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Srinivas Chamakuri

baylor college of medicine

13H指数
40论文数
684被引数
收录论文 22
发表时间
A small molecule inhibits Ebola virus entry through glycoprotein stabilization小分子通过糖蛋白稳定化抑制埃博拉病毒进入
err2026-09-01
err0
errOAAI
errFan Bu; Gang Ye; Kiran L. Sharma; Bruno La Rosa; Murugesan Palaniappan; Martin M. Matzuk; Damian W. Young; Hailey Turner-Hubbard; Kimberly Morsheimer; Callum Owen; Katalin Toth; Michael Cameron; Robert Davey; Srinivas Chamakuri; Peter Dosa; Fang Li
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MYC-Targeting PROTACs Lead to Bimodal Degradation and N-Terminal Truncation
err2025-03-01
err0
PREAI
errBoyd, Shelton R.; Chamakuri, Srinivas; Trostle, Alexander J.; Chen, Hu; Liu, Zhandong; Jian, Antrix; Wang, Jian; Malovannaya, Anna; Young, Damian W.
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Discovery of highly potent and ALK2/ALK 1 selective kinase inhibitors using DNA- encoded chemistry technology
err2024-11-14
err0
errOAAI
errJimmidi, Ravikumar; Monsivais, Diana; Ta, Hai Minh; Sharma, Kiran L.; Bohren, Kurt M.; Chamakuri, Srinivas; Liao, Zian; Li, Feng; Hakenjos, John M.; Li, Jian - Yuan; Mishina, Yuji; Pan, Haichun; Qin, Xuan; Robers, Matthew B.; Sankaran, Banumathi; Tan, Zhi; Tang, Suni; Vasquez, Yasmin M.; Wilkinson, Jennifer; Young, Damian W.; Palmer, Stephen S.; Mackenzie, Kevin R.; Kim, Choel; Matzuk, Martin M.
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Synthesis and Optimization of Small Molecule Inhibitors of Prostate Specific Antigen
err2024-08-05
err0
PREAI
errErickson, Jeffery A.; Jimmidi, Ravikumar; Anamthathmakula, Prashanth; Qin, Xuan; Wang, Jian; Gong, Leyi; Park, Jaehyeon; Koolpe, Gary; Tan, Caitlin; Matzuk, Martin M.; Li, Feng; Chamakuri, Srinivas; Winuthayanon, Wipawee
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Expanding Complex Morpholines Using Systematic Chemical Diversity
err2024-03-20
err1
PREAI
errTang, Sunny Ann; Fults, Afton; Boyd, Shelton R.; Gattu, Nikhil; Tran, Kevin A.; Fan, Jiayi; Mackenzie, Kevin R.; Palzkill, Timothy; Young, Damian W.; Chamakuri, Srinivas
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Chemical Catalysis Guides Structural Identification for the Major In Vivo Metabolite of the BET Inhibitor JQ1
err2024-01-02
err3
errOAAI
errHolmes, Secondra; Jain, Prashi; Rodriguez, Kenneth Guzman; Williams, Jade; Yu, Zhifeng; Cerda-Smith, Christian; Samuel, Errol L. G.; Campbell, James; Hakenjos, John Michael; Monsivais, Diana; Li, Feng; Chamakuri, Srinivas; Matzuk, Martin M.; Santini, Conrad; Mackenzie, Kevin R.; Young, Damian W.
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Exploiting the Carboxylate-Binding Pocket of β-Lactamase Enzymes Using a Focused DNA-Encoded Chemical Library
err2023-12-20
err3
PREAI
errPark, Suhyeorn; Fan, Jiayi; Chamakuri, Srinivas; Palaniappan, Murugesan; Sharma, Kiran; Qin, Xuan; Wang, Jian; Tan, Zhi; Judge, Allison; Hu, Liya; Sankaran, Banumathi; Li, Feng; Prasad, B. V. Venkataram; Matzuk, Martin M.; Palzkill, Timothy
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Heterocyclic Merging of Stereochemically Diverse Chiral Piperazines and Morpholines with Indazoles
err2023-08-29
err2
errOAAI
errViveki, Amol B.; Mansfield, Timothy M.; Tran, Kevin A.; Lenkeit, Evan; Mackenzie, Kevin R.; Young, Damian W.; Chamakuri, Srinivas
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DNA-encoded chemical libraries yield non-covalent and non-peptidic SARS-CoV-2 main protease inhibitors
err2023-08-04
err8
errOAAI
errJimmidi, Ravikumar; Chamakuri, Srinivas; Lu, Shuo; Ucisik, Melek Nihan; Chen, Peng-Jen; Bohren, Kurt M.; Moghadasi, Seyed Arad; Versteeg, Leroy; Nnabuife, Christina; Li, Jian-Yuan; Qin, Xuan; Chen, Ying-Chu; Faver, John C.; Nyshadham, Pranavanand; Sharma, Kiran L.; Sankaran, Banumathi; Judge, Allison; Yu, Zhifeng; Li, Feng; Pollet, Jeroen; Harris, Reuben S.; Matzuk, Martin M.; Palzkill, Timothy; Young, Damian W.
