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Richard R. Tidwell

university system of georgia

53H指数
271论文数
7.3K被引数
收录论文 71
发表时间
Positively selected modifications in the pore of TbAQP2 allow pentamidine to enter Trypanosoma brucei
err2020-08-11
err20
errOAAI
errAlghamdi, Ali H.; Munday, Jane C.; Campagnaro, Gustavo Daniel; Gurvic, Dominik; Svensson, Fredrik; Okpara, Chinyere E.; Kumar, Arvind; Quintana, Juan; Abril, Maria Esther Martin; Milic, Patrik; Watson, Laura; Paape, Daniel; Settimo, Luca; Dimitriou, Anna; Wielinska, Joanna; Smart, Graeme; Anderson, Laura F.; Woodley, Christopher M.; Kelly, Siu Pui Ying; Ibrahim, Hasan M. S.; Hulpia, Fabian; Al-Salabi, Mohammed, I; Eze, Anthonius A.; Sprenger, Teresa; Teka, Ibrahim A.; Gudin, Simon; Weyand, Simone; Field, Mark; Dardonville, Christophe; Tidwell, Richard R.; Carrington, Mark; O'Neill, Paul; Boykin, David W.; Zachariae, Ulrich; De Koning, Harry P.
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In Vitro, In Silico, and In Vivo Analyses of Novel Aromatic Amidines against Trypanosoma cruzi
err2018-02-01
err19
errOAAI
errSantos, Camila C.; Lionel, Jessica R.; Peres, Raiza B.; Batista, Marcos M.; da Silva, Patricia B.; de Oliveira, Gabriel M.; da Silva, Cristiane F.; Batista, Denise G. J.; Souza, Sandra Maria O.; Andrade, Carolina H.; Neves, Bruno J.; Braga, Rodolpho C.; Patrick, Donald A.; Bakunova, Svetlana M.; Tidwell, Richard R.; Soeiro, Maria de Nazare C.
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Role of suppression of the inward rectifier current in terminal action potential repolarization in the failing heart
err2017-08-01
err11
errOAAI
errKlein, Michael G.; Shou, Matie; Stohlman, Jayna; Solhjoo, Soroosh; Haigney, Myles; Tidwell, Richard R.; Goldstein, Robert E.; Flagg, Thomas P.; Haigney, Mark C.
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In Vitro, Ex Vivo, and In Vivo Activities of Diamidines against Trypanosoma congolense and Trypanosoma vivax
err2017-05-01
err10
errOAAI
errGillingwater, Kirsten; Kunz, Christina; Braghiroli, Christiane; Boykin, David W.; Tidwell, Richard R.; Brun, Reto
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Urea Derivatives of 2-Aryl-benzothiazol-5-amines: A New Class of Potential Drugs for Human African Trypanosomiasis
err2016-12-19
err54
errOAAI
errPatrick, Donald A.; Gillespie, J. Robert; McQueen, Joshua; Hulverson, Matthew A.; Ranade, Ranae M.; Creason, Sharon A.; Herbst, Zackary M.; Gelb, Michael H.; Buckner, Frederick S.; Tidwell, Richard R.
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Synthesis of novel amide and urea derivatives of thiazol-2-ethylamines and their activity against Trypanosoma brucei rhodesiense
err2016-06-01
err30
errOAAI
errPatrick, Donald A.; Wenzler, Tanja; Yang, Sihyung; Weiser, Patrick T.; Wang, Michael Zhuo; Brun, Reto; Tidwell, Richard R.
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In Vitro and In Vivo Trypanosomicidal Action of Novel Arylimidamides against Trypanosoma cruzi
err2016-04-01
err24
errOAAI
errGuedes-da-Silva, F. H.; Batista, D. G. J.; Meuser, M. B.; Demarque, K. C.; Fulco, T. O.; Araujo, J. S.; Da Silva, P. B.; Da Silva, C. F.; Patrick, D. A.; Bakunova, S. M.; Bakunov, S. A.; Tidwell, R. R.; Oliveira, G. M.; Britto, C.; Moreira, O. C.; Soeiro, M. N. C.
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Efficacy, Safety, and Dose of Pafuramidine, a New Oral Drug for Treatment of First Stage Sleeping Sickness, in a Phase 2a Clinical Study and Phase 2b Randomized Clinical Studies
err2016-02-16
err19
errOAAI
errBurri, Christian; Yeramian, Patrick D.; Allen, James L.; Merolle, Ada; Serge, Kazadi Kyanza; Mpanya, Alain; Lutumba, Pascal; Ku Mesu, Victor Kande Betu; Mia Bilenge, Constantin Miaka; Fina Lubaki, Jean-Pierre; Mpoo Mpoto, Alfred; Thompson, Mark; Fungula Munungu, Blaise; Manuel, Francisco; Josenando, Theophilo; Bernhard, Sonja C.; Olson, Carol A.; Blum, Johannes; Tidwell, Richard R.; Pohlig, Gabriele
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Efficacy and Safety of Pafuramidine versus Pentamidine Maleate for Treatment of First Stage Sleeping Sickness in a Randomized, Comparator-Controlled, International Phase 3 Clinical Trial
err2016-02-16
err38
errOAAI
errPohlig, Gabriele; Bernhard, Sonja C.; Blum, Johannes; Burri, Christian; Mpanya, Alain; Lubaki, Jean-Pierre Fina; Mpoto, Alfred Mpoo; Munungu, Blaise Fungula; N'tombe, Patrick Mangoni; Deo, Gratias Kambau Manesa; Mutantu, Pierre Nsele; Kuikumbi, Florent Mbo; Mintwo, Alain Fukinsia; Munungi, Augustin Kayeye; Dala, Amadeu; Macharia, Stephen; Bilenge, Constantin Miaka Mia; Mesu, Victor Kande Betu Ku; Franco, Jose Ramon; Dituvanga, Ndinga Dieyi; Tidwell, Richard R.; Olson, Carol A.
