未登录
分享
收藏Development of Practical and Scalable Synthetic Route for 1-(2,2,2-Trifluoroethyl)cyclopropane-1-carboxylic Acid
Karmakar, Sukhen; Ayothiraman, Rajaram; Nandhagopal, Sundar; Dolas, Zulelal; Silamkoti, Arundutt; Venu, Alla; Jami, Srinivasarao; Venkataramani, Arvind; Lakshminarasimhan, Thirumalai; Mukherjee, Sabuj; Gupta, Anuradha; Mathur, Arvind; Melendez Matos, Jeishla L.; Hale, Ian; Eastgate, Martin D.; Gonzalez-Bobes, Francisco
分享
收藏Development of a Mild and Efficient Process for Ir-Catalyzed N-Alkylation of 4-Bromopyridin-2-amine with a Primary Alcohol via Borrowing Hydrogen
Nimmagadda, Krishna; Kalidindi, Srinivas; Bondigela, Siva Sankar; Korapati, Satish; Dasgupta, Debottam; Malik, Noormohamed Abdul; Rao, Prakasa; Maity, Prantik; Coombs, John R.; Hay, Michael; Simmons, Eric M.; Mukherjee, Sabuj; Vaidyanathan, Rajappa; Eastgate, Martin D.; Gonzalez-Bobes, Francisco
分享
收藏Stereocontrolled Radical Thiophosphorylation立体控制自由基硫代磷酸化
Nassir, Molhm; Ociepa, Michal; Zhang, Hai-Jun; Grant, Lauren N.; Simmons, Bryan J.; Oderinde, Martins S.; Kawamata, Yu; Cauley, Anthony N.; Schmidt, Michael A.; Eastgate, Martin D.; Baran, Phil S.
分享
收藏Toward the Development of a Manufacturing Process for Milvexian: Scale-Up Synthesis of the Side Chain
Wagschal, Simon; Broggini, Diego; Cao, Trung D. C.; Schleiss, Pascal; Paun, Kristian; Steiner, Jessica; Merk, Anna-Lena; Harsdorf, Joachim; Fiedler, Winfried; Schirling, Stefan; Hock, Sven; Strittmatter, Tobias; Dijkmans, Jan; Vervest, Ivan; Van Hoegaerden, Tim; Egle, Brecht; Mower, Matthew P.; Liu, Zhi; Cao, Zhiyong; He, Xiaoning; Chen, Lei; Qin, Lei; Tan, Hongyu; Yan, Jun; Cuniere, Nicolas Lucien; Wei, Carolyn S.; Vuyyuru, Venkata; Ayothiraman, Rajaram; Rangaswamy, Sundaramurthy; Jaleel, Mohamed; Vaidyanathan, Rajappa; Eastgate, Martin D.; Klep, Richard; Benhaim, Cyril; Vogels, Ilse; Peeters, Koen; Lemaire, Sebastien
分享
收藏Alternative Approach to the Large-Scale Synthesis of the Densely Functionalized Pyrrolidone BMT-415200
Rakshit, Souvik; Sathasivam, Shunmugaraj; Reddy, Raghurami; Rao, Saladi, V; Shekarappa, Vijaykumar; Kandasamy, Moorthy; Jaleel, Mohamed; Murugan, Saravanan; Bhat, Anuradha; Subramani, Tamilarasan; Lakshminarasimhan, Thirumalai; Gangu, Aravind; Wisniewski, Steven R.; Kopp, Nathaniel; Hale, Ian; Stevens, Jason M.; Rosso, Victor W.; Eastgate, Martin D.; Vaidyanathan, Rajappa
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏Structurally Diverse Bench-Stable Nickel(0) Pre-Catalysts: A Practical Toolkit for In Situ Ligation Protocols结构多样的台式稳定镍 (0) 预催化剂: 用于原位连接方案的实用工具包
Tran, Van T.; Kim, Nana; Rubel, Camille Z.; Wu, Xiangyu; Kang, Taeho; Jankins, Tanner C.; Li, Zi-Qi; Joannou, Matthew V.; Ayers, Sloan; Gembicky, Milan; Bailey, Jake; Sturgell, Emily J.; Sanchez, Brittany B.; Chen, Jason S.; Lin, Song; Eastgate, Martin D.; Wisniewski, Steven R.; Engle, Keary M.
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏Mild and Chemoselective Phosphorylation of Alcohols Using a Ψ-Reagent
Ociepa, Michal; Knouse, Kyle W.; He, David; Vantourout, Julien C.; Flood, Dillon T.; Padial, Natalia M.; Chen, Jason S.; Sanchez, Brittany B.; Sturgell, Emily J.; Zheng, Bin; Qiu, Shenjie; Schmidt, Michael A.; Eastgate, Martin D.; Baran, Phil S.
分享
收藏Scalable Asymmetric Synthesis of the All Cis Triamino Cyclohexane Core of BMS-813160
La Cruz, Thomas E.; Gonzalez-Bobes, Francisco; Eastgate, Martin D.; Sfouggatakis, Chris; Zheng, Bin; Kopp, Nathaniel; Xiao, Yi; Fan, Yu; Galindo, Kay A.; Pathirana, Charles; Galella, Michael A.; Deerberg, Joerg
分享
收藏
分享
收藏P(III) vs P(V): A P(V) Reagent for Thiophosphoramidate Linkages and Application to an Asymmetric Synthesis of a Cyclic Dinucleotide STING Agonist
Zheng, Bin; Hang, Chao; Zhu, Jason; Purdum, Geoffrey E.; Sezen-Edmonds, Melda; Treitler, Daniel S.; Yu, Miao; Yuan, Changxia; Zhu, Ye; Freitag, Adam; Guo, Siwei; Zhu, Guanghui; Hritzko, Ben; Paulson, James; Shackman, Jonathan G.; He, Brian L.; Fu, Weiqing; Tai, Hua Chia; Ayers, Sloan; Park, Hyunsoo; Eastgate, Martin D.; Cohen, Ben; Rogers, Amanda; Wang, Qinggang; Schmidt, Michael A.
分享
收藏Development of a Scalable Synthetic Route to BMS-986251, Part 2: Synthesis of the Tricyclic Core and the API
Kalidindi, Srinivas; Gangu, Aravind S.; Kuppusamy, Sankar; Sathasivam, Shunmugaraj; Shekarappa, Vijaykumar; Murugan, Saravanan; Bondigela, Sivasankar; Kandasamy, Moorthy; Ghanta, Kishore; Vinodini, Arun; Shrikant, Abhishek; Ramachandran, Ravikumar; Gallagher, William P.; Kopp, Nathaniel; Gonzalez-Bobes, Francisco; Eastgate, Martin D.; Vaidyanathan, Rajappa
分享
收藏