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Christophe L. M. J. Verlinde

University of Washington

48H指数
199论文数
7.7K被引数
收录论文 65
发表时间
Spontaneous Selection of Cryptosporidium Drug Resistance in a Calf Model of Infection
err2021-05-18
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errHasan, Muhammad M.; Stebbins, Erin E.; Choy, Robert K. M.; Gillespie, J. Robert; de Hostos, Eugenio L.; Miller, Peter; Mushtaq, Aisha; Ranade, Ranae M.; Teixeira, Jose E.; Verlinde, Christophe L. M. J.; Sateriale, Adam; Zhang, Zhongsheng; Osbourn, Damon M.; Griggs, David W.; Fan, Erkang; Buckner, Frederick S.; Huston, Christopher D.
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Repurposing Infectious Disease Hits as Anti-Cryptosporidium Leads
err2021-03-19
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errHulverson, Matthew A.; Choi, Ryan; McCloskey, Molly C.; Whitman, Grant R.; Ojo, Kayode K.; Michaels, Samantha A.; Somepalli, Mastanbabu; Love, Melissa S.; McNamara, Case W.; Rabago, Lesley M.; Barrett, Lynn K.; Verlinde, Christophe L. M. J.; Arnold, Samuel L. M.; Striepen, Boris; Jimenez-Alfaro, Dolores; Ballell, Lluis; Fernandez, Elena; Greenwood, M. Nicole; de las Heras, Laura; Calderon, Felix; Van Voorhis, Wesley C.
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Structure-guided discovery of selective methionyl-tRNA synthetase inhibitors with potent activity against Trypanosoma brucei
err2020-01-01
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errZhang, Zhongsheng; Barros-Alvarez, Ximena; Gillespie, J. Robert; Ranade, Ranae M.; Huang, Wenlin; Shibata, Sayaka; Molasky, Nora M. R.; Faghih, Omeed; Mushtaq, Aisha; Choy, Robert K. M.; de Hostos, Eugenio; Hol, Wim G. J.; Verlinde, Christophe L. M. J.; Buckner, Frederick S.; Fan, Erkang
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Optimization of Methionyl tRNA-Synthetase Inhibitors for Treatment of Cryptosporidium Infection
err2019-04-01
err43
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errBuckner, Frederick S.; Ranade, Ranae M.; Gillespie, J. Robert; Shibata, Sayaka; Hulverson, Matthew A.; Zhang, Zhongsheng; Huang, Wenlin; Choi, Ryan; Verlinde, Christophe L. M. J.; Hol, Wim G. J.; Ochida, Atsuko; Akao, Yuichiro; Choy, Robert K. M.; Van Voorhis, Wesley C.; Arnold, Sam L. M.; Jumani, Rajiv S.; Huston, Christopher D.; Fan, Erkang
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Development of Methionyl-tRNA Synthetase Inhibitors as Antibiotics for Gram-Positive Bacterial Infections
err2017-11-01
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errFaghih, Omeed; Zhang, Zhongsheng; Ranade, Ranae M.; Gillespie, J. Robert; Creason, Sharon A.; Huang, Wenlin; Shibata, Sayaka; Barros-Alvarez, Ximena; Verlinde, Christophe L. M. J.; Hol, Wim G. J.; Fan, Erkang; Buckner, Frederick S.
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Leishmania donovani tyrosyl-tRNA synthetase structure in complex with a tyrosyl adenylate analog and comparisons with human and protozoan counterparts
err2017-07-01
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errBarros-Alvarez, Ximena; Kerchner, Keshia M.; Koh, Cho Yeow; Turley, Stewart; Pardon, Els; Steyaert, Jan; Ranade, Ranae M.; Gillespie, J. Robert; Zhang, Zhongsheng; Verlinde, Christophe L. M. J.; Fan, Erkang; Buckner, Frederick S.; Hol, Wim G. J.
