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David B. Olsen

merck & co., inc.

48H指数
267论文数
1.0W被引数
收录论文 79
发表时间
Chemovaccination with a late-liver-stage antimalarial induces durable immunity against malaria使用晚期肝脏阶段抗疟药物进行化学疫苗接种可诱导持久的疟疾免疫力
errScience
IF45.8
err2026-08-13
err0
PREAI
errRyan W. J. Steel; Yu Cheng Chua; Waail A. I. Abdalla; Robyn McConville; Amelia Ford; Sabrina Caiazzo; Eva Hesping; Daniel Fernandez-Ruiz; Lauren E. Holz; William R. Heath; John A. McCauley; David B. Olsen; Justin A. Boddey
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Discovery and development of a new oxazolidinone with reduced toxicity for the treatment of tuberculosis用于治疗结核病的新型毒性降低的恶唑烷酮的发现和开发
err2026-01-13
err0
errOAAI
errBrendan M. Crowley; Helena I. Boshoff; Aidan Boving; Vee Y. Tan; Jianghai Zhu; Forrest Hoyt; Randy R. Miller; Julie Ehrhart; Christopher W. Boyce; Katherine Young; Philippe G. Nantermet; Jing Su; Lihu Yang; Ronald E. Painter; Emily B. Corcoran; Jason L. Hoar; Sangmi Oh; David L. Holtzman; Micha Levi; Aparna Anderson; Monicah A. Otieno; Matthew Zimmerman; Firat Kaya; Lisa M. Massoudi; Michelle E. Ramey; Allison A. Bauman; Anne J. Lenaerts; Gregory T. Roberston; Véronique Dartois; Charles D. Wells; Clifton E. Barry; David B. Olsen
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Structure-activity analysis of imino-pyrimidinone-fused pyrrolidines aids the development of dual plasmepsin V and plasmepsin X inhibitors亚氨基嘧啶酮稠合的吡咯烷的结构活性分析有助于双重plasmepsin V和plasmepsin X抑制剂的开发
err2025-03-01
err0
errOAAI
errHodder, Anthony N.; Sleebs, Brad E.; Adams, Greg; Rezazadeh, Sina; Ngo, Anna; Jarman, Kate; Scally, Stephen; Czabotar, Peter; Wang, Hongwu; Mccauley, John A.; Olsen, David B.; Cowman, Alan F.
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COVID-19 vaccine associated myocarditis in Norway - a nationwide validation study
err2024-10-28
err0
PREAI
errSkinningsrud, B.; Vlaisavljevic, K.; Oppedal, L. S.; Endresen, J.; Mohn, V; Fladseth, K.; Lysaker, T. M.; Dahl, J.; Gulseth, H. L.; Olsen, D. B.; Ribe, M.; Estensen, M. E.; Broch, K.; Haugaa, K. H.; Hasselberg, N. E.
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Novel Pan-Coronavirus 3CL Protease Inhibitor MK-7845: Biological and Pharmacological Profiling
err2024-07-18
err0
errOAAI
errAlvarez, Nadine; Adam, Gregory C.; Howe, John A.; Sharma, Vijeta; Zimmerman, Matthew D.; Dolgov, Enriko; Rasheed, Risha; Nizar, Fatima; Sahay, Khushboo; Nelson, Andrew M.; Park, Steven; Zhou, Xiaoyan; Burlein, Christine; Fay, John F.; Iwamoto, Daniel V.; Bahnck-Teets, Carolyn M.; Getty, Krista L.; Lin Goh, Shih; Salhab, Imad; Smith, Keith; Boyce, Christopher W.; Cabalu, Tamara D.; Murgolo, Nicholas; Fox, Nicholas G.; Mayhood, Todd W.; Shurtleff, Valerie W.; Layton, Mark E.; Parish, Craig A.; McCauley, John A.; Olsen, David B.; Perlin, David S.
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Mtb-Selective 5-Aminomethyl Oxazolidinone Prodrugs: Robust Potency and Potential Liabilities
err2024-04-06
err2
PREAI
errBoshoff, Helena I. M.; Young, Katherine; Ahn, Yong-Mo; Yadav, Veena D.; Crowley, Brendan M.; Yang, Lihu; Su, Jing; Oh, Sangmi; Arora, Kriti; Andrews, Jenna; Manikkam, Michelle; Sutphin, Michelle; Smith, Anthony J.; Weiner, Danielle M.; Piazza, Michaela K.; Fleegle, Joel D.; Gomez, Felipe; Dayao, Emmannual K.; Prideaux, Brendan; Zimmerman, Matthew; Kaya, Firat; Sarathy, Jansy; Tan, Vee Yang; Via, Laura E.; Tschirret-Guth, Richard; Lenaerts, Anne J.; Robertson, Gregory T.; Dartois, Veronique; Olsen, David B.; Barry III, Clifton E.
