arrow
返回
J

Joseph P. Vacca

merck & company

57H指数
277论文数
1.0W被引数
收录论文 70
发表时间
Convection enhanced delivery of a novel ATR inhibitor synergizes with systemic lomustine for improved treatment of glioblastoma
err2024-03-22
err0
PREAI
errJosowitz, Alexander; Lee, Teresa; Sundaram, Ranjini K.; Pothupitiya, Jinal; Brown, Eric J.; Sule, Amrita; Beckta, Jason; Wang, Yongheng; Vacca, Joseph; Gilad, Oren; Bindra, Ranjit S.; Saltzman, W. Mark
err分享
err收藏
TNG917 is a clinical-grade, potent and selective inhibitor of EHMT1/2 for the treatment of immune cold tumors
err2024-03-22
err0
PREAI
errLu, Alvin; Haines, Brian; Lei, Ji; Zhang, Wenhai; Zhang, Minjie; Whittington, Douglas A.; Ferdinez, Maria Lucia; Yu, Yi; Meier, Samuel R.; Choi, Ashley; Bejnood, Alborz; Bandi, Madhavi; Lazarides, Katherine; Pan, Xuewen; Gu, Lina; Tsai, Alice W.; Sudsakorn, Sirimas; Liang, Colin; Come, Jon; Williams, Brett; Throner, Scott; Vacca, Joseph; Maxwell, John P.; Anderson, Jannik N.; Huang, Alan; Min, Chengyin; Chen, Yingnan P.
err分享
err收藏
The novel WEE1i, APR-1051, is a potentially well tolerated and effective treatment for cyclin E-overexpressing cancers
err2024-03-22
err0
PREAI
errHansbarger, Molly M.; Rocca, Stephen J.; Ritzmann, Sonia; Vacca, Joseph; Tokiwa, Bridget; Weinstein, Jonathan; Zabierek, Henry; Frye, Justin; Carleton, Michael; Brown, Eric J.; Gilad, Oren
err分享
err收藏
The DNA replication checkpoint inhibitors, ATRN-1051 (WEE1i) and ATRN-119 (ATRi), are potentially well tolerated and effective cancer treatments
err2023-12-01
err0
PREAI
errVacca, Joseph; Rocca, Stephen; Hansbarger, Molly; Ritzmann, Sonia; Frye, Justin; Simpkins, Fiona; Brown, Eric J.; Gilad, Oren
err分享
err收藏
Discovery of KB-0742, a Potent, Selective, Orally Bioavailable Small Molecule Inhibitor of CDK9 for MYC-Dependent Cancers
err2023-11-15
err12
errOAAI
errFreeman, David B.; Hopkins, Tamara D.; Mikochik, Peter J.; Vacca, Joseph P.; Gao, Hua; Naylor-Olsen, Adel; Rudra, Sonali; Li, Huixu; Pop, Marius S.; Villagomez, Rosa A.; Lee, Christina; Li, Heng; Zhou, Minyun; Saffran, Douglas C.; Rioux, Nathalie; Hood, Tressa R.; Day, Melinda A. L.; Mckeown, Michael R.; Lin, Charles Y.; Bischofberger, Norbert; Trotter, B. Wesley
err分享
err收藏
ATRN-119 and ATRN-W1051: Novel and potentially well tolerated ATR and WEE1 inhibitors for targeted cancer treatment
err2023-04-04
err1
PREAI
errVacca, Joseph; Rocca, Stephen; Frye, Justin; Schnell, Steven J.; Hansbarger, Molly; Korbel, Gregory; Simpkins, Fiona; Brown, Eric J.; Gilad, Oren
err分享
err收藏
Characterization of Pyrrolidinyl-hexahydro-pyranopiperazines as a Novel Kappa Opioid Receptor Agonist Scaffold
err2022-06-23
err2
errOAAI
errReed, Brian; Miller, Michael; Michino, Mayako; Butelman, Eduardo R.; Ben-Ezra, Ariel; Pikus, Philip; Morochnik, Michelle; Kim, Yuli; Ripka, Amy; Vacca, Joseph; Kreek, Mary Jeanne
err分享
err收藏
Preclinical pharmacokinetics and pharmacodynamics of KB-0742, a selective, oral CDK9 inhibitor
err2021-12-01
err3
PREAI
errDay, Melinda A. L.; Saffran, Douglas C.; Rioux, Nathalie; Chen, Tom; Lee, Christina; Freeman, David B.; MacKenzie, Crystal; Vacca, Joseph P.; Rahl, Peter B.; Trotter, Benjamin Wesley; Lin, Charles Y.; Kumar, Pavan; DiMartino, Jorge
err分享
err收藏
Modulating Androgen Receptor-Driven Transcription in Prostate Cancer with Selective CDK9 Inhibitors
err2021-02-01
err57
errOAAI
errRichters, Andre; Doyle, Shelby K.; Freeman, David B.; Lee, Christina; Leifer, Becky S.; Jagannathan, Sajjeev; Kabinger, Florian; Koren, Jost Vrabic; Struntz, Nicholas B.; Urgiles, Julie; Stagg, Ryan A.; Curtin, Brice H.; Chatterjee, Deep; Mathea, Sebastian; Mikochik, Peter J.; Hopkins, Tamara D.; Gao, Hua; Branch, Jonathan R.; Xin, Hong; Westover, Lori; Bignan, Gilles C.; Rupnow, Brent A.; Karlin, Kristen L.; Olson, Calla M.; Westbrook, Thomas F.; Vacca, Joseph; Wilfong, Chris M.; Trotter, B. Wesley; Saffran, Douglas C.; Bischofberger, Norbert; Knapp, Stefan; Russo, Joshua W.; Hickson, Ian; Bischoff, James R.; Gottardis, Marco M.; Balk, Steven P.; Lin, Charles Y.; Pop, Marius S.; Koehler, Angela N.
