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Laura H. Heitman

Leiden University

44H指数
299论文数
6.8K被引数
收录论文 66
发表时间
Leveraging Targeted Protein Degradation for G Protein-Coupled Receptors: The Development of CCR2 Molecular Degraders
err2025-12-01
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PREAI
errEssa, Khaled; Ortiz Zacarias, Natalia V.; Roth, Sascha; Xin, Bo-Tao; de Winter, Sabine; van der Horst, Cas; Bleijs, Bente; de Heiden, Richard A.; Voulgaraki, Rodanthi; Neubert, Elsa; Ovaa, Huib; Danen, Erik H. J.; Mulder, Monique P. C.; Moreau, Kevin; van der Es, Daan; Heitman, Laura H.
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Combining AlphaFold with Focused Virtual Library Design in the Development of Novel CCR2 and CCR5 Antagonists结合AlphaFold与定向虚拟库设计在新型CCR2和CCR5拮抗剂开发中的应用
err2025-11-01
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PREAI
errEssa, Khaled; van der Dussen, Kian Noorman; Yao, Yao; Bleijs, Bente; Zacarias, Natalia V. Ortiz; Heitman, Laura H.; van Westen, Gerard J. P.; Jespers, Willem; van der Es, Daan; Sicho, Martin
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Molecular basis of ligand binding and receptor activation at the human A3 adenosine receptor人源A3腺苷受体配体结合与受体激活的分子基础
err2025-08-18
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errOAAI
errLiudi Zhang; Jesse I. Mobbs; Felix M. Bennetts; Hariprasad Venugopal; Anh T. N. Nguyen; Arthur Christopoulos; Daan van der Es; Laura H. Heitman; Lauren T. May; Alisa Glukhova; David M. Thal
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Toward Assay-Aware Bioactivity Model(er)s: Getting a Grip on Biological Context面向 Assay-Aware 生物活性模型:把握生物学背景
err2025-06-30
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errLinde Schoenmaker; Enzo G. Sastrokarijo; Laura H. Heitman; Joost B. Beltman; Willem Jespers; Gerard J.P. van Westen
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The solute carrier superfamily interactome溶质载体超家族互作网络
err2025-05-12
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errOAAI
errFrommelt, Fabian; Ladurner, Rene; Goldmann, Ulrich; Wolf, Gernot; Ingles-Prieto, Alvaro; Lineiro-Retes, Eva; Gelova, Zuzana; Hopp, Ann-Katrin; Christodoulaki, Eirini; Teoh, Shao Thing; Leippe, Philipp; Santini, Brianda L.; Rebsamen, Manuele; Lindinger, Sabrina; Serrano, Iciar; Onstein, Svenja; Klimek, Christoph; Barbosa, Barbara; Pantielieieva, Anastasiia; Dvorak, Vojtech; Hannich, Thomas J.; Schoenbett, Julian; Sansig, Gilles; Mocking, Tamara A. M.; Ooms, Jasper F.; Ijzerman, Adriaan P.; Heitman, Laura H.; Sykacek, Peter; Reinhardt, Juergen; Mueller, Andre C.; Wiedmer, Tabea
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Covalent functionalization of G protein-coupled receptors by small molecular probes
err2025-01-01
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errOAAI
errBeerkens, Bert L. H.; Ijzerman, Adriaan P.; Heitman, Laura H.; van der Es, Daan
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The effect of cancer-associated mutations on ligand binding and receptor function - A case for the 5-HT2C receptor
err2024-12-01
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errFeng, Chenlin; Liu, Rongfang; Brooks, Reno; Wang, Xuesong; Jespers, Willem; Gonzalez, Marina Gorostiola; van Westen, Gerard J. P.; Danen, Erik H. J.; Heitman, Laura H.
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Labeling of CC Chemokine Receptor 2 with a Versatile Intracellular Allosteric Probe
err2024-08-26
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errden Hollander, Lisa S.; Beerkens, Bert L. H.; Dekkers, Sebastian; van Veldhoven, Jacobus P. D.; Zacarias, Natalia V. Ortiz; van der Horst, Cas; Sieders, Elisabeth G.; de Valk, Bert; Wang, Jianhui; Ijzerman, Adriaan P.; van der Es, Daan; Heitman, Laura H.
