未登录 Feasibility of pharmacy-based research opportunity to enhance community testing and surveillance 基于药房的研究机会在增强社区检测和监测方面的可行性 Venditto, Vincent J.; Hudspeth, Brooke; Freeman, Patricia R.; Qasrawi, Lien; Guy, R. Kiplin; Farley, Victoria H.; Johnson, Royce A.; Freeman, Edward; Henson, David; Marion, Ryan; Wagner, Sheridan B.; Doratt, Brianna M.; Messaoudi-Powers, Ilhem 分享 收藏
Antitrypanosomal Chloronitrobenzamides Carrillo, Angela K.; Kadayat, Tara Man; Hwang, Jong Yeon; Chen, Yizhe; Zhu, Fangyi; Holbrook, Gloria; Gillingwater, Kirsten; Connelly, Michele C.; Yang, Lei; Kaiser, Marcel; Guy, R. Kiplin 分享 收藏
Optimization of Orally Bioavailable Antileishmanial 2,4,5-Trisubstituted Benzamides Kim, Ho Shin; Ortiz, Diana; Kadayat, Tara Man; Fargo, Corinne M.; Hammill, Jared T.; Chen, Yizhe; Rice, Amy L.; Begley, Kristin L.; Shoeran, Gaurav; Pistel, William; Yates, Phillip A.; Sanchez, Marco A.; Landfear, Scott M.; Guy, R. Kiplin 分享 收藏
Proteasome inhibition targets the KMT2A transcriptional complex in acute lymphoblastic leukemia (vol 14, 809, 2023) Kamens, Jennifer L.; Nance, Stephanie; Koss, Cary; Xu, Beisi; Cotton, Anitria; Lam, Jeannie W.; Garfinkle, Elizabeth A. R.; Nallagatla, Pratima; Smith, Amelia M. R.; Mitchell, Sharnise; Ma, Jing; Currier, Duane; Wright, William C.; Kavdia, Kanisha; Pagala, Vishwajeeth R.; Kim, Wonil; Wallace, LaShanale M.; Cho, Ji-Hoon; Fan, Yiping; Seth, Aman; Twarog, Nathaniel; Choi, John K.; Obeng, Esther A.; Hatley, Mark E.; Metzger, Monika L.; Inaba, Hiroto; Jeha, Sima; Rubnitz, Jeffrey E.; Peng, Junmin; Chen, Taosheng; Shelat, Anang A.; Guy, R. Kiplin; Gruber, Tanja A. 分享 收藏
Proteasome inhibition targets the KMT2A transcriptional complex in acute lymphoblastic leukemia Kamens, Jennifer L.; Nance, Stephanie; Koss, Cary; Xu, Beisi; Cotton, Anitria; Lam, Jeannie W.; Garfinkle, Elizabeth A. R.; Nallagatla, Pratima; Smith, Amelia M. R.; Mitchell, Sharnise; Ma, Jing; Currier, Duane; Wright, William C.; Kavdia, Kanisha; Pagala, Vishwajeeth R.; Kim, Wonil; Wallace, LaShanale M.; Cho, Ji-Hoon; Fan, Yiping; Seth, Aman; Twarog, Nathaniel; Choi, John K.; Obeng, Esther A.; Hatley, Mark E.; Metzger, Monika L.; Inaba, Hiroto; Jeha, Sima; Rubnitz, Jeffrey E.; Peng, Junmin; Chen, Taosheng; Shelat, Anang A.; Guy, R. Kiplin; Gruber, Tanja A. 分享 收藏
Combining SJ733, an oral ATP4 inhibitor of Plasmodium falciparum, with the pharmacokinetic enhancer cobicistat: An innovative approach in antimalarial drug development Gaur, Aditya H.; Panetta, John C.; Smith, Amber M.; Dallas, Ronald H.; FreemanIII, Burgess B.; Stewart, Tracy B.; Tang, Li; John, Elizabeth; Branum, Kristen C.; Patel, Nehali D.; Ost, Shelley; Heine, Ryan N.; Richardson, Julie L.; Hammill, Jared T.; Bebrevska, Lidiya; Gusovsky, Fabian; Maki, Noritsugu; Yanagi, Toshiharu; Flynn, Patricia M.; McCarthy, James S.; Chalon, Stephan; Guy, R. Kiplin 分享 收藏
Amino-Substituted 3-Aryl- and 3-Heteroarylquinolines as Potential Antileishmanial Agents Hammill, Jared T.; Sviripa, Vitaliy M.; Kril, Liliia M.; Ortiz, Diana; Fargo, Corinne M.; Kim, Ho Shin; Chen, Yizhe; Rector, Jonah; Rice, Amy L.; Domagalska, Malgorzata A.; Begley, Kristin L.; Liu, Chunming; Rangnekar, Vivek M.; Dujardin, Jean-Claude; Watt, David S.; Landfear, Scott M.; Guy, R. Kiplin 分享 收藏
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Evaluation of 1,1-cyclopropylidene as a thioether isostere in the 4-thio- thienopyrimidine (TTP) series of antimalarials Barrows, Robert D.; Hammill, Jared T.; Tran, Michael C.; Falade, Mofolusho O.; Rice, Amy L.; Davis, Christopher W.; Emge, Thomas J.; Rablen, Paul R.; Guy, R. Kiplin; Knapp, Spencer 分享 收藏
