Jan Balzarini - Publications, H-index & Citations

Jan Balzarini

KU Leuven

59H指数

1.1K论文数

1.4W被引数

收录论文 155

发表时间

Benzothiazole Derivatives as Multifunctional Antioxidant Agents for Skin Damage: Structure-Activity Relationship of a Scaffold Bearing a Five-Membered Ring System

ANTIOXIDANTS

IF6.6

2022-02-17

OAAI

Djuidje, Ernestine Nicaise; Barbari, Riccardo; Baldisserotto, Anna; Durini, Elisa; Sciabica, Sabrina; Balzarini, Jan; Liekens, Sandra; Vertuani, Silvia; Manfredini, Stefano

Synthesis and Biological Evaluation of New Antitubulin Agents Containing 2-(3′,4′,5′-trimethoxyanilino)-3,6-disubstituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine Scaffold

MOLECULES

IF4.6

2020-04-07

OAAI

Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Cacciari, Barbara; Balzarini, Jan; Liekens, Sandra; Hamel, Ernest; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Zurlo, Matteo; Finotti, Alessia; Gambari, Roberto

Direct arylation of C60Cl6 and C70Cl8 with carboxylic acids: a synthetic avenue to water-soluble fullerene derivatives with promising antiviral activity

CHEMICAL COMMUNICATIONS

IF4.2

2020-01-01

OAAI

Kraevaya, Olga A.; Peregudov, Alexander S.; Godovikov, Ivan A.; Shchurik, Elena, V; Martynenko, Vyacheslav M.; Shestakov, Alexander F.; Balzarini, Jan; Schols, Dominique; Troshin, Pavel A.

Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3′,4′,5′-trimethoxyphenyl)-3-(2′-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a molecular hybridisation approach

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2018-08-24

OAAI

Preti, Delia; Romagnoli, Romeo; Rondanin, Riccardo; Cacciari, Barbara; Hamel, Ernest; Balzarini, Jan; Liekens, Sandra; Schols, Dominique; Estevez-Sarmiento, Francisco; Quintana, Jose; Estevez, Francisco

2-Alkoxycarbonyl-3-arylamino-5-substituted thiophenes as a novel class of antimicrotubule agents: Design, synthesis, cell growth and tubulin polymerization inhibition

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2018-01-01

OAAI

Romagnoli, Romeo; Kimatrai Salvador, Maria; Schiaffino Ortega, Santiago; Baraldi, Pier Giovanni; Oliva, Paola; Baraldi, Stefania; Carlota Lopez-Cara, Luisa; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Balzarini, Jan; Liekens, Sandra; Mattiuzzo, Elena; Basso, Giuseppe; Viola, Giampietro

Surface Glycans: A Therapeutic Opportunity for Kinetoplastid Diseases (vol. 33, pg. 775, 2017)

Trends in Parasitology

IF6.6

2017-12-01

OAAI

Castillo-Acosta, Victor M.; Balzarini, Jan; Gonzalez-Pacanowska, Dolores

A Multitarget Approach toward the Development of 8-Substituted Purines for Photoprotection and Prevention of UV-Related Damage

CHEMMEDCHEM

IF3.4

2017-05-03

OAAI

Djuidje, Ernestine N.; Dissette, Valeria; Bino, Alessia; Benetti, Simonetta; Balzarini, Jan; Liekens, Sandra; Manfredini, Stefano; Vertuani, Silvia; Baldisserotto, Anna

High mannose-specific lectin Msl mediates key interactions of the vaginal Lactobacillus plantarum isolate CMPG5300

SCIENTIFIC REPORTS

IF3.9

2016-11-17

OAAI

Malik, Shweta; Petrova, Mariya I.; Imholz, Nicole C. E.; Verhoeven, Tine L. A.; Noppen, Sam; Van Damme, Els J. M.; Liekens, Sandra; Balzarini, Jan; Schols, Dominique; Vanderleyden, Jos; Lebeer, Sarah

Conformational States of HIV-1 Reverse Transcriptase for Nucleotide Incorporation vs Pyrophosphorolysis Binding of Foscarnet (vol 11, pg 2158, 2016)

ACS CHEMICAL BIOLOGY

IF3.8

2016-09-26

OAAI

Das, Kalyan; Balzarini, Jan; Miller, Matthew T.; Maguire, Anita R.; DeStefano, Jeffrey J.; Arnold, Eddy

Carbohydrate-Binding Non-Peptidic Pradimicins for the Treatment of Acute Sleeping Sickness in Murine Models

PLOS PATHOGENS

IF4.9

2016-09-23

OAAI

Castillo-Acosta, Victor M.; Ruiz-Perez, Luis M.; Etxebarria, Juan; Reichardt, Niels C.; Navarro, Miguel; Igarashi, Yasuhiro; Liekens, Sandra; Balzarini, Jan; Gonzalez-Pacanowska, Dolores

Niacin esters of chalcones with tumor-selective properties

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2016-06-02

OAAI

Panda, Atulya K.; Das, Umashankar; Roayapalley, Praveen K.; Sakagami, Hiroshi; Kawase, Masami; Balzarini, Jan; De Clercq, Erik; Dimmock, Jonathan R.

