未登录 Deciphering Ibogaine's Matrix Pharmacology: Multiple Transporter Modulation at Serotonin Synapses Hwu, Christopher; Havel, Vaclav; Westergaard, Xavier; Mendieta, Adriana M.; Serrano, Inis C.; Hwu, Jennifer; Walther, Donna; Lankri, David; Selinger, Tim Luca; He, Keer; Liu, Rose; Shern, Tyler P.; Sun, Steven; Ma, Boxuan; Gonzalez, Bruno; Rodriguez, Luisina; Goodman, Hannah J.; Wu, Hunter; Sonders, Mark S.; Baumann, Michael H.; Carrera, Ignacio; Sulzer, David; Sames, Dalibor 分享 收藏
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Oxa-Iboga alkaloids lack cardiac risk and disrupt opioid use in animal models Havel, Vaclav; Kruegel, Andrew C.; Bechand, Benjamin; Mcintosh, Scot; Stallings, Leia; Hodges, Alana; Wulf, Madalee G.; Nelson, Mel; Hunkele, Amanda; Ansonoff, Michael; Pintar, John E.; Hwu, Christopher; Ople, Rohini S.; Abi-Gerges, Najah; Zaidi, Saheem A.; Katritch, Vsevolod; Yang, Mu; Javitch, Jonathan A.; Majumdar, Susruta; Hemby, Scott E.; Sames, Dalibor 分享 收藏
Molecular Design of SERTlight: A Fluorescent Serotonin Probe for Neuronal Labeling in the Brain Lee, Wei-Li; Westergaard, Xavier; Hwu, Christopher; Hwu, Jennifer; Fiala, Tomas; Lacefield, Clay; Boltaev, Umed; Mendieta, Adriana M.; Lin, Lisa; Sonders, Mark S.; Brown, Keaon R.; He, Keer; Asher, Wesley B.; Javitch, Jonathan A.; Sulzer, David; Sames, Dalibor 分享 收藏
Dopamine transporter and synaptic vesicle sorting defects underlie auxilin-associated Parkinson?s disease Vidyadhara, D. J.; Somayaji, Mahalakshmi; Wade, Nigel; Yucel, Betul; Zhao, Helen; Shashaank, N.; Ribaudo, Joseph; Gupta, Jyoti; Lam, TuKiet T.; Sames, Dalibor; Greene, Lois E.; Sulzer, David L.; Chandra, Sreeganga S. 分享 收藏
Pharmacological Mechanism of the Non-hallucinogenic 5-HT2A Agonist Ariadne and Analogs Cunningham, Michael J.; Bock, Hailey A.; Serrano, Inis C.; Bechand, Benjamin; Vidyadhara, D. J.; Bonniwell, Emma M.; Lankri, David; Duggan, Priscilla; Nazarova, Antonina L.; Cao, Andrew B.; Calkins, Maggie M.; Khirsariya, Prashant; Hwu, Christopher; Katritch, Vsevolod; Chandra, Sreeganga S.; McCorvy, John D.; Sames, Dalibor 分享 收藏
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Oxidative Metabolism as a Modulator of Kratom's Biological Actions Chakraborty, Soumen; Uprety, Rajendra; Slocum, Samuel T.; Irie, Takeshi; Le Rouzic, Valerie; Li, Xiaohai; Wilson, Lisa L.; Scouller, Brittany; Alder, Amy F.; Kruegel, Andrew C.; Ansonoff, Michael; Varadi, Andras; Eans, Shainnel O.; Hunkele, Amanda; Allaoa, Abdullah; Kalra, Sanjay; Xu, Jin; Pan, Ying Xian; Pintar, John; Kivell, Bronwyn M.; Pasternak, Gavril W.; Cameron, Michael D.; McLaughlin, Jay P.; Sames, Dalibor; Majumdar, Susruta 分享 收藏