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Orally available nucleoside analog UMM-766 provides protection in a murine model of orthopox disease
err2024-04-02
err2
errOAAI
errMudhasani, Rajini R.; Golden, Joseph W.; Adam, Gregory C.; Hartingh, Timothy J.; Kota, Krishna P.; Ordonez, David; Quackenbush, Corey R.; Tran, Julie P.; Cline, Curtis; Williams, Janice A.; Zeng, Xiankun; Olsen, David B.; Lieberman, Linda A.; Boyce, Christopher; Ginnetti, Anthony; Meinig, J. Matthew; Panchal, Rekha G.; Mucker, Eric M.
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Identification of an inhibitory pocket in falcilysin provides a new avenue for malaria drug development
err2024-04-01
err2
errOAAI
errWirjanata, Grennady; Lin, Jianqing; Dziekan, Jerzy Michal; El Sahili, Abbas; Chung, Zara; Tjia, Seth; Zulkifli, Nur Elyza Binte; Boentoro, Josephine; Tham, Roy; Jia, Lai Si; Go, Ka Diam; Yu, Han; Partridge, Anthony; Olsen, David; Prabhu, Nayana; Sobota, Radoslaw M.; Nordlund, Par; Lescar, Julien; Bozdech, Zbynek
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Invention of MK-7845, a SARS-CoV-2 3CL Protease Inhibitor Employing a Novel Difluorinated Glutamine Mimic
err2024-02-16
err4
PREAI
errShurtleff, Valerie W.; Layton, Mark E.; Parish, Craig A.; Perkins, James J.; Schreier, John D.; Wang, Yunyi; Adam, Gregory C.; Alvarez, Nadine; Bahmanjah, Soheila; Bahnck-Teets, Carolyn M.; Boyce, Christopher W.; Burlein, Christine; Cabalu, Tamara D.; Campbell, Brian T.; Carroll, Steven S.; Chang, Wonsuk; de Lera Ruiz, Manuel; Dolgov, Enriko; Fay, John F.; Fox, Nicholas G.; Goh, Shih Lin; Hartingh, Timothy J.; Hurzy, Danielle M.; Kelly III, Michael J.; Klein, Daniel J.; Klingler, Franca-Maria; Krishnamurthy, Harini; Kudalkar, Shalley; Mayhood, Todd W.; McKenna, Philip M.; Murray, Edward M.; Nahas, Debbie; Nawrat, Christopher C.; Park, Steven; Qian, Dongming; Roecker, Anthony J.; Sharma, Vijeta; Shipe, William D.; Su, Jing; Taggart, Robert V.; Truong, Quang; Wu, Yin; Zhou, Xiaoyan; Zhuang, Ningning; Perlin, David S.; Olsen, David B.; Howe, John A.; McCauley, John A.
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Pharmacological validation of dihydrofolate reductase as a drug target in Mycobacterium abscessus
err2024-01-10
err5
errOAAI
errAragaw, Wassihun Wedajo; Negatu, Dereje A.; Bungard, Christopher J.; Dartois, Veronique A.; El Marrouni, Abdellatif; Nickbarg, Elliott B.; Olsen, David B.; Warrass, Ralf; Dick, Thomas
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The Invention of WM382, a Highly Potent PMIX/X Dual Inhibitor toward the Treatment of MalariaWM382的发明,一种用于治疗疟疾的高效PMIX/X双重抑制剂
err2022-10-12
err8
errOAAI
errRuiz, Manuel de Lera; Favuzza, Paola; Guo, Zhuyan; Zhao, Lianyun; Hu, Bin; Lei, Zhiyu; Zhan, Dongmei; Murgolo, Nicholas; Boyce, Christopher W.; Vavrek, Marissa; Thompson, Jennifer; Ngo, Anna; Jarman, Kate E.; Robbins, Johnathan; Boddey, Justin; Sleebs, Brad E.; Lowes, Kym N.; Cowman, Alan F.; Olsen, David B.; McCauley, John A.
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Activity of Tricyclic Pyrrolopyrimidine Gyrase B Inhibitor against Mycobacterium abscessus
err2022-09-20
err6
errOAAI
errMadani, Abdeldjalil; Negatu, Dereje A.; El Marrouni, Abdellatif; Miller, Randy R.; Boyce, Christopher W.; Murgolo, Nicholas; Bungard, Christopher J.; Zimmerman, Matthew D.; Dartois, Veronique; Gengenbacher, Martin; Olsen, David B.; Dick, Thomas
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Prescribing Patterns of Codeine and Alternative Medicines in Children in Europe
err2022-08-24
err4
errOAAI
errPlueschke, Kelly; Flynn, Robert; Hedenmalm, Karin; Deli, Aikaterini-Christina; Macia-Martinez, Miguel-Angel; Garcia-Poza, Patricia; Olsen, David; Nguyen, Pierre; Quinten, Chantal
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Identification of β-Lactams Active against Mycobacterium tuberculosis by a Consortium of Pharmaceutical Companies and Academic Institutions由制药公司和学术机构组成的财团鉴定对结核分枝杆菌具有活性的 β-内酰胺
err2022-02-22
err14
errOAAI
errGold, Ben; Zhang, Jun; Quezada, Landys Lopez; Roberts, Julia; Ling, Yan; Wood, Madeleine; Shinwari, Wasima; Goullieux, Laurent; Roubert, Christine; Fraisse, Laurent; Bacque, Eric; Lagrange, Sophie; Filoche-Romme, Bruno; Vieth, Michal; Hipskind, Philip A.; Jungheim, Louis N.; Aube, Jeffrey; Scarry, Sarah M.; McDonald, Stacey L.; Li, Kelin; Perkowski, Andrew; Nguyen, Quyen; Dartois, Veronique; Zimmerman, Matthew; Olsen, David B.; Young, Katherine; Bonnett, Shilah; Joerss, Douglas; Parish, Tanya; Boshoff, Helena, I; Arora, Kriti; Barry, Clifton E., III; Guijarro, Laura; Anca, Sara; Rullas, Joaquin; Rodriguez-Salguero, Beatriz; Martinez-Martinez, Maria S.; Porras-De Francisco, Esther; Cacho, Monica; Barros-Aguirre, David; Smith, Paul; Berthel, Steven J.; Nathan, Carl; Bates, Robert H.