err分享
err收藏
PD-L1 IS INDUCED BY THE PERIODONTAL PATHOGEN PORPHYROMONAS GINGIVALIS AND CAN BE BLOCKED BY SMALL MOLECULE GINGIPAIN INHIBITORS, INCLUDING ATUZAGINSTAT
err2020-11-09
err0
errOAAI
errArastu-Kapur, Shirin; Mai Nguyen; Broce, Sean; Vacca, Joseph; Ehmsen, Kirk; Ermini, Florian; Haditsch, Ursula; Martinez-Horta, Aurora; Raha, Debasish; Rodriguez, Leonardo; Lynch, Casey; Dominy, Stephen; Holsinger, Leslie
err分享
err收藏
Targeting oncogenic transcription in prostate cancer with a novel, oral bioavailable, and ultra-selective CDK9 inhibitor
err2020-08-15
err0
PREAI
errRichters, Andre; Freeman, David; Lee, Christina; Kabinger, Florian; Doyle, Shelby; Leifer, Becky; Mikochik, Peter; Jagannathan, Sajjeev; Koren, Jost Vrabic; Karlin, Kristen; Olson, Calla M.; Wilfong, Christopher; Lin, Charles Y.; Saffran, Doug; Vacca, Joseph; Bischofberger, Norbert; Pop, Marius; Koehler, Angela N.
err分享
err收藏
Identification of Highly Specific Diversity-Oriented Synthesis-Derived Inhibitors of Clostridium difficile
err2017-03-07
err13
errOAAI
errDuvall, Jeremy R.; Bedard, Leanne; Naylor-Olsen, Adel M.; Manson, Abigail L.; Bittker, Joshua A.; Sun, Wenye; Fitzgerald, Mark E.; He, Zhenmin; Lee, Maurice D.; Marie, Jean-Charles; Muncipinto, Giovanni; Rush, Diane; Xu, Deming; Xu, Huisheng; Zhang, Mingliang; Earl, Ashlee M.; Palmer, Michelle A.; Foley, Michael A.; Vacca, Joseph P.; Scherer, Christina A.
err分享
err收藏
Discovery of MK-8718, an HIV Protease Inhibitor Containing a Novel Morpholine Aspartate Binding Group
err2016-05-11
err22
errOAAI
errBungard, Christopher J.; Williams, Peter D.; Ballard, Jeanine E.; Bennett, David J.; Beaulieu, Christian; Bahnck-Teets, Carolyn; Carroll, Steve S.; Chang, Ronald K.; Dubost, David C.; Fay, John F.; Diamond, Tracy L.; Greshock, Thomas J.; Hao, Li; Holloway, M. Katharine; Felock, Peter J.; Gesell, Jennifer J.; Su, Hua-Poo; Manikowski, Jesse J.; McKay, Daniel J.; Miller, Mike; Min, Xu; Molinaro, Carmela; Moradei, Oscar M.; Nantermet, Philippe G.; Nadeau, Christian; Sanchez, Rosa I.; Satyanarayana, Tummanapalli; Shipe, William D.; Singh, Sanjay K.; Vouy Linh Truong; Vijayasaradhi, Sivalenka; Wiscount, Catherine M.; Vacca, Joseph P.; Crane, Sheldon N.; McCauley, John A.
