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Conformational dynamics and asymmetry in multimodal inhibition of membrane-bound pyrophosphatases 膜结合焦磷酸酶多模式抑制中的构象动力学与不对称性 Liu, Jianing; Shah, Anokhi; Liu, Xinyu; Wort, Joshua L.; Ma, Yue; Hardman, Katie; Johansson, Niklas G.; Ribeiro, Orquidea; Brookfield, Adam; Bowen, Alice; Yli-Kauhaluoma, Jari; Xhaard, Henri; Jeuken, Lars J. C.; Goldman, Adrian; Pliotas, Christos; Vidilaseris, Keni 分享 收藏
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Switching of hypertrophic signalling towards enhanced cardiomyocyte identity and maturity by a GATA4-targeted compound Pohjolainen, Lotta; Kinnunen, Sini M.; Auno, Samuli; Kiriazis, Alexandros; Pohjavaara, Saana; Kari-Koskinen, Julia; Zore, Matej; Jumppanen, Mikael; Yli-Kauhaluoma, Jari; Talman, Virpi; Ruskoaho, Heikki; Valimaki, Mika J. 分享 收藏
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Probing the Interactions of Thiazole Abietane Inhibitors with the Human Serine Hydrolases ABHD16A and ABHD12 Ahonen, Tiina J.; Ng, Choa P.; Farinha, Beatriz; Almeida, Barbara; Victor, Bruno L.; Reynolds, Christopher; Kalso, Eija; Yli-Kauhaluoma, Jari; Greaves, Jennifer; Moreira, Vania M. 分享 收藏
Azulene as a biphenyl mimetic in orexin/hypocretin receptor agonists Leino, Teppo O.; Turku, Ainoleena; Urvas, Lauri; Adhikari, Karuna; Oksanen, Jouni; Steynen, Yana; Yli-Kauhaluoma, Jari; Xhaard, Henri; Kukkonen, Jyrki P.; Wallen, Erik A. A. 分享 收藏
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Expanding the Paradigm of Structure-Based Drug Design: Molecular Dynamics Simulations Support the Development of New Pyridine-Based Protein Kinase C-Targeted Agonists Lautala, Saara; Provenzani, Riccardo; Tarvainen, Ilari; Sirna, Katia; Karhu, S. Tuuli; Grazhdankin, Evgeni; Lehtinen, Antti K.; Sa'd, Hanan; Koivuniemi, Artturi; Xhaard, Henri; Tuominen, Raimo K.; Talman, Virpi; Bunker, Alex; Yli-Kauhaluoma, Jari 分享 收藏
Selected strategies to fight pathogenic bacteria Plotniece, Aiva; Sobolev, Arkadij; Supuran, Claudiu T.; Carta, Fabrizio; Bjoerkling, Fredrik; Franzyk, Henrik; Yli-Kauhaluoma, Jari; Augustyns, Koen; Cos, Paul; De Vooght, Linda; Govaerts, Matthias; Aizawa, Juliana; Tammela, Paeivi; Zalubovskis, Raivis 分享 收藏
Utilizing PET and MALDI Imaging for Discovery of a Targeted Probe for Brain Endocannabinoid α/β-Hydrolase Domain 6 (ABHD6) Mardon, Karine; Patel, Jayendra Z.; Savinainen, Juha R.; Stimson, Damion H. R.; Oyagawa, Caitlin R. M.; Grimsey, Natasha L.; Migotto, Mary-anne; Njiru, Grace F. M.; Hamilton, Brett R.; Cowin, Gary; Yli-Kauhaluoma, Jari; Vanduffel, Wim; Blakey, Idriss; Bhalla, Rajiv; Cawthorne, Christopher; Celen, Sofie; Bormans, Guy; Thurecht, Kristofer J.; Ahamed, Muneer 分享 收藏
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Anthranilamides with quinoline and β-carboline scaffolds: design, synthesis, and biological activity 喹啉和 β-咔啉支架的邻氨基苯甲酰胺: 设计,合成和生物活性 Beus, Maja; Persoons, Leentje; Daelemans, Dirk; Schols, Dominique; Savijoki, Kirsi; Varmanen, Pekka; Yli-Kauhaluoma, Jari; Pavic, Kristina; Zorc, Branka 分享 收藏
Computationally prioritized drugs inhibit SARS-CoV-2 infection and syncytia formation Serra, Angela; Fratello, Michele; Federico, Antonio; Ojha, Ravi; Provenzani, Riccardo; Tasnadi, Ervin; Cattelani, Luca; del Giudice, Giusy; Kinaret, Pia A. S.; Saarimaki, Laura A.; Pavel, Alisa; Kuivanen, Suvi; Cerullo, Vincenzo; Vapalahti, Olli; Horvath, Peter; Di Lieto, Antonio; Yli-Kauhaluoma, Jari; Balistreri, Giuseppe; Greco, Dario 分享 收藏