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Antonio Macchiarulo

University of Perugia
H指数:43
被引数:9,226

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Targeting oxysterol-binding protein (OSBP) as a novel strategy to inhibit herpes simplex virus 2 (HSV-2) replication: First structure-activity relationship study of antiviral cholenamide derivatives

靶向氧甾醇结合蛋白(OSBP)作为抑制单纯疱疹病毒2型(HSV-2)复制的新型策略：抗病毒胆酰胺衍生物的首个构效关系研究

European Journal of Medicinal Chemistry
IF5.9
2026-08-010
PRE
Civra, Andrea; Nigro, Fatima; Porporato, Domiziana; Costantino, Matteo; Bianconi, Elisa; Zambri, Federico; De March, Matteo; De Conto, Marco; Carosati, Emanuele; Macchiarulo, Antonio; Lembo, David; Marinozzi, Maura
Synthesis and structure-activity relationship study of a library of 1-substituted [1,2,4]triazolo[4,3-a]quinolines as valuable chemical probes for paraxonase-2 (PON2)

1-取代的[1,2,4]三唑并[4,3-a]喹啉库的合成及构效关系研究，将其作为帕罗尼酶-2（PON2）的有价值的化学探针

Journal of Enzyme Inhibition and Medicinal Chemistry
IF5.4
2026-03-260
OA
Elisa Bianconi; Eros Antonio Lampitella; Fatima Nigro; Ludovica Rossi; Federico Zambri; Simone Fava; Maria Marone; Elena Porzio; Antonio Macchiarulo; Giuseppe Manco; Maura Marinozzi
Design, Synthesis, and Biological Characterization of Macromolecular Ester Prodrugs of a Selective Cyclooxygenase-2 Inhibitor

选择性环氧化酶-2抑制剂的大分子酯前药的设计、合成与生物特性研究

CHEMMEDCHEM
IF3.4
2025-11-010
OAAI
Saletti, Mario; Paolino, Marco; Venditti, Jacopo; Giuliani, Germano; Rossi, Antonietta; D'avino, Danilo; Perna, Sara; Varfaj, Ina; Sardella, Roccaldo; Macchiarulo, Antonio; Maramai, Samuele; Lamponi, Stefania; Cappelli, Andrea; Anzini, Maurizio
Optimization of potent, broad-spectrum, and specific anti-influenza compounds targeting RNA polymerase PA-PB1 heterodimerization
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
IF5.9
2024-11-012
PRE
Bonomini, Anna; Felicetti, Tommaso; Pacetti, Martina; Bertagnin, Chiara; Coletti, Alice; Giammarino, Federica; De Angelis, Marta; Poggialini, Federica; Macchiarulo, Antonio; Sabatini, Stefano; Mercorelli, Beatrice; Nencioni, Lucia; Vicenti, Ilaria; Dreassi, Elena; Cecchetti, Violetta; Tabarrini, Oriana; Loregian, Arianna; Massari, Serena
A microbially produced AhR ligand promotes a Tph1-driven tolerogenic program in multiple sclerosis

微生物产生的AhR配体促进多发性硬化症的Tph1-driven耐受计划

SCIENTIFIC REPORTS
IF3.9
2024-03-203
OAAI
Zelante, Teresa; Paolicelli, Giuseppe; Fallarino, Francesca; Gargaro, Marco; Vascelli, Gianluca; De Zuani, Marco; Fric, Jan; Laznickova, Petra; Kohoutkova, Marcela Hortova; Macchiarulo, Antonio; Dolciami, Daniela; Pieraccini, Giuseppe; Gaetani, Lorenzo; Scalisi, Giulia; Trevisan, Caterina; Frossi, Barbara; Pucillo, Carlo; De Luca, Antonella; Nunzi, Emilia; Spaccapelo, Roberta; Pariano, Marilena; Borghi, Monica; Boscaro, Francesca; Romoli, Riccardo; Mancini, Andrea; Gentili, Lucia; Renga, Giorgia; Costantini, Claudio; Puccetti, Matteo; Giovagnoli, Stefano; Ricci, Maurizio; Antonini, Martina; Calabresi, Paolo; Puccetti, Paolo; Di Filippo, Massimiliano; Romani, Luigina
Design, synthesis, and biological evaluation of first-in-class indomethacin-based PROTACs degrading SARS-CoV-2 main protease and with broad-spectrum antiviral activity

降解SARS-CoV-2主要蛋白酶并具有广谱抗病毒活性的基于吲哚美辛的PROTACs的设计，合成和生物学评价

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
IF5.9
2024-03-0110
OAAI
Desantis, Jenny; Bazzacco, Alessandro; Eleuteri, Michela; Tuci, Sara; Bianconi, Elisa; Macchiarulo, Antonio; Mercorelli, Beatrice; Loregian, Arianna; Goracci, Laura
Combining Solid-State NMR with Structural and Biophysical Techniques to Design Challenging Protein-Drug Conjugates

将固态NMR与结构和生物物理技术相结合，以设计具有挑战性的蛋白质-药物缀合物

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
IF16.9
2023-06-220
OAAI
Cerofolini, Linda; Vasa, Kristian; Bianconi, Elisa; Salobehaj, Maria; Cappelli, Giulia; Bonciani, Alice; Licciardi, Giulia; Perez-Rafols, Anna; Padilla-Cortes, Luis; Antonacci, Sabrina; Rizzo, Domenico; Ravera, Enrico; Viglianisi, Caterina; Calderone, Vito; Parigi, Giacomo; Luchinat, Claudio; Macchiarulo, Antonio; Menichetti, Stefano; Fragai, Marco
A multicentric consortium study demonstrates that dimethylarginine dimethylaminohydrolase 2 is not a dimethylarginine dimethylaminohydrolase
NATURE COMMUNICATIONS
IF15.7
2023-06-099
OAAI
Ragavan, Vinitha N.; Nair, Pramod C.; Jarzebska, Natalia; Angom, Ramcharan Singh; Ruta, Luana; Bianconi, Elisa; Grottelli, Silvia; Tararova, Natalia D.; Ryazanskiy, Daniel; Lentz, Steven R.; Tommasi, Sara; Martens-Lobenhoffer, Jens; Suzuki-Yamamoto, Toshiko; Kimoto, Masumi; Rubets, Elena; Chau, Sarah; Chen, Yingjie; Hu, Xinli; Bernhardt, Nadine; Spieth, Peter M.; Weiss, Norbert; Bornstein, Stefan R.; Mukhopadhyay, Debabrata; Bode-Boeger, Stefanie M.; Maas, Renke; Wang, Ying; Macchiarulo, Antonio; Mangoni, Arduino A.; Cellini, Barbara; Rodionov, Roman N.

研究方向

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R
Roberto Pellicciari
H 指数:57论文数:458被引数:1.6万
A
Andrea Carotti
H 指数:30论文数:182被引数:2,901
A
Antimo Gioiello
H 指数:36论文数:178被引数:6,832
R
Roccaldo Sardella
H 指数:30论文数:186被引数:3,023
E
Emidio Camaioni
H 指数:33论文数:152被引数:4,545
C
Ciriana Orabona
H 指数:46论文数:125被引数:1.2万
A
Alice Coletti
H 指数:13论文数:36被引数:729
G
Gabriele Costantino
H 指数:44论文数:243被引数:7,204
F
Francesca Fallarino
H 指数:73论文数:270被引数:2.4万
M
Maura Marinozzi
H 指数:29论文数:162被引数:2,893