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Highly Selective Drug-Derived Fluorescent Probes for the Cannabinoid Receptor Type 1 (CB1R)大麻素受体1型 (CB1R) 的高选择性药物衍生荧光探针
err2024-07-11
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errMach, Leonard; Omran, Anahid; Bouma, Jara; Radetzki, Silke; Sykes, David A.; Guba, Wolfgang; Li, Xiaoting; Hoeffelmeyer, Calvin; Hentsch, Axel; Gazzi, Thais; Mostinski, Yelena; Wasinska-Kalwa, Malgorzata; de Molnier, Fabio; van der Horst, Cas; von Kries, Jens Peter; Vendrell, Marc; Hua, Tian; Veprintsev, Dmitry B.; Heitman, Laura H.; Grether, Uwe; Nazare, Marc
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N-Acyl-N-Alkyl Sulfonamide Probes for Ligand-Directed Covalent Labeling of GPCRs: The Adenosine A2B Receptor as Case Study
err2024-06-26
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errBeerkens, Bert L. H.; Andrianopoulou, Vasiliki; Wang, Xuesong; Liu, Rongfang; van Westen, Gerard J. P.; Jespers, Willem; Ijzerman, Adriaan P.; Heitman, Laura H.; van der Es, Daan
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Exploring novel dilazep derivatives as hENT1 inhibitors and potentially covalent molecular tools
err2024-06-15
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errDilweg, Majlen A.; Gorostiola Gonzalez, Marina; de Ruiter, Martijn D.; Meijboom, Nadine J.; van Veldhoven, Jacobus P. D.; Liu, Rongfang; Jespers, Willem; van Westen, Gerard J. P.; Heitman, Laura H.; Ijzerman, Adriaan P.; van der Es, Daan
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Still in Search for an EAAT Activator: GT949 Does Not Activate EAAT2, nor EAAT3 in Impedance and Radioligand Uptake Assays
err2024-03-13
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errvan Veggel, Lieve; Mocking, Tamara A. M.; Sijben, Hubert J.; Liu, Rongfang; Gonzalez, Marina Gorostiola; Dilweg, Majlen A.; Royakkers, Jeroen; Li, Anna; Kumar, Vijay; Dong, Yin Yao; Bullock, Alex; Sauer, David B.; Dilien, Hanne; van Westen, Gerard J. P.; Schreiber, Rudy; Heitman, Laura H.; Vanmierlo, Tim
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Stereochemical optimization of N,2-substituted cycloalkylamines as norepinephrine reuptake inhibitors
err2024-01-01
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PREAI
errDilweg, Majlen A.; Mocking, Tamara A. M.; Maragkoudakis, Pantelis; van Westen, Gerard J. P.; Heitman, Laura H.; Ijzerman, Adriaan P.; Jespers, Willem; van der Es, Daan
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Visualization of membrane localization and the functional state of CB2R pools using matched agonist and inverse agonist probe pairs
err2024-01-01
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errWasinska-Kalwa, M.; Omran, A.; Mach, L.; Scipioni, L.; Bouma, J.; Li, X.; Radetzki, S.; Mostinski, Y.; Schippers, M.; Gazzi, T.; van der Horst, C.; Brennecke, B.; Hanske, A.; Kolomeets, Y.; Guba, W.; Sykes, D.; von Kries, J. P.; Broichhagen, J.; Hua, T.; Veprintsev, D.; Heitman, L. H.; Oddi, S.; MacCarrone, M.; Grether, U.; Nazare, M.
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Amonoacylglycerol lipase inhibitor showing therapeutic efficacy in mice without central side effects or dependence
err2023-12-05
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errJiang, Ming; Huizenga, Mirjam C. W.; Wirt, Jonah L.; Paloczi, Janos; Amedi, Avand; van den Berg, Richard J. B. H. N.; Benz, Joerg; Collin, Ludovic; Deng, Hui; Di, Xinyu; Driever, Wouter F.; Florea, Bogdan I.; Grether, Uwe; Janssen, Antonius P. A.; Hankemeier, Thomas; Heitman, Laura H.; Lam, Tsang-Wai; Mohr, Florian; Pavlovic, Anto; Ruf, Iris; van den Hurk, Helma; Stevens, Anna F.; van der Vliet, Daan; van der Wel, Tom; Wittwer, Matthias B.; van Boeckel, Constant A. A.; Pacher, Pal; Hohmann, Andrea G.; van der Stelt, Mario
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