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Metabolism, Pharmacokinetics, and Tissue Distribution of a Selective FK506-Binding Protein 12 F36V Mutant Degrader in Mice 代谢、药代动力学及组织分布:一种选择性FK506结合蛋白12 F36V突变体降解剂在小鼠中的研究 Zhou, Shenzhi; Qin, Xuan; Tran, Kevin; Wang, Jian; Ji, Xingyu; Mackenzie, Kevin R.; Chamakuri, Srinivas; Wang, Jin; Li, Feng 分享 收藏
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Discovery of highly potent and ALK2/ALK 1 selective kinase inhibitors using DNA- encoded chemistry technology Jimmidi, Ravikumar; Monsivais, Diana; Ta, Hai Minh; Sharma, Kiran L.; Bohren, Kurt M.; Chamakuri, Srinivas; Liao, Zian; Li, Feng; Hakenjos, John M.; Li, Jian - Yuan; Mishina, Yuji; Pan, Haichun; Qin, Xuan; Robers, Matthew B.; Sankaran, Banumathi; Tan, Zhi; Tang, Suni; Vasquez, Yasmin M.; Wilkinson, Jennifer; Young, Damian W.; Palmer, Stephen S.; Mackenzie, Kevin R.; Kim, Choel; Matzuk, Martin M. 分享 收藏
Synthesis and Optimization of Small Molecule Inhibitors of Prostate Specific Antigen Erickson, Jeffery A.; Jimmidi, Ravikumar; Anamthathmakula, Prashanth; Qin, Xuan; Wang, Jian; Gong, Leyi; Park, Jaehyeon; Koolpe, Gary; Tan, Caitlin; Matzuk, Martin M.; Li, Feng; Chamakuri, Srinivas; Winuthayanon, Wipawee 分享 收藏
Expanding Complex Morpholines Using Systematic Chemical Diversity Tang, Sunny Ann; Fults, Afton; Boyd, Shelton R.; Gattu, Nikhil; Tran, Kevin A.; Fan, Jiayi; Mackenzie, Kevin R.; Palzkill, Timothy; Young, Damian W.; Chamakuri, Srinivas 分享 收藏
Chemical Catalysis Guides Structural Identification for the Major In Vivo Metabolite of the BET Inhibitor JQ1 Holmes, Secondra; Jain, Prashi; Rodriguez, Kenneth Guzman; Williams, Jade; Yu, Zhifeng; Cerda-Smith, Christian; Samuel, Errol L. G.; Campbell, James; Hakenjos, John Michael; Monsivais, Diana; Li, Feng; Chamakuri, Srinivas; Matzuk, Martin M.; Santini, Conrad; Mackenzie, Kevin R.; Young, Damian W. 分享 收藏
Exploiting the Carboxylate-Binding Pocket of β-Lactamase Enzymes Using a Focused DNA-Encoded Chemical Library Park, Suhyeorn; Fan, Jiayi; Chamakuri, Srinivas; Palaniappan, Murugesan; Sharma, Kiran; Qin, Xuan; Wang, Jian; Tan, Zhi; Judge, Allison; Hu, Liya; Sankaran, Banumathi; Li, Feng; Prasad, B. V. Venkataram; Matzuk, Martin M.; Palzkill, Timothy 分享 收藏
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DNA-encoded chemical libraries yield non-covalent and non-peptidic SARS-CoV-2 main protease inhibitors Jimmidi, Ravikumar; Chamakuri, Srinivas; Lu, Shuo; Ucisik, Melek Nihan; Chen, Peng-Jen; Bohren, Kurt M.; Moghadasi, Seyed Arad; Versteeg, Leroy; Nnabuife, Christina; Li, Jian-Yuan; Qin, Xuan; Chen, Ying-Chu; Faver, John C.; Nyshadham, Pranavanand; Sharma, Kiran L.; Sankaran, Banumathi; Judge, Allison; Yu, Zhifeng; Li, Feng; Pollet, Jeroen; Harris, Reuben S.; Matzuk, Martin M.; Palzkill, Timothy; Young, Damian W. 分享 收藏
Gain-of-Signal Assays for Probing Inhibition of SARS-CoV-2 Mpro/3CLpro in Living Cells Moghadasi, Seyed Arad; Esler, Morgan A.; Otsuka, Yuka; Becker, Jordan T.; Moraes, Sofia N.; Anderson, Constance B.; Chamakuri, Srinivas; Belica, Christopher; Wick, Chloe; Harki, Daniel A.; Young, Damian W.; Scampavia, Louis; Spicer, Timothy P.; Shi, Ke; Aihara, Hideki; Brown, William L.; Harris, Reuben S. 分享 收藏
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Oleic acid is an endogenous ligand of TLX/NR2E1 that triggers hippocampal neurogenesis 油酸是触发海马神经发生的TLX/NR2E1的内源性配体 Kandel, Prasanna; Semerci, Fatih; Mishra, Rachana; Choi, William; Bajic, Aleksandar; Baluya, Dodge; Ma, LiHua; Chen, Kevin; Cao, Austin C.; Phongmekhin, Tipwarin; Matinyan, Nick; Jimenez-Panizo, Alba; Chamakuri, Srinivas; Raji, Idris O.; Chang, Lyra; Fuentes-Prior, Pablo; MacKenzie, Kevin R.; Benn, Caroline L.; Estebanez-Perpina, Eva; Venken, Koen; Moore, David D.; Young, Damian W.; Maletic-Savatic, Mirjana 分享 收藏
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DNA-encoded chemistry technology yields expedient access to SARS-CoV-2 Mpro inhibitors Chamakuri, Srinivas; Lu, Shuo; Ucisik, Melek Nihan; Bohren, Kurt M.; Chen, Ying-Chu; Du, Huang-Chi; Faver, John C.; Jimmidi, Ravikumar; Li, Feng; Li, Jian-Yuan; Nyshadham, Pranavanand; Palmer, Stephen S.; Pollet, Jeroen; Qin, Xuan; Ronca, Shannon E.; Sankaran, Banumathi; Sharma, Kiran L.; Tan, Zhi; Versteeg, Leroy; Yu, Zhifeng; Matzuk, Martin M.; Palzkill, Timothy; Young, Damian W. 分享 收藏
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