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收藏Deciphering RNA G-quadruplex function during the early steps of HIV-1 infection
Amrane, Samir; Jaubert, Chloe; Bedrat, Amina; Rundstadler, Tiffany; Recordon-Pinson, Patricia; Aknin, Cindy; Guedin, Aurore; De Rache, Aurore; Bartolucci, Laura; Diene, Ibra; Lemoine, Frederic; Gascuel, Olivier; Pratviel, Genevieve; Mergny, Jean-Louis; Andreola, Marie-Line
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收藏SARS-CoV-2 Nsp3 unique domain SUD interacts with guanine quadruplexes and G4-ligands inhibit this interaction
Lavigne, Marc; Helynck, Olivier; Rigolet, Pascal; Boudria-Souilah, Rofia; Nowakowski, Mireille; Baron, Bruno; Brule, Sebastien; Hoos, Sylviane; Raynal, Bertrand; Guittat, Lionel; Beauvineau, Claire; Petres, Stephane; Granzhan, Anton; Guillon, Jean; Pratviel, Genevieve; Teulade-Fichou, Marie-Paule; England, Patrick; Mergny, Jean-Louis; Munier-Lehmann, Helene
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收藏New 8-Nitroquinolinone Derivative Displaying Submicromolar in Vitro Activities against Both Trypanosoma brucei and cruzi
Pedron, Julien; Boudot, Clotilde; Brossas, Jean-Yves; Pinault, Emilie; Bourgeade-Delmas, Sandra; Sournia-Saquet, Alix; Boutet-Robinet, Elisa; Destere, Alexandre; Tronnet, Antoine; Berge, Justine; Bonduelle, Colin; Deraeve, Celine; Pratviel, Genevieve; Stigliani, Jean-Luc; Paris, Luc; Mazier, Dominique; Corvaisier, Sophie; Since, Marc; Malzert-Freon, Aureprimelie; Wyllie, Susan; Milne, Rachel; Fairlamb, Alan H.; Valentin, Alexis; Courtioux, Bertrand; Verhaeghe, Pierre
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收藏G-Quadruplex binding optimization by gold(iii) insertion into the center of a porphyrin
Pipier, Angelique; De Rache, Aurore; Modeste, Coralie; Amrane, Samir; Mothes-Martin, Emmanuelle; Stigliani, Jean-Luc; Calsou, Patrick; Mergny, Jean-Louis; Pratviel, Genevieve; Gomez, Dennis
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收藏Antitrypanosomatid Pharmacomodulation at Position 3 of the 8-Nitroquinolin-2(1H)-one Scaffold Using Palladium-Catalysed Cross-Coupling Reactions
Pedron, Julien; Boudot, Clotilde; Bourgeade-Delmas, Sandra; Sournia-Saquet, Alix; Paloque, Lucie; Rastegari, Maryam; Abdoulaye, Mansour; El-Kashef, Hussein; Bonduelle, Colin; Pratviel, Genevieve; Wyllie, Susan; Fairlamb, Alan H.; Courtioux, Bertrand; Verhaeghe, Pierre; Valentin, Alexis
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收藏8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a] pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductases
Fersing, Cyril; Boudot, Clotilde; Pedron, Julien; Hutter, Sebastien; Primas, Nicolas; Castera-Ducros, Caroline; Bourgeade-Delmas, Sandra; Sournia-Saquet, Alix; Moreau, Alain; Cohen, Anita; Stigliani, Jean-Luc; Pratviel, Genevieve; Crozet, Maxime D.; Wyllie, Susan; Fairlamb, Alan; Valentin, Alexis; Rathelot, Pascal; Azas, Nadine; Courtioux, Bertrand; Verhaeghe, Pierre; Vanelle, Patrice
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收藏Novel 8-nitroquinolin-2(1H)-ones as NTR-bioactivated antikinetoplastid molecules: Synthesis, electrochemical and SAR study
Pedron, Julien; Boudot, Clotilde; Hutter, Sebastien; Bourgeade-Delmas, Sandra; Stigliani, Jean -Luc; Sournia-Saquet, Alix; Moreau, Alain; Boutet-Robinet, Elisa; Paloque, Lucie; Mothes, Emmanuelle; Laget, Michele; Vendier, Laure; Pratviel, Genevieve; Wyllie, Susan; Fairlamb, Alan; Azas, Nadine; Courtioux, Bertrand; Valentin, Alexis; Verhaeghe, Pierre
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收藏Crystal structure of the enoyl-ACP reductase of Mycobacterium tuberculosis (InhA) in the apo-form and in complex with the active metabolite of isoniazid pre-formed by a biomimetic approach
Chollet, Aurelien; Mourey, Lionel; Lherbet, Christian; Delbot, Alexandra; Julien, Sylviane; Baltas, Michel; Bernadou, Jean; Pratviel, Genevieve; Maveyraud, Laurent; Bernardes-Genisson, Vania
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收藏Cobalt(III)porphyrin to target G-quadruplex DNA
Sabater, Laurent; Fang, Pei-Ju; Chang, Chi-Fon; De Rache, Aurore; Prado, Enora; Dejeu, Jerome; Garofalo, Antonio; Lin, Jung-Hsin; Mergny, Jean-Louis; Defrancq, Eric; Pratviel, Genevieve
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