未登录Phenotypic Hit Identification and Optimization of Novel Pan-TEAD and Subtype-Selective Inhibitors表型筛选识别和优化新型泛TEAD及亚型选择性抑制剂
Heinrich, Timo; Gambardella, Alessia; Schwarz, Daniel; Petersson, Carl; Gunera, Jakub; Garg, Sakshi; Schneider, Richard; Keil, Marina; Grimmeisen, Lisa; Unzue Lopez, Andrea; Schilke, Heike; Weitzel, Thomas; Kolb, Christian; Diehl, Patrizia; Doerfel, Benjamin; Anlauf, Uwe; Reither, Vivian; Rettig, Corinna; Opelt, Beate; Delp, Andrea; Wildner, Nicole; Musil, Djordje; Friedrich, Erik; Burgdorf, Lars; Fuchss, Thomas; Albers, Lisa; Sousa, Pedro M. F.; Freire, Filipe; M. Bandeiras, Tiago; Wienke, Dirk
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收藏MoA Studies of the TEAD P-Site Binding Ligand MSC-4106 and Its Optimization to TEAD1-Selective Amide M3686
Heinrich, Timo; Schwarz, Daniel; Petersson, Carl; Gunera, Jakub; Garg, Sakshi; Schneider, Richard; Keil, Marina; Grimmeisen, Lisa; Unzue Lopez, Andrea; Albers, Lisa; Schlesiger, Sarah; Gambardella, Alessia; Bomke, Joerg; Carswell, Emma; Schilke, Heike; Diehl, Patrizia; Doerfel, Benjamin; Musil, Djordje; Trivier, Elisabeth; Broome, Rebecca; Marshall, Sam; Balsiger, Alexander; Friedrich, Erik; Lemos, Ana R.; Santos, Sandra P.; Sousa, Pedro M. F.; Freire, Filipe; Bandeiras, Tiago M.; Bortoluzzi, Alessio; Wienke, Dirk
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收藏Three million images and morphological profiles of cells treated with matched chemical and genetic perturbations用匹配的化学和遗传扰动处理的细胞的300万张图像和形态特征
Chandrasekaran, Srinivas Niranj; Cimini, Beth A.; Goodale, Amy; Miller, Lisa; Kost-Alimova, Maria; Jamali, Nasim; Doench, John G.; Fritchman, Briana; Skepner, Adam; Melanson, Michelle; Kalinin, Alexandr A.; Arevalo, John; Haghighi, Marzieh; Caicedo, Juan C.; Kuhn, Daniel; Hernandez, Desiree; Berstler, James; Shafqat-Abbasi, Hamdah; Root, David E.; Swalley, Susanne E.; Garg, Sakshi; Singh, Shantanu; Carpenter, Anne E.
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收藏Optimizing the Cell Painting assay for image-based profiling优化基于图像的分析的细胞绘画分析
Cimini, Beth A.; Chandrasekaran, Srinivas Niranj; Kost-Alimova, Maria; Miller, Lisa; Goodale, Amy; Fritchman, Briana; Byrne, Patrick; Garg, Sakshi; Jamali, Nasim; Logan, David J.; Concannon, John B.; Lardeau, Charles-Hugues; Mouchet, Elizabeth; Singh, Shantanu; Abbasi, Hamdah Shafqat; Aspesi, Jr Peter; Boyd, Justin D.; Gilbert, Tamara; Gnutt, David; Hariharan, Santosh; Hernandez, Desiree; Hormel, Gisela; Juhani, Karolina; Melanson, Michelle; Mervin, Lewis H.; Monteverde, Tiziana; Pilling, James E.; Skepner, Adam; Swalley, Susanne E.; Vrcic, Anita; Weisbart, Erin; Williams, Guy; Yu, Shan; Zapiec, Bolek; Carpenter, Anne E.
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收藏Optimization of TEAD P-Site Binding Fragment Hit into In Vivo Active Lead MSC-4106
Heinrich, Timo; Peterson, Carl; Schneider, Richard; Garg, Sakshi; Schwarz, Daniel; Gunera, Jakub; Seshire, Anita; Koetzner, Lisa; Schlesiger, Sarah; Musil, Djordje; Schilke, Heike; Doerfel, Benjamin; Diehl, Patrizia; Boepple, Pia; Lemos, Ana R.; Sousa, Pedro M. F.; Freire, Filipe; Bandeiras, Tiago M.; Carswell, Emma; Pearson, Nicholas; Sirohi, Sameer; Hooker, Mollie; Trivier, Elisabeth; Broome, Rebecca; Balsiger, Alexander; Crowden, Abigail; Dillon, Christian; Wienke, Dirk
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收藏Unconventional secretory processing diversifies neuronal ion channel properties
Hanus, Cyril; Geptin, Helene; Tushev, Georgi; Garg, Sakshi; Alvarez-Castelao, Beatriz; Sambandan, Sivakumar; Kochen, Lisa; Hafner, Anne-Sophie; Langer, Julian D.; Schuman, Erin M.
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收藏Direct visualization of newly synthesized target proteins in situ
Dieck, Susanne Tom; Kochen, Lisa; Hanus, Cyril; Heumueller, Maximilian; Bartnik, Ina; Nassim-Assir, Belquis; Merk, Katrin; Mosler, Thorsten; Garg, Sakshi; Bunse, Stefanie; Tirrell, David A.; Schuman, Erin M.
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