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Chemotherapy of Second Stage Human African Trypanosomiasis: Comparison between the Parenteral Diamidine DB829 and Its Oral Prodrug DB868 in Vervet Monkeys
err2015-02-05
err22
errOAAI
errThuita, John K.; Wolf, Kristina K.; Murilla, Grace A.; Bridges, Arlene S.; Boykin, David W.; Mutuku, James N.; Liu, Qiang; Jones, Susan K.; Gem, Charles O.; Ching, Shelley; Tidwell, Richard R.; Wang, Michael Z.; Paine, Mary F.; Brun, Reto
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In Vitro and In Vivo Evaluation of 28DAP010, a Novel Diamidine for Treatment of Second-Stage African Sleeping Sickness
err2014-08-01
err18
errOAAI
errWenzler, Tanja; Yang, Sihyung; Patrick, Donald A.; Braissant, Olivier; Ismail, Mohamed A.; Tidwell, Richard R.; Boykin, David W.; Wang, Michael Zhuo; Brun, Reto
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In Vitro and In Vivo Biological Effects of Novel Arylimidamide Derivatives against Trypanosoma cruzi
err2014-07-01
err33
errOAAI
errTimm, Bruno Lisboa; da Silva, Patricia Bernadino; Batista, Marcos Meuser; Guedes da Silva, Francisca Hildemagna; da Silva, Cristiane Frana; Tidwell, Richard R.; Patrick, Donald A.; Jones, Susan Kilgore; Bakunov, Stanislav A.; Bakunova, Svetlana M.; Soeiro, Maria de Nazare C.
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CYP1A1 and CYP1B1-Mediated Biotransformation of the Antitrypanosomal Methamidoxime Prodrug DB844 Forms Novel Metabolites Through Intramolecular Rearrangement
err2014-01-01
err9
errOAAI
errJu, Wujian; Yang, Sihyung; Ansede, John H.; Stephens, Chad E.; Bridges, Arlene S.; Voyksner, Robert D.; Ismail, Mohamed A.; Boykin, David W.; Tidwell, Richard R.; Hall, James Edwin; Wang, Michael Zhuo
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Antiprotozoal activity of dicationic 3,5-diphenylisoxazoles, their prodrugs and aza-analogues
err2014-01-01
err16
PREAI
errPatrick, Donald A.; Bakunov, Stanislav A.; Bakunova, Svetlana M.; Wenzler, Tanja; Brun, Reto; Tidwell, Richard R.
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Synthesis and antiprotozoal activities of benzyl phenyl ether diamidine derivatives
err2013-09-01
err24
PREAI
errPatrick, Donald A.; Bakunov, Stanislav A.; Bakunova, Svetlana M.; Jones, Susan Kilgore; Wenzler, Tanja; Barszcz, Todd; Kumar, Arvind; Boykin, David W.; Werbovetz, Karl A.; Brun, Reto; Tidwell, Richard R.
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Synthesis and Antiprotozoal Activity of Dicationic m-Terphenyl and 1,3-Dipyridylbenzene Derivatives
err2013-06-24
err42
PREAI
errPatrick, Donald A.; Ismail, Mohamed A.; Arafa, Reem K.; Wenzler, Tanja; Zhu, Xiaohua; Pandharkar, Trupti; Jones, Susan Kilgore; Werbovetz, Karl A.; Brun, Reto; Boykin, David W.; Tidwell, Richard R.
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Structure-activity relationships of pentamidine-affected ion channel trafficking and dofetilide mediated rescue
err2013-06-21
err20
errOAAI
errVarkevisser, R.; Houtman, M. J. C.; Linder, T.; de Git, K. C. G.; Beekman, H. D. M.; Tidwell, R. R.; IJzerman, A. P.; Stary-Weinzinger, A.; Vos, M. A.; van der Heyden, M. A. G.
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Safety, Pharmacokinetic, and Efficacy Studies of Oral DB868 in a First Stage Vervet Monkey Model of Human African Trypanosomiasis
err2013-06-06
err16
errOAAI
errThuita, John K.; Wolf, Kristina K.; Murilla, Grace A.; Liu, Qiang; Mutuku, James N.; Chen, Yao; Bridges, Arlene S.; Mdachi, Raymond E.; Ismail, Mohamed A.; Ching, Shelley; Boykin, David W.; Hall, James Edwin; Tidwell, Richard R.; Paine, Mary F.; Brun, Reto; Wang, Michael Zhuo
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Efficient and specific cardiac IK1 inhibition by a new pentamidine analogue
err2013-04-25
err35
PREAI
errTakanari, Hiroki; Nalos, Lukas; Stary-Weinzinger, Anna; de Git, Kathy C. G.; Varkevisser, Rosanne; Linder, Tobias; Houtman, Marien J. C.; Peschar, Maaike; de Boer, Teun P.; Tidwell, Richard R.; Rook, Martin B.; Vos, Marc A.; van der Heyden, Marcel A. G.
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A Mouse Diversity Panel Approach Reveals the Potential for Clinical Kidney Injury Due to DB289 Not Predicted by Classical Rodent Models
err2012-08-31
err52
errOAAI
errHarrill, Alison H.; DeSmet, Kristina D.; Wolf, Kristina K.; Bridges, Arlene S.; Eaddy, J. Scott; Kurtz, C. Lisa; Hall, J. Ed.; Paine, Mary F.; Tidwell, Richard R.; Watkins, Paul B.
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