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收藏Targeting PSMD14 combined with arachidonic acid induces synthetic lethality via FADS1 m6A modification in triple-negative breast cancer靶向PSMD14联合花生四烯酸通过FADS1 m6A修饰在 triple-negative breast cancer 中诱导合成致死效应
Yu, Yuanhang; Hu, Jin; Wang, Wenwen; Lei, Hao; Xi, Zihan; Zhang, Peiyi; Zhao, Ende; Lu, Chong; Chen, Hengyu; Liu, Chunping; Li, Lei
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收藏A novel regimen for pancreatic ductal adenocarcinoma targeting MEK, BCL-xL, and EGFR
Han, Song; Tushoski-Aleman, Gerik W.; Zhang, Peiyi; Zheng, Guangrong; Zhou, Daohong; Huo, Zhiguang; Licht, Jonathan; George, Thomas J.; Allegra, Carmen; Trevino, Jose G.; Hughes, Steven J.
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收藏Protein Degrader WH25244 Eliminates Venetoclax Resistance Factors: Mutant or Hyperphosphorylated BCL2, and BCL-XL蛋白降解剂WH25244消除Venetoclax耐药因子:突变型或过度磷酸化BCL2,以及BCL-XL
Rohena, Daisy Y. Diaz; Mitchell, Andrew D.; Wang, Jing; Chamberlain, Stephanie; Liu, Chaomei; Sanchez II, John R.; Williams, Charmelle D.; Wathan, Trisha K.; Slawin, Bailey; Bowman, Kevin; Yuan, Yaxia; Zhang, Peiyi; Hu, Wanyi; Zheng, Guangrong; Wierda, William G.; Jain, Nitin; Davids, Matthew S.; Zhou, Daohong; Woyach, Jennifer A.; Sampath, Deepa
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收藏Development and crystal structures of a potent second-generation dual degrader of BCL-2 and BCL-xL
Nayak, Digant; Lv, Dongwen; Yuan, Yaxia; Zhang, Peiyi; Hu, Wanyi; Nayak, Anindita; Ruben, Eliza A.; Lv, Zongyang; Sung, Patrick; Hromas, Robert; Zheng, Guangrong; Zhou, Daohong; Olsen, Shaun K.
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收藏AhR agonist tapinarof ameliorates lupus autoimmunity by suppressing Tfh cell differentiation via regulation of the JAK2-STAT3 signaling pathway
Zhang, Ying; Pan, Yanyan; Zhang, Peiyi; Wang, Fang; Han, Ying; Li, Kailin; Jiang, Wen; Wang, Jue; Luan, Yun; Xin, Qian
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收藏Co-targeting BCL-XL and BCL-2 by PROTAC 753B eliminates leukemia cells and enhances efficacy of chemotherapy by targeting senescent cells
Jia, Yannan; Han, Lina; Ramage, Cassandra L.; Wang, Zhe; Weng, Connie C.; Yang, Lei; Colla, Simona; Ma, Helen; Zhang, Weiguo; Andreeff, Michael; Daver, Naval; Jain, Nitin; Pemmaraju, Naveen; Bhalla, Kapil; Mustjoki, Satu; Zhang, Peiyi; Zheng, Guangrong; Zhou, Daohong; Zhang, Qi; Konopleva, Marina
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收藏Co-targeting BCL-XL and MCL-1 with DT2216 and AZD8055 synergistically inhibit small-cell lung cancer growth without causing on-target toxicities in mice
Khan, Sajid; Kellish, Patrick; Connis, Nick; Thummuri, Dinesh; Wiegand, Janet; Zhang, Peiyi; Zhang, Xuan; Budamagunta, Vivekananda; Hua, Nan; Yang, Yang; De, Umasankar; Jin, Lingtao; Zhang, Weizhou; Zheng, Guangrong; Hromas, Robert; Hann, Christine; Zajac-Kaye, Maria; Kaye, Frederic J.; Zhou, Daohong
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收藏Targeting BCL-XL in fibrolamellar hepatocellular carcinoma
Shebl, Bassem; Ng, Denise; Lalazar, Gadi; Rosemore, Carly; Finkelstein, Tova M.; Migler, Rachael D.; Zheng, Guangrong; Zhang, Peiyi; Jiang, Caroline S.; Qureshi, Adam; Vaughan, Roger; Yarchoan, Mark; de Jong, Ype P.; Rice, Charles M.; Coffino, Philip; Ortiz, Michael V.; Zhou, Daohong; Simon, Sanford M.
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收藏The presence of vessels encapsulating tumor clusters is associated with an immunosuppressive tumor microenvironment in hepatocellular carcinoma包裹肿瘤簇的血管的存在与肝细胞癌中免疫抑制肿瘤微环境有关
Zhang, Peiyi; Ono, Atsushi; Fujii, Yasutoshi; Hayes, Clair Nelson; Tamura, Yosuke; Miura, Ryoichi; Shirane, Yuki; Nakahara, Hikaru; Yamauchi, Masami; Uchikawa, Shinsuke; Uchida, Takuro; Teraoka, Yuji; Fujino, Hatsue; Nakahara, Takashi; Murakami, Eisuke; Miki, Daiki; Kawaoka, Tomokazu; Okamoto, Wataru; Makokha, Grace Naswa; Imamura, Michio; Arihiro, Koji; Kobayashi, Tsuyoshi; Ohdan, Hideki; Fujita, Masashi; Nakagawa, Hidewaki; Chayama, Kazuaki; Aikata, Hiroshi
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