Tumour-specific cytotoxicity and structure-activity relationships of novel 1-[3-(2-methoxyethylthio)propionyl]-3,5-bis(benzylidene)-4-piperidones

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2016-05-01

PREAI

Hossain, Mohammad; Das, Umashankar; Umemura, Naoki; Sakagami, Hiroshi; Balzarini, Jan; De Clercq, Erik; Kawase, Masami; Dimmock, Jonathan R.

Design, Synthesis and Evaluation of Antiproliferative Activity of New Benzimidazolehydrazones 新型苯并咪唑腙的设计、合成及抗增殖活性评价

MOLECULES

IF4.6

2016-04-30

OAAI

Onnis, Valentina; Demurtas, Monica; Deplano, Alessandro; Balboni, Gianfranco; Baldisserotto, Anna; Manfredini, Stefano; Pacifico, Salvatore; Liekens, Sandra; Balzarini, Jan

Screening Platform toward New Anti-HIV Aptamers Set on Molecular Docking and Fluorescence Quenching Techniques

ANALYTICAL CHEMISTRY

IF6.7

2016-02-05

PREAI

Oliviero, Giorgia; Stornaiuolo, Mariano; D'Atri, Valentina; Nici, Fabrizia; Yousif, Ali Munaim; D'Errico, Stefano; Piccialli, Gennaro; Mayol, Luciano; Novellino, Ettore; Marinelli, Luciana; Grieco, Paolo; Carotenuto, Alfonso; Noppen, Sam; Liekens, Sandra; Balzarini, Jan; Borbone, Nicola

A novel family of diarylpyrimidines (DAPYs) featuring a diatomic linker: Design, synthesis and anti-HIV activities

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2015-10-01

PREAI

Gu, Shuang-Xi; Qiao, Heng; Zhu, Yuan-Yuan; Shu, Qi-Chao; Liu, Hui; Ju, Xiu-Lian; De Clercq, Erik; Balzarini, Jan; Pannecouque, Christophe

Curcumin-inspired cytotoxic 3,5-bis(arylmethylene)-1-(N-(ortho-substituted aryl) maleamoyl)-4-piperidones: A novel group of topoisomerase II alpha inhibitors

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2015-10-01

PREAI

Jha, Amitabh; Duffield, Katherine M.; Ness, Matthew R.; Ravoori, Sujatha; Andrews, Gabrielle; Bhullar, Khushwant S.; Rupasinghe, H. P. Vasantha; Balzarini, Jan

Antiproliferative activities of halogenated pyrrolo[3,2-d]pyrimidines

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2015-08-01

OAAI

Temburnikar, Kartik W.; Ross, Christina R.; Wilson, Gerald M.; Balzarini, Jan; Cawrse, Brian M.; Seley-Radtke, Katherine L.

Design, synthesis and bioevaluation of novel 6-(4-Hydroxypiperidino)naphthalen-2-ol-based potential Selective Estrogen Receptor Modulators for breast cancer

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2015-03-01

PREAI

Jha, Amitabh; Yadav, Yogesh; Naidu, Ajay B.; Rao, V. Kameswara; Kumar, Anil; Parmar, Virinder S.; MacDonald, William J.; Too, Catherine K. L.; Balzarini, Jan; Barden, Christopher J.; Cameron, T. Stanley

Dipeptidyl-Peptidase IV (DPP IV/CD26)-Activated Prodrugs: A Successful Strategy for Improving Water Solubility and Oral Bioavailability

CURRENT MEDICINAL CHEMISTRY

IF3.5

2015-02-16

OAAI

Velazquez, Sonsoles; de Castro, Sonia; Diez-Torrubia, Alberto; Balzarini, Jan; Camarasa, Maria-Jose

Synthesis and biological evaluation of phosphoramidate prodrugs of two analogues of 2-deoxy-D-ribose-1-phosphate directed to the discovery of two carbasugars as new potential anti-HIV leads 两种2-脱氧-d-核糖-1-磷酸类似物的氨基磷酸酯前药的合成和生物学评估，旨在发现两种carbasugars作为新的潜在抗HIV线索

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2015-02-01

OAAI

Hamon, Nadege; Slusarczyk, Magdalena; Serpi, Michaela; Balzarini, Jan; McGuigan, Christopher

研究方向