Sergey Zozulya - Publications, H-index & Citations

Sergey Zozulya

enamine biology (bienta)/enamine ltd

30H指数

114论文数

4.5K被引数

收录论文 34

发表时间

Expanding Chemical Space of N-Acyl Sulfonamides for Carbonic Anhydrase Inhibitor Discovery 扩展N-酰基磺酰胺的化学空间以发现碳酸酐酶抑制剂

European Journal of Medicinal Chemistry

IF5.9

2025-10-23

PREAI

Oleksii V. Gavrylenko; Bohdan V. Vashchenko; Vasyl Naumchyk; Oleksii Chuk; Olga Kuchuk; Alla Pogribna; Anzhelika I. Konovets; Volodymyr S. Brovarets; Sergey A. Zozulya; Dmytro S. Radchenko; Oleksandr O. Grygorenko; Yurii S. Moroz

The molecular features of non-peptidic nucleophilic substrates and acceptor proteins determine the efficiency of sortagging

RSC CHEMICAL BIOLOGY

IF3.1

2025-01-01

OAAI

Bondarchuk, Tetiana; Zhuravel, Elena; Shyshlyk, Oleh; Debelyy, Mykhaylo O.; Pokholenko, Oleksandr; Vaskiv, Diana; Pogribna, Alla; Kuznietsova, Mariana; Hrynyshyn, Yevhenii; Nedialko, Oleksandr; Brovarets, Volodymyr; Zozulya, Sergey A.

Synthetic Amine Linkers for Efficient Sortagging

BIOCONJUGATE CHEMISTRY

IF3.9

2024-07-12

PREAI

Bondarchuk, Tetiana; Vaskiv, Diana; Zhuravel, Elena; Shyshlyk, Oleh; Hrynyshyn, Yevhenii; Nedialko, Oleksandr; Pokholenko, Oleksandr; Pohribna, Alla; Kuchuk, Olga; Brovarets, Volodymyr; Zozulya, Sergey

Discovery of New Agonists and Antagonists for Ectopically Expressed Olfactory Receptor OR51E1

JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

IF3.8

2023-06-01

OAAI

Henry, Taylor; Wang, Qiang; Pronin, Alexey; Zhuravel, Olena; Zozulya, Sergey; Slepak, Vladlen

Strained contacts with the cell membrane may influence ligand affinity to G protein coupled receptors: a case of free fatty acid receptor 1 agonists

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2021-07-22

OAAI

Lukin, Alexey; Bakholdina, Anna; Chudinov, Mikhail; Onopchenko, Oleksandra; Zhuravel, Elena; Zozulya, Sergey; Gureev, Maxim; Krasavin, Mikhail

Small-Molecule Chemical Knockdown of MuRF1 in Melanoma Bearing Mice Attenuates Tumor Cachexia Associated Myopathy 黑色素瘤荷瘤小鼠中MuRF1的小分子化学敲低可减轻与肿瘤恶病质相关的肌病

CELLS

IF5.2

2020-10-11

OAAI

Adams, Volker; Gussen, Victoria; Zozulya, Sergey; Cruz, Andre; Moriscot, Anselmo; Linke, Axel; Labeit, Siegfried

Synthesis, biological evaluation, and modeling studies of 1,3-disubstituted cyclobutane-containing analogs of combretastatin A4

JOURNAL OF MOLECULAR STRUCTURE

IF4.7

2020-06-01

OAAI

Malashchuk, Andrii; Chernykh, Anton, V; Hurmach, Vasyl V.; Platonov, Maxim O.; Onopchenko, Oleksandra; Zozulya, Sergey; Daniliuc, Constantin G.; Dobrydnev, Alexey, V; Kondratov, Ivan S.; Moroz, Yuriy S.; Grygorenko, Oleksandr O.

A prospective compound screening contest identified broader inhibitors for Sirtuin 1

SCIENTIFIC REPORTS

IF3.9

2019-12-20

OAAI

Chiba, Shuntaro; Ohue, Masahito; Gryniukova, Anastasiia; Borysko, Petro; Zozulya, Sergey; Yasuo, Nobuaki; Yoshino, Ryunosuke; Ikeda, Kazuyoshi; Shin, Woong-Hee; Kihara, Daisuke; Iwadate, Mitsuo; Umeyama, Hideaki; Ichikawa, Takaaki; Teramoto, Reiji; Hsin, Kun-Yi; Gupta, Vipul; Kitano, Hiroaki; Sakamoto, Mika; Higuchi, Akiko; Miura, Nobuaki; Yura, Kei; Mochizuki, Masahiro; Ramakrishnan, Chandrasekaran; Thangakani, A. Mary; Velmurugan, D.; Gromiha, M. Michael; Nakane, Itsuo; Uchida, Nanako; Hakariya, Hayase; Tan, Modong; Nakamura, Hironori K.; Suzuki, Shogo D.; Ito, Tomoki; Kawatani, Masahiro; Kudoh, Kentaroh; Takashina, Sakurako; Yamamoto, Kazuki Z.; Moriwaki, Yoshitaka; Oda, Keita; Kobayashi, Daisuke; Okuno, Tatsuya; Minami, Shintaro; Chikenji, George; Prathipati, Philip; Nagao, Chioko; Mohsen, Attayeb; Ito, Mari; Mizuguchi, Kenji; Honma, Teruki; Ishida, Takashi; Hirokawa, Takatsugu; Akiyama, Yutaka; Sekijima, Masakazu

Screening of benzenesulfonamide in combination with chemically diverse fragments against carbonic anhydrase by differential scanning fluorimetry

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2019-12-04

OAAI

Krasavin, Mikhail; Kalinin, Stanislav; Zozulya, Sergey; Gryniukova, Anastasiia; Borysko, Petro; Angeli, Andrea; Supuran, Claudiu T.