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Structure-guided design of novel Trypanosoma brucei Methionyl-tRNA synthetase inhibitors
err2016-11-01
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errHuang, Wenlin; Zhang, Zhongsheng; Barros-Alvarez, Ximena; Koh, Cho Yeow; Ranade, Ranae M.; Gillespie, J. Robert; Creason, Sharon A.; Shibata, Sayaka; Verlinde, Christophe L. M. J.; Hol, Wim G. J.; Buckner, Frederick S.; Fan, Erkang
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5-Fluoroimidazo[4,5-b]pyridine Is a Privileged Fragment That Conveys Bioavailability to Potent Trypanosomal Methionyl-tRNA Synthetase Inhibitors
err2016-04-11
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errZhang, Zhongsheng; Koh, Cho Yeow; Ranade, Ranae M.; Shibata, Sayaka; Gillespie, J. Robert; HuIverson, Matthew A.; Huang, Wenlin; Nguyen, Jasmine; Pendem, Nagendar; Gelb, Michael H.; Verlinde, Christophe L. M. J.; Hol, Wim G. J.; Buckner, Frederick S.; Fan, Erkang
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Inhibitors of Methionyl-tRNA Synthetase Have Potent Activity against Giardia intestinalis Trophozoites
err2015-11-01
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errRanade, Ranae M.; Zhang, Zhongsheng; Gillespie, J. Robert; Shibata, Sayaka; Verlinde, Christophe L. M. J.; Hol, Wim G. J.; Fan, Erkang; Buckner, Frederick S.
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Structures of Trypanosoma brucei Methionyl-tRNA Synthetase with Urea-Based Inhibitors Provide Guidance for Drug Design against Sleeping Sickness
err2014-04-17
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errKoh, Cho Yeow; Kim, Jessica E.; Wetzel, Allan B.; de van der Schueren, Will J.; Shibata, Sayaka; Ranade, Ranae M.; Liu, Jiyun; Zhang, Zhongsheng; Gillespie, J. Robert; Buckner, Frederick S.; Verlinde, Christophe L. M. J.; Fan, Erkang; Hol, Wim G. J.
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Development of potent and selective Plasmodium falciparum calcium-dependent protein kinase 4 (PfCDPK4) inhibitors that the transmission of malaria to mosquitoes
err2014-03-01
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errVidadala, Rama Subba Rao; Ojo, Kayode K.; Johnson, Steven M.; Zhang, Zhongsheng; Leonard, Stephen E.; Mitra, Arinjay; Choi, Ryan; Reid, Molly C.; Keyloun, Katelyn R.; Fox, Anna M. W.; Kennedy, Mark; Silver-Brace, Tiffany; Hume, Jen C. C.; Kappe, Stefan; Verlinde, Christophe L. M. J.; Fan, Erkang; Merritt, Ethan A.; Van Voorhis, Wesley C.; Maly, Dustin J.
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Potent and Selective Inhibitors of CDPK1 from T. gondii and C. parvum Based on a 5-Aminopyrazole-4-carboxamide Scaffold
err2013-11-20
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errZhang, Zhongsheng; Ojo, Kayode K.; Vidadala, RamaSubbaRao; Huang, Wenlin; Geiger, Jennifer A.; Scheele, Suzanne; Choi, Ryan; Reid, Molly C.; Keyloun, Katelyn R.; Rivas, Kasey; Siddaramaiah, Latha Kallur; Comess, Kenneth M.; Robinson, Kenneth P.; Merta, Philip J.; Kifle, Lemma; Hol, Wim G. J.; Parsons, Marilyn; Merritt, Ethan A.; Maly, Dustin J.; Verlinde, Christophe L. M. J.; Van Voorhis, Wesley C.; Fan, Erkang
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A Specific Inhibitor of PfCDPK4 Blocks Malaria Transmission: Chemical-genetic Validation
err2013-10-10
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errOjo, Kayode K.; Eastman, Richard T.; Vidadala, RamaSubbaRao; Zhang, Zhongsheng; Rivas, Kasey L.; Choi, Ryan; Lutz, Justin D.; Reid, Molly C.; Fox, Anna M. W.; Hulverson, Matthew A.; Kennedy, Mark; Isoherranen, Nina; Kim, Laura M.; Comess, Kenneth M.; Kempf, Dale J.; Verlinde, Christophe L. M. J.; Su, Xin-zhuan; Kappe, Stefan H. I.; Maly, Dustin J.; Fan, Erkang; Van Voorhis, Wesley C.