err分享
err收藏
MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants (vol 56, pg 4161, 2012)
err2014-08-01
err2
errOAAI
errSumma, Vincenzo; Ludmerer, Steven W.; McCauley, John A.; Fandozzi, Christine; Burlein, Christine; Claudio, Giuliano; Coleman, Paul J.; DiMuzio, Jillian M.; Ferrara, Marco; Di Filippo, Marcello; Gates, Adam T.; Graham, Donald J.; Harper, Steven; Hazuda, Daria J.; Huang, Qian; McHale, Carolyn; Monteagudo, Edith; Pucci, Vincenzo; Rowley, Michael; Rudd, Michael T.; Soriano, Aileen; Stahlhut, Mark W.; Vacca, Joseph P.; Olsen, David B.; Liverton, Nigel J.; Carroll, Steven S.
err分享
err收藏
Novel Quinoline-Based P2-P4 Macrocyclic Derivatives As Pan-Genotypic HCV NS3/4a Protease Inhibitors
err2014-01-09
err26
errOAAI
errShah, Unmesh; Jayne, Charles; Chackalamannil, Samuel; Velazquez, Francisco; Guo, Zhuyan; Buevich, Alexei; Howe, John A.; Chase, Robert; Soriano, Aileen; Agrawal, Sony; Rudd, Michael T.; McCauley, John A.; Liverton, Nigel J.; Romano, Joseph; Bush, Kimberly; Coleman, Paul J.; Grise-Bard, Christiane; Brochu, Marie-Christine; Charron, Sylvie; Aulakh, Virender; Bachand, Benoit; Beaulieu, Patrick; Zaghdane, Helmi; Bhat, Sathesh; Han, Yongxin; Vacca, Joseph P.; Davies, Ian W.; Weber, Ann E.; Venkatraman, Srikanth
err分享
err收藏
Discovery of MK-8742: An HCV NS5A Inhibitor with Broad Genotype Activity
err2013-10-14
err188
errOAAI
errCoburn, Craig A.; Meinke, Peter T.; Chang, Wei; Fandozzi, Christine M.; Graham, Donald J.; Hu, Bin; Huang, Qian; Kargman, Stacia; Kozlowski, Joseph; Liu, Rong; McCauley, John A.; Nomeir, Amin A.; Soll, Richard M.; Vacca, Joseph P.; Wang, Dahai; Wu, Hao; Zhong, Bin; Olsen, David B.; Ludmerer, Steven W.
err分享
err收藏
MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants
err2012-08-01
err210
errOAAI
errSumma, Vincenzo; Ludmerer, Steven W.; McCauley, John A.; Fandozzi, Christine; Burlein, Christine; Claudio, Giuliano; Coleman, Paul J.; DiMuzio, Jillian M.; Ferrara, Marco; Di Filippo, Marcello; Gates, Adam T.; Graham, Donald J.; Harper, Steven; Hazuda, Darla J.; McHale, Carolyn; Monteagudo, Edith; Pucci, Vincenzo; Rowley, Michael; Rudd, Michael T.; Soriano, Aileen; Stahlhut, Mark W.; Vacca, Joseph P.; Olsen, David B.; Liverton, Nigel J.; Carroll, Steven S.
err分享
err收藏
Discovery of MK-5172, a Macrocyclic Hepatitis C Virus NS3/4a Protease Inhibitor
err2012-03-02
err160
errOAAI
errHarper, Steven; McCauley, John A.; Rudd, Michael T.; Ferrara, Marco; DiFilippo, Marcello; Crescenzi, Benedetta; Koch, Uwe; Petrocchi, Alessia; Holloway, M. Katharine; Butcher, John W.; Romano, Joseph J.; Bush, Kimberly J.; Gilbert, Kevin F.; McIntyre, Charles J.; Nguyen, Kevin T.; Nizi, Emanuela; Carroll, Steven S.; Ludmerer, Steven W.; Burlein, Christine; DiMuzio, Jillian M.; Graham, Donald J.; McHale, Carolyn M.; Stahlhut, Mark W.; Olsen, David B.; Monteagudo, Edith; Cianetti, Simona; Giuliano, Claudio; Pucci, Vincenzo; Trainor, Nicole; Fandozzi, Christine M.; Rowley, Michael; Coleman, Paul J.; Vacca, Joseph P.; Summa, Vincenzo; Liverton, Nigel J.
err分享
err收藏
Design and Synthesis of Conformationally Constrained Inhibitors of Non-Nucleoside Reverse Transcriptase
err2011-10-28
err37
PREAI
errGomez, Robert; Jolly, Samson J.; Williams, Theresa; Vacca, Joseph P.; Torrent, Maricel; McGaughey, Georgia; Lai, Ming-Tain; Felock, Peter; Munshi, Vandna; DiStefano, Daniel; Flynn, Jessica; Miller, Mike; Yan, Youwei; Reid, John; Sanchez, Rosa; Liang, Yuexia; Paton, Brenda; Wan, Bang-Lin; Anthony, Neville
err分享
err收藏