人类变异体对受体功能的影响
err2026-09-17
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errOAAI
errMarta Lopez-Balastegui; Shuangyu Lian; Wenwen Gao; Florence Gbahou; Tomasz M. Stepniewski; Julie Dam; Ralf Jockers; Jana Selent
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Peptide ligand discovery of G protein-coupled receptorsG蛋白偶联受体肽配体的发现
err2026-07-16
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PREAI
errJulius Hermes; Marin Matic; Ho Yan Yeung; Qianru Jiang; Lauri Urvas; Elizaveta Korchevaya; Tomasz Stepniewski; Alexandre Murza; Jana Selent; Michael Freissmuth; Christian Heinis; Pierre-Luc Boudreault; Jens Carlsson; Tao Che; Helena Safavi-Hemami; Alexander S. Hauser; Christian W. Gruber
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Structural mechanism for noncanonical GPCR signaling in the Hedgehog pathwayHedgehog通路中非典型GPCR信号传导的结构机制
err2026-04-01
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PREAI
errSteiner, William P.; Iverson, Nathan; Liu, Guibing; Venkatakrishnan, Varun; Wu, Jian; Stepniewski, Tomasz Maciej; Michaelson, Zachary; Brockel, Jan W.; Zhu, Ju-Fen; Bruystens, Jessica G. H.; Lee, Annabel; Nelson, Isaac; Bertinetti, Daniela; Arveseth, Corvin D.; Tan, Gerald; Spaltenstein, Paul; Xu, Jiewei; Huttenhain, Ruth; Kay, Michael S.; Herberg, Friedrich W.; Cao, Erhu; Selent, Jana; Anand, Ganesh S.; Dunbrack Jr, Roland L.; Taylor, Susan S.; Myers, Benjamin R.
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Location-biased β-arrestin conformations direct GPCR signaling位置偏好性的β-arrestin构象指导GPCR信号传导
err2026-03-24
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PREAI
errUyen Pham; Anand Chundi; Tomasz M. Stępniewski; Srikrishna Darbha; Dylan S. Eiger; Sonia Gazula; Julia Gardner; Chloe Hicks; Jana Selent; Sudarshan Rajagopal
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Rare variant in intracellular loop-2 alters the spatial distribution and transducer coupling selectivity of the ghrelin receptorghrelin受体胞内环-2中的稀有变异改变了其空间分布和转导蛋白偶联选择性。
err2026-03-13
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errOAAI
errElsa M. Balfe; Alexandre Torbey; Tomasz M. Stepniewski; Yang Zhou; Lara Kohlenbach; Jade A. Sency; Asuka Inoue; Lauren M. Slosky; Jana Selent; Lawrence S. Barak; Joshua D. Gross
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Distinctive patterns of G protein coupling induced by the structurally similar 5-HT2A receptor ligands ketanserin and altanserin in human prefrontal cortex结构相似的5-HT2A受体配体ketanserin和altanserin在人前额皮质中诱导的G蛋白偶联特异性模式
err2025-09-24
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errOAAI
errPatricia Miranda-Azpiazu; Carolina Muguruza; Tomasz Maciej Stepniewski; Itziar Muneta-Arrate; David Moreira; José Brea; Luis F. Callado; María Isabel Loza; Javier González-Maeso; Jana Selent; Rebeca Diez-Alarcia; J.Javier Meana
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Loss-of-function Gαs rare disease variants exert mutation-specific effects on GPCR signaling失活功能型Gαs罕见病变异体对GPCR信号传导产生突变特异性的影响
err2025-05-20
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PREAI
errRedfern-Nichols, Theo; O'Brien, Shannon L.; Huang, Xianglin; Medel-Lacruz, Brian; Calebiro, Davide; Selent, Jana; Ladds, Graham; Marti-Solano, Maria
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Computational Design and Evaluation of Peptides to Target SARS-CoV-2 Spike-ACE2 Interaction靶向SARS-CoV-2 Spike-ACE2相互作用的多肽的计算设计和评估
err2025-04-14
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errOAAI
errAlmabhouh, Saja; Cecon, Erika; Basubas, Florence; Molina-Fernandez, Ruben; Maciej Stepniewski, Tomasz; Selent, Jana; Jockers, Ralf; Rahmeh, Amal; Oliva, Baldo; Fernandez-Fuentes, Narcis
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Discovery and characterization of small-molecule TGR5 ligands with agonistic activity
err2024-10-01
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errOAAI
errPapadopoulos, M. Giovanna E.; Perhal, Alexander F.; Medel-Lacruz, Brian; Ladurner, Angela; Selent, Jana; Dirsch, Verena M.; Kolb, Peter
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The path to the G protein-coupled receptor structural landscape: Major milestones and future directions
err2024-08-29
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errOAAI
errKogut-Guenthel, Malgorzata M.; Zara, Zeenat; Nicoli, Alessandro; Steuer, Alexandra; Lopez-Balastegui, Marta; Selent, Jana; Karanth, Sanjai; Koehler, Melanie; Ciancetta, Antonella; Abiko, Layara Akemi; Hagn, Franz; Di Pizio, Antonella
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Phosphorylation patterns in the AT1R C-terminal tail specify distinct downstream signaling pathways
err2024-08-13
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errOAAI
errGareri, Clarice; Pfeiffer, Conrad T.; Jiang, Xue; Paulo, Joao A.; Gygi, Steven P.; Pham, Uyen; Chundi, Anand; Wingler, Laura M.; Staus, Dean P.; Stepniewski, Tomasz Maciej; Selent, Jana; Lucero, Emilio Y.; Grogan, Alyssa; Rajagopal, Sudarshan; Rockman, Howard A.
