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收藏Design, synthesis and biological evaluation of bisnoralcohol derivatives as novel IRF4 inhibitors for the treatment of multiple myeloma
Zhang, Jing-Zan; Zhang, Lin; Ding, Xin; Wu, Min; Zhang, De-Jie; Wu, Yujie; Liu, Mingyao; Li, Chen-Chen; Yi, Zhengfang; Qiu, Wen-Wei
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收藏IRE1α inhibitor reduces cisplatin resistance in ovarian cancer by modulating IRE1α/XBP1 pathway
Lv, Shiyi; Zhang, Lin; Wu, Min; Zhu, Shuangshuang; Wang, Yixue; Liu, Layang; Li, Yunxuan; Zhang, Ting; Wu, Yujie; Chen, Huang; Liu, Mingyao; Yi, Zhengfang
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收藏A Small-Molecule BCL6 Inhibitor as an Anti-Proliferative Agent for Diffuse Large B-Cell Lymphoma一种小分子BCL6抑制剂作为弥漫性大b细胞淋巴瘤的抗增殖剂
Xing, Yajing; Guo, Weikai; Wu, Min; Xie, Jiuqing; Huang, Dongxia; Hu, Pan; Zhou, Miaoran; Zhang, Lin; Zhong, Yadong; Liu, Mingyao; Chen, Yihua; Yi, Zhengfang
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收藏Remodeling the immune microenvironment for gastric cancer therapy through antagonism of prostaglandin E2 receptor 4
Guo, Mengmeng; Hu, Pan; Xie, Jiayi; Tang, Kefu; Hu, Shixiu; Sun, Jialiang; He, Yundong; Li, Jing; Lu, Weiqiang; Liu, Huirong; Liu, Mingyao; Yi, Zhengfang; Peng, Shihong
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收藏Targeting STAT3 by a small molecule suppresses pancreatic cancer progression (vol 40, pg 1440, 2021)
Chen, Huang; Bian, Aiwu; Yang, Lian-fang; Yin, Xuan; Wang, Jie; Ti, Chaowen; Miao, Ying; Peng, Shihong; Xu, Shifen; Liu, Mingyao; Qiu, Wen-Wei; Yi, Zhengfang
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收藏Discovery of the Highly Selective and Potent STAT3 Inhibitor for Pancreatic Cancer Treatment发现用于胰腺癌治疗的高选择性和有效的STAT3抑制剂
Chen, Huang; Bian, Aiwu; Zhou, Wenbo; Miao, Ying; Ye, Jiangnan; Li, Jiahui; He, Peng; Zhang, Qiansen; Sun, Yue; Sun, Zhenliang; Ti, Chaowen; Chen, Yihua; Yi, Zhengfang; Liu, Mingyao
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收藏WB518, a novel STAT3 inhibitor, effectively alleviates IMQ and TPA-induced animal psoriasis by inhibiting STAT3 phosphorylation and Keratin 17新型STAT3抑制剂WB518通过抑制STAT3磷酸化和角蛋白17有效缓解IMQ和TPA诱导的动物银屑病
Ti, Chaowen; Chen, Huang; Zhou, Wenbo; Bian, Aiwu; Hu, Pan; Miao, Ying; Shao, Ting; Liu, Mingyao; Chen, Yihua; Yi, Zhengfang
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收藏Discovery of a Highly Potent and Selective MYOF Inhibitor with Improved Water Solubility for the Treatment of Gastric Cancer发现一种具有改善水溶性的高效选择性MYOF抑制剂,用于治疗胃癌
Gu, Haijun; Zhang, Ting; Guan, Tian; Wu, Min; Li, Shen; Li, Yunqi; Guo, Mengmeng; Zhang, Lin; Peng, Yangrui; Mi, Dazhao; Liu, Mingyao; Yi, Zhengfang; Chen, Yihua
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收藏A small molecule BCL6 inhibitor as chemosensitizers in acute myeloid leukemia小分子BCL6抑制剂作为急性髓系白血病的化学增敏剂
Zhang, Lin; Wu, Min; Guo, Weikai; Zhu, Shuangshuang; Li, Shen; Lv, Shiyi; Li, Yan; Liu, Layang; Xing, Yajing; Chen, Huang; Liu, Mingyao; Peng, Shihong; Chen, Yihua; Yi, Zhengfang
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收藏Combined treatment of disulfiram with PARP inhibitors suppresses ovarian cancer双硫仑与PARP抑制剂联合治疗可抑制卵巢癌
Tang, Bin; Wu, Min; Zhang, Lin; Jian, Shuyi; Lv, Shiyi; Lin, Tongyuan; Zhu, Shuangshuang; Liu, Layang; Wang, Yixue; Yi, Zhengfang; Jiang, Feiyun
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收藏Discovery of 1,5-diaryl-1,2,4-triazole derivatives as myoferlin inhibitors and their antitumor effects in pancreatic cancer1,5-二芳基-1,2,4-三唑衍生物作为myoferlin抑制剂的发现及其在胰腺癌中的抗肿瘤作用
Gu, Haijun; Zhang, Ting; Li, Yunqi; He, Yuan; Guan, Tian; Kan, Weiqiong; He, Peng; Yi, Zhengfang; Chen, Yihua
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收藏Discovery of a Novel Potent STAT3 Inhibitor HP590 with Dual p-Tyr705/Ser727 Inhibitory Activity for Gastric Cancer Treatment
He, Peng; Miao, Ying; Sun, Yue; Bian, Aiwu; Jin, Wangrui; Ye, Jiangnan; Chen, Huang; He, Jia; Peng, Yangrui; Gu, Haijun; Liu, Mingyao; Yi, Zhengfang; Chen, Yihua
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收藏Discovery of 2-Amino-3-cyanothiophene Derivatives as PotentSTAT3 Inhibitors for the Treatment of Osteosarcoma Growth and Metastasis
Jin, Wangrui; Zhang, Tao; Zhou, Wenbo; He, Peng; Sun, Yue; Hu, Shijia; Chen, Huang; Ma, Xinglong; Peng, Yangrui; Yi, Zhengfang; Liu, Mingyao; Chen, Yihua
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收藏A novel small-molecule activator of unfolded protein response suppresses castration-resistant prostate cancer growth
Chen, Huang; Miao, Ying; Bian, Aiwu; Ye, Jiangnan; Wang, Jing; Cong, Xiaonan; Jian, Shuyi; Yi, Zhengfang; Liang, Lin; Sun, Zhenliang; Yang, Fan; Ding, Tao
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收藏An orally available small molecule BCL6 inhibitor effectively suppresses diffuse large B cell lymphoma cells growth in vitro and in vivo一种可口服的小分子BCL6抑制剂可有效抑制体内和体外弥漫性大b细胞淋巴瘤细胞的生长
Xing, Yajing; Guo, Weikai; Wu, Min; Xie, Jiuqing; Huang, Dongxia; Hu, Pan; Zhou, Miaoran; Zhang, Lin; Zhang, Qiansen; Wang, Peili; Wang, Xin; Wang, Guixue; Wu, Huangan; Zhou, Cili; Chen, Yihua; Liu, Mingyao; Yi, Zhengfang; Sun, Zhenliang
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