A Novel Mitragynine Analog with Low-Efficacy Mu Opioid Receptor Agonism Displays Antinociception with Attenuated Adverse Effects Chakraborty, Soumen; DiBerto, Jeffrey F.; Faouzi, Abdelfattah; Bernhard, Sarah M.; Gutridge, Anna M.; Ramsey, Steven; Zhou, Yuchen; Provasi, Davide; Nuthikattu, Nitin; Jilakara, Rahul; Nelson, Melissa N. F.; Asher, Wesley B.; Eans, Shainnel O.; Wilson, Lisa L.; Chintala, Satyanarayana M.; Filizola, Marta; van Rijn, Richard M.; Margolis, Elyssa B.; Roth, Bryan L.; McLaughlin, Jay P.; Che, Tao; Sames, Dalibor; Javitch, Jonathan A.; Majumdar, Susruta 分享 收藏
Site selective C-H functionalization of Mitragyna alkaloids reveals a molecular switch for tuning opioid receptor signaling efficacy Bhowmik, Srijita; Galeta, Juraj; Havel, Vaclav; Nelson, Melissa; Faouzi, Abdelfattah; Bechand, Benjamin; Ansonoff, Mike; Fiala, Tomas; Hunkele, Amanda; Kruegel, Andrew C.; Pintar, John E.; Majumdar, Susruta; Javitch, Jonathan A.; Sames, Dalibor 分享 收藏
Chemical Targeting of Voltage Sensitive Dyes to Specific Cells and Molecules in the Brain Fiala, Tomas; Wang, Jihang; Dunn, Matthew; Sebej, Peter; Nwadibia, Ekeoma; Martinez, Diana M.; Cheetham, Claire E. J.; Fogle, Keri J.; Palladino, Michael J.; Bando, Yuki; Yuste, Rafael; Freyberg, Zachary; Sulzer, David; Sames, Dalibor; Choi, Se Joon; Fialova, Eva 分享 收藏
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7-Hydroxymitragynine Is an Active Metabolite of Mitragynine and a Key Mediator of Its Analgesic Effects Kruegel, Andrew C.; Uprety, Rajendra; Grinnell, Steven G.; Langreck, Cory; Pekarskaya, Elizabeth A.; Le Rouzic, Valerie; Ansonoff, Michael; Gassaway, Madalee M.; Pintar, John E.; Pasternak, Gavril W.; Javitch, Jonathan A.; Majumdar, Susruta; Sames, Dalibor 分享 收藏
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Designing a norepinephrine optical tracer for imaging individual noradrenergic synapses and their activity in vivo Dunn, Matthew; Henke, Adam; Clark, Samuel; Kovalyova, Yekaterina; Kempadoo, Kimberly A.; Karpowicz, Richard J.; Kandel, Eric R., Jr.; Sulzer, David; Sames, Dalibor 分享 收藏
Toward Serotonin Fluorescent False Neurotransmitters: Development of Fluorescent Dual Serotonin and Vesicular Monoamine Transporter Substrates for Visualizing Serotonin Neurons 走向5-羟色胺荧光假神经递质: 开发用于可视化5-羟色胺神经元的荧光双重5-羟色胺和囊泡单胺转运蛋白底物 Henke, Adam; Kovalyova, Yekaterina; Dunn, Matthew; Dreier, Dominik; Gubernator, Niko G.; Dincheva, Iva; Hwu, Christopher; Sebej, Peter; Ansorge, Mark S.; Sulzer, David; Sames, Dalibor 分享 收藏
Identification of Fluorescent Small Molecule Compounds for Synaptic Labeling by Image-Based, High-Content Screening Dunn, Matthew; Boltaev, Umed; Beskow, Anne; Pampou, Sergey; Realubit, Ronald; Meira, Torcato; Silva, Joao Vaz; Reeb, Rose; Karan, Charles; Jockusch, Steffen; Sulzer, David; Chang, Young Tae; Sames, Dalibor; Waites, Clarissa L. 分享 收藏
Multiplex quantitative assays indicate a need for re-evaluating reported small-molecule TrkB agonists Boltaev, Umed; Meyer, Yves; Tolibzoda, Farangis; Jacques, Teresa; Gassaway, Madalee; Xu, Qihong; Wagner, Florence; Zhang, Yan-Ling; Palmer, Michelle; Holson, Edward; Sames, Dalibor 分享 收藏