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DNA-Dependent Binding of Nargenicin to DnaE1 Inhibits Replication in Mycobacterium tuberculosis
err2022-02-10
err15
errOAAI
errChengalroyen, Melissa D.; Mason, Mandy K.; Borsellini, Alessandro; Tassoni, Raffaella; Abrahams, Garth L.; Lynch, Sasha; Ahn, Yong-Mo; Ambler, Jon; Young, Katherine; Crowley, Brendan M.; Olsen, David B.; Warner, Digby F.; Barry, Clifton E., III; Boshoff, Helena I. M.; Lamers, Meindert H.; Mizrahi, Valerie
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The Tuberculosis Drug Accelerator at year 10: what have we learned?
err2021-07-05
err39
errOAAI
errAldridge, Bree B.; Barros-Aguirre, David; Barry, Clifton E., III; Bates, Robert H.; Berthel, Steven J.; Boshoff, Helena I.; Chibale, Kelly; Chu, Xin-Jie; Cooper, Christopher B.; Dartois, Veronique; Duncan, Ken; Fotouhi, Nader; Gusovsky, Fabian; Hipskind, Philip A.; Kempf, Dale J.; Lelievre, Joel; Lenaerts, Anne J.; McNamara, Case W.; Mizrahi, Valerie; Nathan, Carl; Olsen, David B.; Parish, Tanya; Petrassi, H. Michael; Pym, Alexander; Rhee, Kyu Y.; Robertson, Gregory T.; Rock, Jeremy Michael; Rubin, Eric J.; Russell, Betsy; Russell, David G.; Sacchettini, James C.; Schnappinger, Dirk; Schrimpf, Michael; Upton, Anna M.; Warner, Peter; Wyatt, Paul Graham; Yuan, Ying
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Generation of SARS-CoV-2 reporter replicon for high-throughput antiviral screening and testing用于高通量抗病毒筛选和测试的SARS-CoV-2报告复制子的生成
err2021-03-25
err71
errOAAI
errHe, Xi; Quan, Shuo; Xu, Min; Rodriguez, Silveria; Goh, Shih Lin; Wei, Jiajie; Fridman, Arthur; Koeplinger, Kenneth A.; Carroll, Steve S.; Grobler, Jay A.; Espeseth, Amy S.; Olsen, David B.; Hazuda, Daria J.; Wang, Dai
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SARS-CoV-2 tropism, entry, replication, and propagation: Considerations for drug discovery and development
err2021-02-17
err149
errOAAI
errMurgolo, Nicholas; Therien, Alex G.; Howell, Bonnie; Klein, Daniel; Koeplinger, Kenneth; Lieberman, Linda A.; Adam, Gregory C.; Flynn, Jessica; McKenna, Philip; Swaminathan, Gokul; Hazuda, Daria J.; Olsen, David B.
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Structure-Guided Drug Design of 6-Substituted Adenosine Analogues as Potent Inhibitors of Mycobacterium tuberculosis Adenosine Kinase
err2019-04-19
err11
errOAAI
errCrespo, Roberto A.; Dang, Qun; Zhou, Nian E.; Guthrie, Liam M.; Snavely, Thomas C.; Dong, Wen; Loesch, Kimberly A.; Suzuki, Takao; You, Lanying; Wang, Wei; O'Malley, Theresa; Parish, Tanya; Olsen, David B.; Sacchettini, James C.
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Discovery and Structure-Activity-Relationship Study of N-Alkyl-5-hydroxypyrimidinone Carboxamides as Novel Antitubercular Agents Targeting Decaprenylphosphoryl-β-D-ribose 2′-Oxidase
err2018-10-10
err32
errOAAI
errOh, Sangmi; Park, Yumi; Engelhart, Curtis A.; Wallach, Joshua B.; Schnappinger, Dirk; Arora, Kriti; Manikkam, Michelle; Gac, Brian; Wang, Hongwu; Murgolo, Nicholas; Olsen, David B.; Goodwin, Michael; Sutphin, Michelle; Weiner, Danielle M.; Via, Laura E.; Boshoff, Helena I. M.; Barry, Clifton E., III
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