未登录Rebastinib inhibits FoxO1 activity and reduces dexamethasone-induced atrophy and its-related gene expression in cultured myotubesRebastinib抑制FoxO1活性,并降低地塞米松诱导的萎缩及其相关基因在培养的肌管中的表达。
Sato, Tomoki; Morita, Akihito; Watanabe, Yui; Naito, Yumi; Kawaji, Haruka; Nakagawa, Takumi; Hamaguchi, Hiroki; Manabe, Yasuko; Fujii, Nobuharu L.; Ogo, Naohisa; Asai, Akira; Kamei, Yasutomi; Miura, Shinji
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收藏STAT3 inhibition suppresses adaptive survival of ALK-rearranged lung cancer cells through transcriptional modulation of apoptosis
Yanagimura, Naohiro; Takeuchi, Shinji; Fukuda, Koji; Arai, Sachiko; Tanimoto, Azusa; Nishiyama, Akihiro; Ogo, Naohisa; Takahashi, Hiroyuki; Asai, Akira; Watanabe, Satoshi; Kikuchi, Toshiaki; Yano, Seiji
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收藏Chemical augmentation of mitochondrial electron transport chains tunes T cell activation threshold in tumors
Dotsu, Yosuke; Muraoka, Daisuk; Ogo, Naohisa; Sonoda, Yudai; Yasui, Kiyoshi; Yamaguchi, Hiroyuki; Yagita, Hideo; Mukae, Hiroshi; Asai, Akira; Ikeda, Hiroaki
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收藏Design, synthesis, and evaluation of a novel prodrug, a S-trityl-L-cysteine derivative targeting kinesin spindle protein
Fukai, Ryota; Ogo, Naohisa; Ichida, Taiki; Yamane, Masayoshi; Sawada, Jun-ichi; Miyoshi, Nao; Murakami, Hisashi; Asai, Akira
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收藏Efficacy of combination treatment using YHO-1701, an orally active STAT3 inhibitor, with molecular-targeted agents on cancer cell lines
Taniguchi, Keisuke; Konishi, Hiroaki; Yoshinaga, Akiko; Tsugane, Momomi; Takahashi, Hiroyuki; Nishisaka, Fukiko; Shishido, Yoshiyuki; Asai, Akira
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收藏Discovery of Carbono(di)thioates as Indoleamine 2,3-Dioxygenase 1 Inhibitors发现碳 (二) 硫代酸酯作为吲哚胺2,3-双加氧酶1抑制剂
Kumazawa, Miyuki; Tejima, Manabu; Fukuda, Miwa; Takeda, Shota; Suzuki, Kenji; Mizumoto, Yukiko; Sato, Kakeru; Waki, Minoru; Miyachi, Hiroyuki; Asai, Akira; Takikawa, Osamu; Hashimoto, Tomoko; Ohno, Osamu; Matsuno, Kenji
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收藏Towards the Inhibition of Protein-Protein Interactions (PPIs) in STAT3: Insights into a New Class of Benzothiadiazole Derivatives
Mori, Matteo; Gilardoni, Ettore; Regazzoni, Luca; Pedretti, Alessandro; Colombo, Diego; Parkinson, Gary; Asai, Akira; Meneghetti, Fiorella; Villa, Stefania; Gelain, Arianna
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收藏Discovery of a Potent Anticancer Agent PVHD303 with in Vivo Activity发现具有体内活性的有效抗癌剂PVHD303
Suzuki, Yumiko; Otake, Ayana; Ueno, Satoshi; Hayashi, Kensuke; Ishii, Hirosuke; Miyoshi, Nao; Kuroiwa, Kenta; Tachikawa, Masashi; Fujimaki, Yuki; Nishiyama, Kotaro; Manabe, Kei; Yamazaki, Ryuta; Asai, Akira
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收藏Impact of combination therapy with anti-PD-1 blockade and a STAT3 inhibitor on the tumor-infiltrating lymphocyte status
Ashizawa, Tadashi; Iizuka, Akira; Maeda, Chie; Tanaka, Emiko; Kondou, Ryota; Miyata, Haruo; Sugino, Takashi; Kawata, Takuya; Deguchi, Shoichi; Mitsuya, Koichi; Hayashi, Nakamasa; Asai, Akira; Ito, Mamoru; Yamaguchi, Ken; Akiyama, Yasuto
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收藏Involvement of phosphatidylinositol metabolism in aluminum-induced malate secretion in Arabidopsis
Wu, Liujie; Sadhukhan, Ayan; Kobayashi, Yuriko; Ogo, Naohisa; Tokizawa, Mutsutomo; Agrahari, Raj Kishan; Ito, Hiroki; Iuchi, Satoshi; Kobayashi, Masatomo; Asai, Akira; Koyama, Hiroyuki
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收藏Antigen delivery targeted to tumor-associated macrophages overcomes tumor immune resistance靶向肿瘤相关巨噬细胞的抗原递送克服了肿瘤免疫抗性
Muraoka, Daisuke; Seo, Naohiro; Hayashi, Tae; Tahara, Yoshiro; Fujii, Keisuke; Tawara, Isao; Miyahara, Yoshihiro; Okamori, Kana; Yagita, Hideo; Imoto, Seiya; Yamaguchi, Rui; Komura, Mitsuhiro; Miyano, Satoru; Goto, Masahiro; Sawada, Shin-ichi; Asai, Akira; Ikeda, Hiroaki; Akiyoshi, Kazunari; Harada, Naozumi; Shiku, Hiroshi
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