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Applying molecular hybridization to design a new class of pyrazolo[3,4-d] pyrimidines as Src inhibitors active in hepatocellular carcinoma (vol 280, 116929, 2024) Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia 分享 收藏
Applying molecular hybridization to design a new class of pyrazolo[3,4-d] pyrimidines as Src inhibitors active in hepatocellular carcinoma Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia 分享 收藏
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4-Trifluoromethyl bithiazoles as broad-spectrum antimicrobial agents for virus-related bacterial infections or co-infections Barbieri, Francesca; Carlen, Vincent; Martina, Maria Grazia; Sannio, Filomena; Cancade, Sacha; Perini, Cecilia; Restori, Margherita; Crespan, Emmanuele; Maga, Giovanni; Docquier, Jean-Denis; Cagno, Valeria; Radi, Marco 分享 收藏
Normal and pathogenic variation of RFC1 repeat expansions: implications for clinical diagnosis RFC1重复扩增的正常和致病性变异: 对临床诊断的意义 Dominik, Natalia; Magri, Stefania; Curro, Riccardo; Abati, Elena; Facchini, Stefano; Corbetta, Marinella; Macpherson, Hannah; Di Bella, Daniela; Sarto, Elisa; Stevanovski, Igor; Chintalaphani, Sanjog R.; Akcimen, Fulya; Manini, Arianna; Vegezzi, Elisa; Quartesan, Ilaria; Montgomery, Kylie-Ann; Pirota, Valentina; Crespan, Emmanuele; Perini, Cecilia; Grupelli, Glenda Paola; Tomaselli, Pedro J.; Marques, Wilson; Shaw, Joseph; Polke, James; Salsano, Ettore; Fenu, Silvia; Pareyson, Davide; Pisciotta, Chiara; Tofaris, George K.; Nemeth, Andrea H.; Ealing, John; Radunovic, Aleksandar; Kearney, Seamus; Kumar, Kishore R.; Vucic, Steve; Kennerson, Marina; Reilly, Mary M.; Houlden, Henry; Deveson, Ira; Tucci, Arianna; Taroni, Franco; Cortese, Andrea 分享 收藏
Identification and Biological Characterization of the Pyrazolo[3,4-d]pyrimidine Derivative SI388 Active as Src Inhibitor Contadini, Claudia; Cirotti, Claudia; Carbone, Anna; Norouzi, Mehrdad; Cianciusi, Annarita; Crespan, Emmanuele; Perini, Cecilia; Maga, Giovanni; Barila, Daniela; Musumeci, Francesca; Schenone, Silvia 分享 收藏
Truncating Variants in RFC1 in Cerebellar Ataxia, Neuropathy, and Vestibular Areflexia Syndrome Ronco, Riccardo; Perini, Cecilia; Curro, Riccardo; Dominik, Natalia; Facchini, Stefano; Gennari, Alice; Simone, Roberto; Stuart, Skye; Nagy, Sara; Vegezzi, Elisa; Quartesan, Ilaria; El-Saddig, Amar; Lavin, Timothy; Tucci, Arianna; Szymura, Agnieszka; Novis De Farias, Luiz Eduardo; Gary, Alexander; Delfeld, Megan; Kandikatla, Priscilla; Niu, Nifang; Tawde, Sanjukta; Shaw, Joseph; Polke, James; Reilly, Mary M.; Wood, Nick W.; Crespan, Emmanuele; Gomez, Christopher; Chen, Jin Yun Helen; Schmahmann, Jeremy Dan; Gosal, David; Houlden, Henry; Das, Soma; Cortese, Andrea 分享 收藏
Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against Glioblastoma Multiforme Poggialini, Federica; Vagaggini, Chiara; Brai, Annalaura; Pasqualini, Claudia; Crespan, Emmanuele; Maga, Giovanni; Perini, Cecilia; Cabella, Noemi; Botta, Lorenzo; Musumeci, Francesca; Frosini, Maria; Schenone, Silvia; Dreassi, Elena 分享 收藏
Synthesis and biological activity evaluation of 3-(hetero) arylideneindolin-2-ones as potential c-Src inhibitors Princiotto, Salvatore; Musso, Loana; Manetti, Fabrizio; Marcellini, Valentina; Maga, Giovanni; Crespan, Emmanuele; Perini, Cecilia; Zaffaroni, Nadia; Beretta, Giovanni Luca; Dallavalle, Sabrina 分享 收藏
Towards Innovative Antibacterial Correctors for Cystic Fibrosis Targeting the Lung Microbiome with a Multifunctional Effect Martina, Maria Grazia; Sannio, Filomena; Crespan, Emmanuele; Pavone, Marialaura; Simoncini, Alice; Barbieri, Francesca; Perini, Cecilia; Pesce, Emanuela; Maga, Giovanni; Pedemonte, Nicoletta; Docquier, Jean-Denis; Radi, Marco 分享 收藏
System-oriented optimization of multi-target 2,6-diaminopurine derivatives: Easily accessible broad-spectrum antivirals active against flaviviruses, influenza virus and SARS-CoV-2 多目标2,6-二氨基嘌呤衍生物的系统导向优化: 易于获得的对黄病毒,流感病毒和SARS-CoV-2具有活性的广谱抗病毒药物 Vicenti, Ilaria; Martina, Maria Grazia; Boccuto, Adele; De Angelis, Marta; Giavarini, Giorgia; Dragoni, Filippo; Marchi, Serena; Trombetta, Claudia Maria; Crespan, Emmanuele; Maga, Giovanni; Eydoux, Cecilia; Decroly, Etienne; Montomoli, Emanuele; Nencioni, Lucia; Zazzi, Maurizio; Radi, Marco 分享 收藏
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses 磷脂酰肌醇4-激酶 (PI4KIIIβ) 的双噻唑抑制剂作为广谱抗病毒药物阻断SARS-CoV-2,寨卡病毒和人类鼻病毒的复制 Grazia Martina, Maria; Vicenti, Ilaria; Bauer, Lisa; Crespan, Emmanuele; Rango, Enrico; Boccuto, Adele; Olivieri, Noemi; Incerti, Matteo; Zwaagstra, Marleen; Allodi, Marika; Bertoni, Simona; Dreassi, Elena; Zazzi, Maurizio; van Kuppeveld, Frank J. M.; Maga, Giovanni; Radi, Marco 分享 收藏
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New indolylarylsulfone non-nucleoside reverse transcriptase inhibitors show low nanomolar inhibition of single and double HIV-1 mutant strains Nalli, Marianna; Armijos Rivera, Jorge, I; Masci, Domiziana; Coluccia, Antonio; Badia, Roger; Riveira-Munoz, Eva; Brambilla, Alessandro; Cinquina, Elisabetta; Turriziani, Ombretta; Falasca, Francesca; Catalano, Myriam; Limatola, Cristina; Este, Jose A.; Maga, Giovanni; Silvestri, Romano; Crespan, Emmanuele; La Regina, Giuseppe 分享 收藏
Multitarget CFTR Modulators Endowed with Multiple Beneficial Side Effects for Cystic Fibrosis Patients: Toward a Simplified Therapeutic Approach Tassini, Sabrina; Langron, Emily; Delang, Leen; Mirabelli, Carmen; Lanko, Kristina; Crespan, Emmanuele; Kissova, Miroslava; Tagliavini, Giulia; Fonto, Greta; Bertoni, Simona; Palese, Simone; Giorgio, Carmine; Ravanetti, Francesca; Ragionieri, Luisa; Zamperini, Claudio; Mancini, Arianna; Dreassi, Elena; Maga, Giovanni; Vergani, Paola; Neyts, Johan; Radi, Marco 分享 收藏