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A novel potent class I HDAC inhibitor reverses the STAT4/p66Shc apoptotic defect in B cells from chronic lymphocytic leukemia patients Rossi, Sara; Tatangelo, Vanessa; Dichiara, Maria; Butini, Stefania; Gemma, Sandra; Brogi, Simone; Pasquini, Silvia; Cappello, Martina; Vincenzi, Fabrizio; Varani, Katia; Lopresti, Ludovica; Malchiodi, Margherita; Carrara, Chiara; Gozzetti, Alessandro; Bocchia, Monica; Marotta, Giuseppe; Patrussi, Laura; Carullo, Gabriele; Baldari, Cosima T.; Campiani, Giuseppe 分享 收藏
Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence Bedini, Annalida; Elisi, Gian Marco; Fanini, Fabiola; Retini, Michele; Scalvini, Laura; Pasquini, Silvia; Contri, Chiara; Varani, Katia; Spadoni, Gilberto; Mor, Marco; Vincenzi, Fabrizio; Rivara, Silvia 分享 收藏
2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A1 Adenosine Receptor Positive Allosteric Modulators Oliva, Paola; Suresh, R. Rama; Pasquini, Silvia; Salmaso, Veronica; Will, Edward J.; Tosh, Dilip K.; Gao, Zhan-Guo; Liu, Naili; Gavrilova, Oksana; Vincenzi, Fabrizio; Varani, Katia; Jacobson, Kenneth A. 分享 收藏
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MAM-2201 acute administration impairs motor, sensorimotor, prepulse inhibition, and memory functions in mice: a comparison with its analogue AM-2201 Corli, Giorgia; Tirri, Micaela; Bilel, Sabrine; Arfe, Raffaella; Coccini, Teresa; Roda, Elisa; Marchetti, Beatrice; Vincenzi, Fabrizio; Zauli, Giorgio; Borea, Pier Andrea; Locatelli, Carlo Alessandro; Varani, Katia; Marti, Matteo 分享 收藏
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Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania 分享 收藏
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2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto 分享 收藏
Synthesis of Unsymmetrical Squaramides as Allosteric GSK-3β Inhibitors Promoting β-Catenin-Mediated Transcription of TCF/LEF in Retinal Pigment Epithelial Cells Carullo, Gabriele; Bottoni, Laura; Pasquini, Silvia; Papa, Alessandro; Contri, Chiara; Brogi, Simone; Calderone, Vincenzo; Orlandini, Maurizio; Gemma, Sandra; Varani, Katia; Butini, Stefania; Galvagni, Federico; Vincenzi, Fabrizio; Campiani, Giuseppe 分享 收藏
Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability Federico, Stefano; Khan, Tuhina; Fontana, Anna; Brogi, Simone; Benedetti, Rosaria; Sarno, Federica; Carullo, Gabriele; Pezzotta, Alex; Saraswati, Akella Prasanth; Passaro, Eugenia; Pozzetti, Luca; Papa, Alessandro; Relitti, Nicola; Gemma, Sandra; Butini, Stefania; Pistocchi, Anna; Ramunno, Anna; Vincenzi, Fabrizio; Varani, Katia; Tatangelo, Vanessa; Patrussi, Laura; Baldari, Cosima T.; Saponara, Simona; Gorelli, Beatrice; Lamponi, Stefania; Valoti, Massimo; Saccoccia, Fulvio; Giannaccari, Marialaura; Ruberti, Giovina; Herp, Daniel; Jung, Manfred; Altucci, Lucia; Campiani, Giuseppe 分享 收藏
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Pathophysiological Role and Medicinal Chemistry of A2A Adenosine Receptor Antagonists in Alzheimer's Disease A2A腺苷受体拮抗剂在阿尔茨海默病中的病理生理作用和药物化学 Merighi, Stefania; Borea, Pier Andrea; Varani, Katia; Vincenzi, Fabrizio; Travagli, Alessia; Nigro, Manuela; Pasquini, Silvia; Suresh, R. Rama; Kim, Sung Won; Volkow, Nora D.; Jacobson, Kenneth A.; Gessi, Stefania 分享 收藏
4-Heteroaryl Substituted Amino-3,5-Dicyanopyridines as New Adenosine Receptor Ligands: Novel Insights on Structure-Activity Relationships and Perspectives Catarzi, Daniela; Varano, Flavia; Vigiani, Erica; Calenda, Sara; Melani, Fabrizio; Varani, Katia; Vincenzi, Fabrizio; Pasquini, Silvia; Mennini, Natascia; Nerli, Giulia; Dal Ben, Diego; Volpini, Rosaria; Colotta, Vittoria 分享 收藏
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