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Relevance of G protein-coupled receptor (GPCR) dynamics for receptor activation, signalling bias and allosteric modulation
err2024-07-08
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errOAAI
errLopez-Balastegui, Marta; Stepniewski, Tomasz Maciej; Kogut-Guenthel, Malgorzata M.; Di Pizio, Antonella; Rosenkilde, Mette Marie; Mao, Jiafei; Selent, Jana
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Altered desensitization and internalization patterns of rodent versus human glucose-dependent insulinotropic polypeptide (GIP) receptors. An important drug discovery challenge
err2024-07-01
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errGasbjerg, Laerke Smidt; Rasmussen, Rasmus Syberg; Dragan, Adrian; Lindquist, Peter; Melchiorsen, Josefine Ulrikke; Stepniewski, Tomasz Maciej; Schiellerup, Sine; Tordrup, Esther Karen; Gadgaard, Sarina; Kizilkaya, Husun Sheyma; Willems, Sabine; Zhong, Yi; Wang, Yi; Wright, Shane C.; Lauschke, Volker M.; Hartmann, Bolette; Holst, Jens Juul; Selent, Jana; Rosenkilde, Mette Marie
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G protein-specific mechanisms in the serotonin 5-HT2A receptor regulate psychosis-related effects and memory deficits
err2024-05-29
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errOAAI
errKossatz, Elk; Diez-Alarcia, Rebeca; Gaitonde, Supriya A.; Ramon-Duaso, Carla; Stepniewski, Tomasz Maciej; Aranda-Garcia, David; Muneta-Arrate, Itziar; Tepaz, Elodie; Saen-Oon, Suwipa; Soliva, Robert; Shahraki, Aida; Moreira, David; Brea, Jose; Loza, Maria Isabel; de la Torre, Rafael; Kolb, Peter; Bouvier, Michel; Meana, J. Javier; Robledo, Patricia; Selent, Jana
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Pharmacological fingerprint of antipsychotic drugs at the serotonin 5-HT2A receptor
err2024-04-02
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errOAAI
errGaitonde, Supriya A.; Avet, Charlotte; Revenga, Mario de la Fuente; Blondel-Tepaz, Elodie; Shahraki, Aida; Pastor, Adrian Morales; Talagayev, Valerij; Robledo, Patricia; Kolb, Peter; Selent, Jana; Gonzalez-Maeso, Javier; Bouvier, Michel
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Exploiting thiol-functionalized benzosiloxaboroles for achieving diverse substitution patterns - synthesis, characterization and biological evaluation of promising antibacterial agents
err2024-01-01
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errNowicki, Krzysztof; Krajewska, Joanna; Stepniewski, Tomasz M.; Wielechowska, Monika; Winska, Patrycja; Kaczmarczyk, Anna; Korpowska, Julia; Selent, Jana; Marek-Urban, Paulina H.; Durka, Krzysztof; Wozniak, Krzysztof; Laudy, Agnieszka E.; Lulinski, Sergiusz
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Impact of membrane lipid polyunsaturation on dopamine D2 receptor ligand binding and signaling (vol 28, pg 1960, 2023)
err2023-08-07
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errOAAI
errJobin, Marie-Lise; De Smedt-Peyrusse, Veronique; Ducrocq, Fabien; Baccouch, Rim; Oummadi, Asma; Pedersen, Maria Hauge; Medel-Lacruz, Brian; Angelo, Maria-Florencia; Villette, Sandrine; Van Delft, Pierre; Fouillen, Laetitia; Mongrand, Sebastien; Selent, Jana; Tolentino-Cortez, Tarson; Barreda-Gomez, Gabriel; Gregoire, Stephane; Masson, Elodie; Durroux, Thierry; Javitch, Jonathan A.; Guixa-Gonzalez, Ramon; Alves, Isabel D.; Trifilieff, Pierre
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