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收藏Granulocyte-macrophage colony-stimulating factor (GM-CSF) as a therapeutic target in psoriasis: randomized, controlled investigation using namilumab, a specific human anti-GM-CSF monoclonal antibody
Papp, K. A.; Gooderham, M.; Jenkins, R.; Vender, R.; Szepietowski, J. C.; Wagner, T.; Hunt, B.; Souberbielle, B.; Hartman, I; Kunynetz, R.; Lynde, C.; Narbutt, J.; Poulin, Y.; Poznanska, M.; Raman, M.; Reich, K.; Rosoph, L.; Septe, M.; Viba, D.; Wasel, N.; Zachariae, C.; Falk, T. M.
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收藏Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of Single Rising TAK-438 (Vonoprazan) Doses in Healthy Male Japanese/non-Japanese Subjects
Sakurai, Yuuichi; Nishimura, Akira; Kennedy, Gale; Hibberd, Mark; Jenkins, Richard; Okamoto, Hiroyuki; Yoneyama, Tomoki; Jenkins, Helen; Ashida, Kiyoshi; Irie, Shin; Taeubel, Joerg
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收藏Randomised clinical trial: safety, tolerability, pharmacokinetics and pharmacodynamics of repeated doses of TAK-438 (vonoprazan), a novel potassium-competitive acid blocker, in healthy male subjects
Jenkins, H.; Sakurai, Y.; Nishimura, A.; Okamoto, H.; Hibberd, M.; Jenkins, R.; Yoneyama, T.; Ashida, K.; Ogama, Y.; Warrington, S.
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收藏Increases in Oxidized Low-Density Lipoprotein and Other Inflammatory and Adhesion Molecules With a Concomitant Decrease in High-Density Lipoprotein in the Individuals Exposed to Arsenic in Bangladesh
Karim, Md Rezaul; Rahman, Mashiur; Islam, Khairul; Al Mamun, Abdullah; Hossain, Shakhawoat; Hossain, Ekhtear; Aziz, Abdul; Yeasmin, Fouzia; Agarwal, Smita; Hossain, Md Imam; Saud, Zahangir Alam; Nikkon, Farjana; Hossain, Mostaque; Mandal, Abul; Jenkins, Richard O.; Haris, Parvez I.; Miyataka, Hideki; Himeno, Seiichiro; Hossain, Khaled
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收藏AZD8055 Is a Potent, Selective, and Orally Bioavailable ATP-Competitive Mammalian Target of Rapamycin Kinase Inhibitor with In vitro and In vivo Antitumor ActivityAZD8055是雷帕霉素激酶抑制剂的有效,选择性和口服生物可利用的ATP竞争性哺乳动物靶标,具有体外和体内抗肿瘤活性
Chresta, Christine M.; Davies, Barry R.; Hickson, Ian; Harding, Tom; Cosulich, Sabina; Critchlow, Susan E.; Vincent, John P.; Ellston, Rebecca; Jones, Darren; Sini, Patrizia; James, Dominic; Howard, Zoe; Dudley, Phillippa; Hughes, Gareth; Smith, Lisa; Maguire, Sharon; Hummersone, Marc; Malagu, Karine; Menear, Keith; Jenkins, Richard; Jacobsen, Matt; Smith, Graeme C. M.; Guichard, Sylvie; Pass, Martin
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收藏AZD6244 (ARRY-142886), a potent inhibitor of mitogen-activated protein kinase/extracellular signal-regulated kinase kinase 1/2 kinases:: mechanism of action in vivo, pharmacokinetic/pharmacodynamic relationship, and potential for combination in preclinical models
Davies, Barry R.; Logie, Armelle; McKay, Jennifer S.; Martin, Paul; Steele, Samantha; Jenkins, Richard; Cockerill, Mark; Cartlidge, Sue; Smith, Paul D.
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