Synthesis and Structure-Activity Relationship of Dual-Stage Antimalarial Pyrazolo[3,4-b]pyridines Eagon, Scott; Hammill, Jared T.; Sigal, Martina; Ahn, Kevin J.; Tryhorn, Julia E.; Koch, Grant; Belanger, Briana; Chaplan, Cory A.; Loop, Lauren; Kashtanova, Anna S.; Yniguez, Kenya; Lazaro, Horacio; Wilkinson, Steven P.; Rice, Amy L.; Falade, Mofolusho O.; Takahashi, Rei; Kim, Katie; Cheung, Ashley; DiBernardo, Celine; Kimball, Joshua J.; Winzeler, Elizabeth A.; Eribez, Korina; Mittal, Nimisha; Gamo, Francisco-Javier; Crespo, Benigno; Churchyard, Alisje; Garcia-Barbazan, Irene; Baum, Jake; Anderson, Marc O.; Laleu, Benoit; Guy, R. Kiplin 分享 收藏
Bromodomain-Selective BET Inhibitors Are Potent Antitumor Agents against MYC-Driven Pediatric Cancer Slavish, P. Jake; Chi, Liying; Yun, Mi-Kyung; Tsurkan, Lyudmila; Martinez, Nancy E.; Jonchere, Barbara; Chai, Sergio C.; Connelly, Michele; Waddell, M. Brett; Das, Sourav; Neale, Geoffrey; Li, Zhenmei; Shadrick, William R.; Olsen, Rachelle R.; Freeman, Kevin W.; Low, Jonathan A.; Price, Jeanine E.; Young, Brandon M.; Bharatham, Nagakumar; Boyd, Vincent A.; Yang, Jun; Lee, Richard E.; Morfouace, Marie; Roussel, Martine F.; Chen, Taosheng; Savic, Daniel; Guy, R. Kiplin; White, Stephen W.; Shelat, Anang A.; Potter, Philip M. 分享 收藏
Safety, tolerability, pharmacokinetics, and antimalarial efficacy of a novel Plasmodium falciparum ATP4 inhibitor SJ733: a first-in-human and induced blood-stage malaria phase 1a/b trial Gaur, Aditya H.; McCarthy, James S.; Panetta, John C.; Dallas, Ronald H.; Woodford, John; Tang, Li; Smith, Amber M.; Stewart, Tracy B.; Branum, Kristen C.; Freeman, Burgess B., III; Patel, Nehali D.; John, Elizabeth; Chalon, Stephan; Ost, Shelley; Heine, Ryan N.; Richardson, Julie L.; Christensen, Robbin; Flynn, Patricia M.; Van Gessel, Yvonne; Mitasev, Branko; Moehrle, Joerg J.; Gusovsky, Fabian; Bebrevska, Lidiya; Guy, R. Kiplin 分享 收藏
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Ventromorphins: A New Class of Small Molecule Activators of the Canonical BMP Signaling Pathway (vol 12, pg 2436, 2017) Genthe, Jamie R.; Min, Jaeki; Farmer, Dana M.; Shelat, Anang A.; Grenet, Jose A.; Lin, Wenwei; Finkelstein, David; Vrijens, Karen; Chen, Taosheng; Guy, R. Kiplin; Clements, Wilson K.; Roussel, Martine F. 分享 收藏
A high-throughput screen indicates gemcitabine and JAK inhibitors may be useful for treating pediatric AML Drenberg, Christina D.; Shelat, Anang; Dang, Jinjun; Cotton, Anitria; Orwick, Shelley J.; Li, Mengyu; Jeon, Jae Yoon; Fu, Qiang; Buelow, Daelynn R.; Pioso, Marissa; Hu, Shuiying; Inaba, Hiroto; Ribeiro, Raul C.; Rubnitz, Jeffrey E.; Gruber, Tanja A.; Guy, R. Kiplin; Baker, Sharyn D. 分享 收藏
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Identification of Toll-like receptor signaling inhibitors based on selective activation of hierarchically acting signaling proteins Ippagunta, Sirish K.; Pollock, Julie A.; Sharma, Naina; Lin, Wenwei; Chen, Taosheng; Tawaratsumida, Kazuki; High, Anthony A.; Min, Jaeki; Chen, Yizhe; Guy, R. Kiplin; Redecke, Vanessa; Katzenellenbogen, John A.; Hacker, Hans 分享 收藏
Cysteine modifiers suggest an allosteric inhibitory site on the CAL PDZ domain Zhao, Yu; Cushing, Patrick R.; Smithson, David C.; Pellegrini, Maria; Pletnev, Alexandre A.; Al-Ayyoubi, Sahar; Grassetti, Andrew V.; Gerber, Scott A.; Guy, R. Kiplin; Madden, Dean R. 分享 收藏
Cysteine modification reveals an allosteric inhibitory site on the CAL PDZ domain (vol 38, BSR20180231, 2018) Zhao, Yu; Cushing, Patrick R.; Smithson, David C.; Pellegrini, Maria; Pletnev, Alexandre A.; Al-Ayyoubi, Sahar; Grassetti, Andrew V.; Gerber, Scott A.; Guy, R. Kiplin; Madden, Dean R. 分享 收藏