未登录Machine learning-driven insights into retention mechanism in IAM chromatography of anticancer sulfonamides: Implications for biological efficacy机器学习驱动的抗肿瘤磺酰胺在IAM色谱中保留机制的见解:对生物效力的启示
Nisterenko, Wiktor; Zolnowska, Beata; Deng, Jiayin; Zgoda, Dominika; Rozycka, Alicja; Greber, Katarzyna Ewa; Pogorzelska, Aneta; Szafranski, Krzysztof; Bulakowska, Anita; Tomorowicz, Lukasz; Kawiak, Anna; Sawicki, Wieslaw; Ouyang, Defang; Slawinski, Jaroslaw; Ciura, Krzesimir
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收藏Modification of gradient HPLC method for determination of small molecules' affinity to human serum albumin under column safety conditions: Robustness and chemometrics study
Wozinski, Mateusz; Greber, Katarzyna Ewa; Pastewska, Monika; Kolasinski, Piotr; Hewelt-Belka, Weronika; Zolnowska, Beata; Slawinski, Jaroslaw; Szulczyk, Daniel; Sawicki, Wieslaw; Ciura, Krzesimir
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收藏Target-based drug discovery through inversion of quantitative structure-drug-property relationships and molecular simulation: CA IX-sulphonamide complexes
Zuvela, Petar; Liu, J. Jay; Yi, Myunggi; Pomastowski, Pawel P.; Sagandykova, Gulyaim; Belka, Mariusz; David, Jonathan; Baczek, Tomasz; Szafranski, Krzysztof; Zolnowska, Beata; Slawinski, Jaroslaw; Supuran, Claudiu T.; Wong, Ming Wah; Buszewski, Boguslaw
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收藏Synthesis, molecular structure, and metabolic stability of new series of N′-(2-alkylthio-4-chloro-5-methylbenzenesulfonyl)-1-(5-phenyl-1H- pyrazol-1-yl)amidine as potential anti-cancer agents
Pogorzelska, Aneta; Slawinski, Jaroslaw; Kawiak, Anna; Zolnowska, Beata; Chojnacki, Jaroslaw; Stasilojc, Grzegorz; Ulenberg, Szymon; Szafranski, Krzysztof; Baczek, Tomasz
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收藏Novel 2-(2-arylmethylthio-4-chloro-5-methylbenzenesulfonyl)-1-(1,3,5-triazin-2-ylamino)guanidine derivatives: Inhibition of human carbonic anhydrase cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII, anticancer activity, and molecular modeling studies
Zolnowska, Beata; Slawinski, Jaroslaw; Szafranski, Krzysztof; Angeli, Andrea; Supuran, Claudiu T.; Kawiak, Anna; Wieczor, Milosz; Zielinska, Joanna; Baczek, Tomasz; Bartoszewska, Sylwia
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收藏Novel 2-(2-alkylthiobenzenesulfony1)-3-(phenylprop-2-ynylideneamino)guanidine derivatives as potent anticancer agents - Synthesis, molecular structure, QSAR studies and metabolic stability
Pogorzelska, Aneta; Slawinski, Jaroslaw; Zolnowska, Beata; Szafranski, Krzysztof; Kawiak, Anna; Chojnacki, Jaroslaw; Ulenberg, Szymon; Zielinska, Joanna; Baczek, Tomasz
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收藏Novel 2-benzylthio-5-(1,3,4-oxadiazol-2-yl)benzenesulfonamides with anticancer activity: Synthesis, QSAR study, and metabolic stability
Slawinski, Jaroslaw; Szafranski, Krzysztof; Pogorzelska, Aneta; Zolnowska, Beata; Kawiak, Anna; Macur, Katarzyna; Belka, Mariusz; Baczek, Tomasz
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收藏Synthesis, QSAR studies, and metabolic stability of novel 2-alkylthio-4-chloro-N-(5-oxo-4,5-dihydro-1,2,4-triazin-3-yl)benzenesulfonamide derivatives as potential anticancer and apoptosis-inducing agents
Zolnowska, Beata; Slawinski, Jaroslaw; Pogorzelska, Aneta; Szafranski, Krzysztof; Kawiak, Anna; Stasilojc, Grzegorz; Belka, Mariusz; Zielinska, Joanna; Baczek, Tomasz
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收藏Novel 5-Substituted 2-(Aylmethylthio)-4-chloro-N-( 5-aryl-1,2,4-triazin-3-yl)benzenesulfonamides: Synthesis, Molecular Structure, Anticancer Activity, Apoptosis-Inducing Activity and Metabolic Stability
Zolnowska, Beata; Slawinski, Jaroslaw; Pogorzelska, Aneta; Szafranski, Krzysztof; Kawiak, Anna; Stasilojc, Grzegorz; Belka, Mariusz; Ulenberg, Szymon; Baczek, Tomasz; Chojnacki, Jaroslaw
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收藏Synthesis of Novel Pyrido[4,3-e][1,2,4]triazino[3,2-c][1,2,4] thiadiazine 6,6-dioxide Derivatives with Potential Anticancer Activity具有潜在抗癌活性的新型吡啶并 [4,3-e][1,2,4] 三嗪 [3,2-c][1,2,4] 噻二嗪6,6-二氧化物衍生物的合成
Slawinski, Jaroslaw; Grzonek, Aleksandra; Zolnowska, Beata; Kawiak, Anna
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收藏Synthesis, Molecular Structure, Metabolic Stability and QSAR Studies of a Novel Series of Anticancer N-Acylbenzenesulfonamides
Zolnowska, Beata; Slawinski, Jaroslaw; Belka, Mariusz; Baczek, Tomasz; Kawiak, Anna; Chojnacki, Jaroslaw; Pogorzelska, Aneta; Szafranski, Krzysztof
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