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Gain-of-Signal Assays for Probing Inhibition of SARS-CoV-2 Mpro/3CLpro in Living Cells
errMBIO
IF4.7
err2022-06-28
err22
errOAAI
errMoghadasi, Seyed Arad; Esler, Morgan A.; Otsuka, Yuka; Becker, Jordan T.; Moraes, Sofia N.; Anderson, Constance B.; Chamakuri, Srinivas; Belica, Christopher; Wick, Chloe; Harki, Daniel A.; Young, Damian W.; Scampavia, Louis; Spicer, Timothy P.; Shi, Ke; Aihara, Hideki; Brown, William L.; Harris, Reuben S.
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Trisubstituted triumph
err2022-06-06
err0
PREAI
errYoung, Damian W.; Chamakuri, Srinivas
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A Concise Synthetic Method for Constructing 3-Substituted Piperazine-2-Acetic Acid Esters from 1,2-Diamines
err2022-05-25
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errOAAI
errChamakuri, Srinivas; Tang, Sunny Ann; Tran, Kevin A.; Guduru, Shiva Krishna Reddy; Bolin, Peter K.; MacKenzie, Kevin R.; Young, Damian W.
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Oleic acid is an endogenous ligand of TLX/NR2E1 that triggers hippocampal neurogenesis油酸是触发海马神经发生的TLX/NR2E1的内源性配体
err2022-03-25
err42
errOAAI
errKandel, Prasanna; Semerci, Fatih; Mishra, Rachana; Choi, William; Bajic, Aleksandar; Baluya, Dodge; Ma, LiHua; Chen, Kevin; Cao, Austin C.; Phongmekhin, Tipwarin; Matinyan, Nick; Jimenez-Panizo, Alba; Chamakuri, Srinivas; Raji, Idris O.; Chang, Lyra; Fuentes-Prior, Pablo; MacKenzie, Kevin R.; Benn, Caroline L.; Estebanez-Perpina, Eva; Venken, Koen; Moore, David D.; Young, Damian W.; Maletic-Savatic, Mirjana
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Design and construction of a stereochemically diverse piperazine-based DNA-encoded chemical library
err2021-10-01
err10
PREAI
errChamakuri, Srinivas; Chung, Mee-Kyung; Samuel, Errol L. G.; Tran, Kevin A.; Chen, Ying-Chu; Nyshadham, Pranavanand; Santini, Conrad; Matzuk, Martin M.; Young, Damian W.
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DNA-encoded chemistry technology yields expedient access to SARS-CoV-2 Mpro inhibitors
err2021-08-23
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errOAAI
errChamakuri, Srinivas; Lu, Shuo; Ucisik, Melek Nihan; Bohren, Kurt M.; Chen, Ying-Chu; Du, Huang-Chi; Faver, John C.; Jimmidi, Ravikumar; Li, Feng; Li, Jian-Yuan; Nyshadham, Pranavanand; Palmer, Stephen S.; Pollet, Jeroen; Qin, Xuan; Ronca, Shannon E.; Sankaran, Banumathi; Sharma, Kiran L.; Tan, Zhi; Versteeg, Leroy; Yu, Zhifeng; Matzuk, Martin M.; Palzkill, Timothy; Young, Damian W.
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Synthesis of Enantiomerically Pure 6-Substituted-Piperazine-2-Acetic Acid Esters as Intermediates for Library Production (vol 83, pg 6541, 2018)
err2019-03-11
err0
PREAI
errChamakuri, Srinivas; Jain, Prashi; Guduru, Shiva Reddy Krishna; Arney, J. Winston; MacKenzie, Kevin R.; Santini, Conrad; Young, Damian W.
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Synthesis of Enantiomerically Pure 5-Substituted Piperazine-2-Acetic Acid Esters as Intermediates for Library Production
err2019-03-08
err12
PREAI
errJain, Prashi; Raji, Idris O.; Chamakuri, Srinivas; MacKenzie, Kevin R.; Ebright, Brandon T.; Santini, Conrad; Young, Damian W.
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Synthesis of Enantiomerically Pure 3-Substituted Piperazine-2-acetic Acid Esters as Intermediates for Library Production
err2018-09-05
err19
PREAI
errGuduru, Shiva Krishna Reddy; Chamakuri, Srinivas; Raji, Idris O.; MacKenzie, Kevin R.; Santini, Conrad; Young, Damian W.
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Synthesis of Enantiomerically Pure 6-Substituted-Piperazine-2-Acetic Acid Esters as Intermediates for Library Production
err2018-05-11
err21
PREAI
errChamakuri, Srinivas; Jain, Prashi; Guduru, Shiva Krishna Reddy; Arney, J. Winston; MacKenzie, Kevin R.; Santini, Conrad; Young, Damian W.
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