Further validation of strecker-type α-aminonitriles as a new class of potent human carbonic anhydrase II inhibitors: hit expansion within the public domain using differential scanning fluorimetry leads to chemotype refinement

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2019-11-22

OAAI

Krasavin, Mikhail; Kalinin, Stanislav; Zozulya, Sergey; Griniukova, Anastasia; Borysko, Petro; Angeli, Andrea; Supuran, Claudiu T.

Difluoro-Substituted Bicyclo[1.1.1]pentanes for Medicinal Chemistry: Design, Synthesis, and Characterization

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2019-09-25

111

PREAI

Bychek, Roman M.; Hutskalova, Valeriia; Bas, Yuliya P.; Zaporozhets, Olga A.; Zozulya, Sergey; Levterov, Vadym V.; Mykhailiuk, Pavel K.

Photochemical In-Flow Synthesis of 2,4-Methanopyrrolidines: Pyrrolidine Analogues with Improved Water Solubility and Reduced Lipophilicity

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2018-10-25

PREAI

Levterov, Vadym V.; Michurin, Oleg; Borysko, Petro O.; Zozulya, Sergey; Sadkova, Iryna V.; Tolmachev, Andrey A.; Mykhailiuk, Pavel K.

Straightforward hit identification approach in fragment-based discovery of bromodomain-containing protein 4 (BRD4) inhibitors

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2018-07-01

PREAI

Borysko, Petro; Moroz, Yurii S.; Vasylchenko, Oleksandr V.; Hurmach, Vasyl V.; Starodubtseva, Anastasia; Stefanishena, Natalia; Nesteruk, Kateryna; Zozulya, Sergey; Kondratov, Ivan S.; Grygorenko, Oleksandr O.

Synthesis of Multifunctional Spirocyclic Azetidines and Their Application in Drug Discovery

CHEMISTRY-A EUROPEAN JOURNAL

IF3.7

2018-02-15

PREAI

Kirichok, Alexander A.; Shton, Irina O.; Pishel, Irina M.; Zozulya, Sergey A.; Borysko, Petro O.; Kubyshkin, Vladimir; Zaporozhets, Olha A.; Tolmachev, Andrei A.; Mykhailiuk, Pavel K.

Photochemical Synthesis of 2-Azabicyclo[3.2.0]heptanes: Advanced Building Blocks for Drug Discovery. Synthesis of 2,3-Ethanoproline

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2018-01-16

PREAI

Druzhenko, Tetiana; Skalenko, Yevhen; Samoilenko, Maryna; Denisenko, Aleksandr; Zozulya, Sergey; Borysko, Petro O.; Sokolenko, Maria I.; Tarasov, Alexandr; Mykhailiuk, Pavel K.

Continued SAR exploration of 1,2,4-thiadiazole-containing scaffolds in the design of free fatty acid receptor 1 (GPR40) agonists

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2017-11-01

PREAI

Krasavin, Mikhail; Lukin, Alexei; Bakholdina, Anna; Zhurilo, Nikolay; Onopchenko, Oleksandra; Borysko, Petro; Zozulya, Sergey; Moore, Daniel; Tikhonova, Irina G.

An iterative compound screening contest method for identifying target protein inhibitors using the tyrosine-protein kinase Yes

SCIENTIFIC REPORTS

IF3.9

2017-09-20

OAAI

Chiba, Shuntaro; Ishida, Takashi; Ikeda, Kazuyoshi; Mochizuki, Masahiro; Teramoto, Reiji; Taguchi, Y-h.; Iwadate, Mitsuo; Umeyama, Hideaki; Ramakrishnan, Chandrasekaran; Thangakani, A. Mary; Velmurugan, D.; Gromiha, M. Michael; Okuno, Tatsuya; Kato, Koya; Minami, Shintaro; Chikenji, George; Suzuki, Shogo D.; Yanagisawa, Keisuke; Shin, Woong-Hee; Kihara, Daisuke; Yamamoto, Kazuki Z.; Moriwaki, Yoshitaka; Yasuo, Nobuaki; Yoshino, Ryunosuke; Zozulya, Sergey; Borysko, Petro; Stavniichuk, Roman; Honma, Teruki; Hirokawa, Takatsugu; Akiyama, Yutaka; Sekijima, Masakazu

Photochemical Synthesis of 3-Azabicyclo[3.2.0]heptanes: Advanced Building Blocks for Drug Discovery

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2017-08-25

PREAI

Denisenko, Aleksandr V.; Druzhenko, Tetiana; Skalenko, Yevhen; Samoilenko, Maryna; Grygorenko, Oleksandr O.; Zozulya, Sergey; Mykhailiuk, Pavel K.

Polar aromatic periphery increases agonist potency of spirocyclic free fatty acid receptor (GPR40) agonists inspired by LY2881835

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2017-02-01

OAAI

Krasavin, Mikhail; Lukin, Alexey; Bagnyukova, Dania; Zhurilo, Nikolay; Golovanov, Aleksei; Zozulya, Sergey; Zahanich, Ihor; Moore, Daniel; Tikhonova, Irina G.

Free fatty acid receptor 1 (GPR40) agonists containing spirocyclic periphery inspired by LY2881835

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2016-11-01

OAAI

Krasavin, Mikhail; Lukin, Alexey; Bagnyukova, Dania; Zhurilo, Nikolay; Zahanich, Ihor; Zozulya, Sergey; Ihalainen, Jouni; Forsberg, Markus M.; Lehtonen, Marko; Rautio, Jarkko; Moore, Daniel; Tikhonova, Irina G.

研究方向