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Diaryl-Aminoindazole with Extensive In Vitro Mycobactericidal Activity Dependent on Exposure to Reactive Nitrogen Species Warrier, Thulasi; Martinez-Hoyos, Maria; Porras De Francisco, Esther; Lenaerts, Anne J.; Gruppo, Veronica; Robertson, Gregory T.; Li, Kelin; Aube, Jeffrey; Bonnet, Isabelle; Jiang, Xiuju; Dartois, Veronique; Prideaux, Brendan; Mundhra, Shashirekha; Nathan, Carl F.; Mendoza-Losana, Alfonso 分享 收藏
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Redirecting raltitrexed from cancer cell thymidylate synthase to Mycobacterium tuberculosis phosphopantetheinyl transferase Singh, Amrita; Ottavi, Samantha; Krieger, Inna; Planck, Kyle; Perkowski, Andrew; Kaneko, Takushi; Davis, Andrew M.; Suh, Christine; Zhang, David; Goullieux, Laurent; Alex, Alexander; Roubert, Christine; Gardner, Mark; Preston, Marian; Smith, Dave M.; Ling, Yan; Roberts, Julia; Cautain, Bastien; Upton, Anna; Cooper, Christopher B.; Serbina, Natalya; Tanvir, Zaid; Mosior, John; Ouerfelli, Ouathek; Yang, Guangli; Gold, Ben S.; Rhee, Kyu Y.; Sacchettini, James C.; Fotouhi, Nader; Aube, Jeffrey; Nathan, Carl 分享 收藏
Mycobacterium tuberculosis PptT Inhibitors Based on Heterocyclic Replacements of Amidinoureas Ottavi, Samantha; Li, Kelin; Cacioppo, Jackson G. G.; Perkowski, Andrew J. J.; Ramesh, Remya; Gold, Ben S. S.; Ling, Yan; Roberts, Julia; Singh, Amrita; Zhang, David; Mosior, John; Goullieux, Laurent; Roubert, Christine; Bacque, Eric; Sacchettini, James C. C.; Nathan, Carl F. F.; Aube, Jeffrey 分享 收藏
Dual-pharmacophore artezomibs hijack the Plasmodium eubiquitin-proteasome system to kill malaria parasites while overcoming drug resistance Zhan, Wenhu; Li, Daqiang; Subramanyaswamy, Shubha Bevkal; Liu, Yi Jing; Yang, Changmei; Zhang, Hao; Harris, Jacob C.; Wang, Rong; Zhu, Songbiao; Rocha, Hedy; Sherman, Julian; Qin, Junling; Herring, Mikayla; Simwela, Nelson V.; Waters, Andrew P.; Sukenick, George; Cui, Liwang; Rodriguez, Ana; Deng, Haiteng; Nathan, Carl F.; Kirkman, Laura A.; Lin, Gang 分享 收藏
Structure-Activity Relationship Studies of Antimalarial Plasmodium Proteasome Inhibitors-Part II Zhang, Hao; Ginn, John; Zhan, Wenhu; Leung, Annie; Liu, Yi J.; Toita, Akinori; Okamoto, Rei; Wong, Tzu-Tshin; Imaeda, Toshihiro; Hara, Ryoma; Michino, Mayako; Yukawa, Takafumi; Chelebieva, Sevil; Tumwebaze, Patrick K.; Vendome, Jeremie; Beuming, Thijs; Sato, Kenjiro; Aso, Kazuyoshi; Rosenthal, Philip J.; Cooper, Roland A.; Liverton, Nigel; Foley, Michael; Meinke, Peter T.; Nathan, Carl F.; Kirkman, Laura A.; Lin, Gang 分享 收藏
Transcriptional Biomarkers of Differentially Detectable Mycobacterium tuberculosis in Patient Sputum Zainabadi, Kayvan; Saito, Kohta; Mishra, Saurabh; Walsh, Kathleen Frances; Mathurin, Laurent Daniel; Vilbrun, Stalz Charles; Ocheretina, Oksana; Pape, Jean William; Fitzgerald, Daniel W.; Nathan, Carl F.; Lee, Myung Hee 分享 收藏
Mayako Michino-Jeremie Vendome Zhang, Hao; Ginn, John; Zhan, Wenhu; Liu, Yi J.; Leung, Annie; Toita, Akinori; Okamoto, Rei; Wong, Tzu-Tshin; Imaeda, Toshihiro; Hara, Ryoma; Yukawa, Takafumi; Michino, Mayako; Vendome, Jeremie; Beuming, Thijs; Sato, Kenjiro; Aso, Kazuyoshi; Meinke, Peter T.; Nathan, Carl F.; Kirkman, Laura A.; Lin, Gang 分享 收藏