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Induced Resistance to Methionyl-tRNA Synthetase Inhibitors in Trypanosoma brucei Is Due to Overexpression of the Target
err2013-07-01
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errRanade, Ranae M.; Gillespie, J. Robert; Shibata, Sayaka; Verlinde, Christophe L. M. J.; Fan, Erkang; Hol, Wim G. J.; Buckner, Frederick S.
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Pharmacological Characterization, Structural Studies, and In Vivo Activities of Anti-Chagas Disease Lead Compounds Derived from Tipifarnib
err2012-09-01
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errBuckner, Frederick S.; Bahia, Maria Terezinha; Suryadevara, Praveen Kumar; White, Karen L.; Shackleford, David M.; Chennamaneni, Naveen Kumar; Hulverson, Matthew A.; Laydbak, Joy U.; Chatelain, Eric; Scandale, Ivan; Verlinde, Christophe L. M. J.; Charman, Susan A.; Lepesheva, Galina I.; Gelb, Michael H.
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Urea-Based Inhibitors of Trypanosoma brucei Methionyl-tRNA Synthetase: Selectivity and in Vivo Characterization布氏锥虫甲硫氨酰-tRNA合成酶的尿素抑制剂: 选择性和体内表征
err2012-07-11
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errShibata, Sayaka; Gillespie, J. Robert; Ranade, Ranae M.; Koh, Cho Yeow; Kim, Jessica E.; Laydbak, Joy U.; Zucker, Frank H.; Hol, Wim G. J.; Verlinde, Christophe L. M. J.; Buckner, Frederick S.; Fan, Erkang
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Transmission of malaria to mosquitoes blocked by bumped kinase inhibitors
err2012-06-01
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errOjo, Kayode K.; Pfander, Claudia; Mueller, Natascha R.; Burstroem, Charlotte; Larson, Eric T.; Bryan, Cassie M.; Fox, Anna M. W.; Reid, Molly C.; Johnson, Steven M.; Murphy, Ryan C.; Kennedy, Mark; Mann, Henning; Leibly, David J.; Hewitt, Stephen N.; Verlinde, Christophe L. M. J.; Kappe, Stefan; Merritt, Ethan A.; Maly, Dustin J.; Billker, Oliver; Van Voorhis, Wesley C.
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Multiple Determinants for Selective Inhibition of Apicomplexan Calcium-Dependent Protein Kinase CDPK1
err2012-03-13
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errLarson, Eric T.; Ojo, Kayode K.; Murphy, Ryan C.; Johnson, Steven M.; Zhang, Zhongsheng; Kim, Jessica E.; Leibly, David J.; Fox, Anna M. W.; Reid, Molly C.; Dale, Edward J.; Perera, B. Gayani K.; Kim, Jae; Hewitt, Stephen N.; Hol, Wim G. J.; Verlinde, Christophe L. M. J.; Fan, Erkang; Van Voorhis, Wesley C.; Maly, Dustin J.; Merritt, Ethan A.
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Screening a fragment cocktail library using ultrafiltration使用超滤筛选片段鸡尾酒库
err2011-07-13
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errShibata, Sayaka; Zhang, Zhongsheng; Korotkov, Konstantin V.; Delarosa, Jaclyn; Napuli, Alberto; Kelley, Angela M.; Mueller, Natasha; Ross, Jennifer; Zucker, Frank H.; Buckner, Frederick S.; Merritt, Ethan A.; Verlinde, Christophe L. M. J.; Van Voorhis, Wesley C.; Hol, Wim G. J.; Fan, Erkang
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Selective Inhibitors of Methionyl-tRNA Synthetase Have Potent Activity against Trypanosoma brucei Infection in Mice
err2011-05-01
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errShibata, Sayaka; Gillespie, J. Robert; Kelley, Angela M.; Napuli, Alberto J.; Zhang, Zhongsheng; Kovzun, Kuzma V.; Pefley, Ranae M.; Lam, Jocelyn; Zucker, Frank H.; Van Voorhis, Wesley C.; Merritt, Ethan A.; Hol, Wim G. J.; Verlinde, Christophe L. M. J.; Fan, Erkang; Buckner, Frederick S.
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