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Identification of β-Lactams Active against Mycobacterium tuberculosis by a Consortium of Pharmaceutical Companies and Academic Institutions 由制药公司和学术机构组成的财团鉴定对结核分枝杆菌具有活性的 β-内酰胺 Gold, Ben; Zhang, Jun; Quezada, Landys Lopez; Roberts, Julia; Ling, Yan; Wood, Madeleine; Shinwari, Wasima; Goullieux, Laurent; Roubert, Christine; Fraisse, Laurent; Bacque, Eric; Lagrange, Sophie; Filoche-Romme, Bruno; Vieth, Michal; Hipskind, Philip A.; Jungheim, Louis N.; Aube, Jeffrey; Scarry, Sarah M.; McDonald, Stacey L.; Li, Kelin; Perkowski, Andrew; Nguyen, Quyen; Dartois, Veronique; Zimmerman, Matthew; Olsen, David B.; Young, Katherine; Bonnett, Shilah; Joerss, Douglas; Parish, Tanya; Boshoff, Helena, I; Arora, Kriti; Barry, Clifton E., III; Guijarro, Laura; Anca, Sara; Rullas, Joaquin; Rodriguez-Salguero, Beatriz; Martinez-Martinez, Maria S.; Porras-De Francisco, Esther; Cacho, Monica; Barros-Aguirre, David; Smith, Paul; Berthel, Steven J.; Nathan, Carl; Bates, Robert H. 分享 收藏
Oxidative damage and delayed replication allow viable Mycobacterium tuberculosis to go undetected Saito, Kohta; Mishra, Saurabh; Warrier, Thulasi; Cicchetti, Nico; Mi, Jianjie; Weber, Elaina; Jiang, Xiuju; Roberts, Julia; Gouzy, Alexandre; Kaplan, Ellen; Brown, Christopher D.; Gold, Ben; Nathan, Carl 分享 收藏
Characterization of Phosphopantetheinyl Hydrolase from Mycobacterium tuberculosis Pandey, Shilpika; Singh, Amrita; Yang, Guangli; d'Andrea, Felipe B.; Jiang, Xiuju; Hartman, Travis E.; Mosior, John W.; Bourland, Ronnie; Gold, Ben; Roberts, Julia; Geiger, Annie; Tang, Su; Rhee, Kyu; Ouerfelli, Ouathek; Sacchettini, James C.; Nathan, Carl F.; Burns-Huang, Kristin 分享 收藏
Tres Cantos Open Lab: celebrating a decade of innovation in collaboration to combat endemic infectious diseases COMMENT Calderon, Felix; Ballell, Lluis; Barros, David; Bilbe, Graeme; Cammack, Nicholas; Gabarro, Raquel; Halsey, Audra; Heaton, Penny M.; Kang, Gagandeep; Mizrahi, Valerie; Nathan, Carl; Strange, Mike E.; Williams, Pauline M.; Winzeler, Elizabeth A.; Fairlamb, Alan H. 分享 收藏
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Characterization of Differentially Detectable Mycobacterium tuberculosis in the Sputum of Subjects with Drug-Sensitive or Drug-Resistant Tuberculosis before and after Two Months of Therapy Zainabadi, Kayvan; Walsh, Kathleen Frances; Vilbrun, Stalz Charles; Mathurin, Laurent Daniel; Lee, Myung Hee; Saito, Kohta; Mishra, Saurabh; Ocheretina, Oksana; Pape, Jean William; Nathan, Carl; Fitzgerald, Daniel W. 分享 收藏
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The Tuberculosis Drug Accelerator at year 10: what have we learned? Aldridge, Bree B.; Barros-Aguirre, David; Barry, Clifton E., III; Bates, Robert H.; Berthel, Steven J.; Boshoff, Helena I.; Chibale, Kelly; Chu, Xin-Jie; Cooper, Christopher B.; Dartois, Veronique; Duncan, Ken; Fotouhi, Nader; Gusovsky, Fabian; Hipskind, Philip A.; Kempf, Dale J.; Lelievre, Joel; Lenaerts, Anne J.; McNamara, Case W.; Mizrahi, Valerie; Nathan, Carl; Olsen, David B.; Parish, Tanya; Petrassi, H. Michael; Pym, Alexander; Rhee, Kyu Y.; Robertson, Gregory T.; Rock, Jeremy Michael; Rubin, Eric J.; Russell, Betsy; Russell, David G.; Sacchettini, James C.; Schnappinger, Dirk; Schrimpf, Michael; Upton, Anna M.; Warner, Peter; Wyatt, Paul Graham; Yuan, Ying 分享 收藏