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A. Ganesan

liverpool john moores university

51H指数
250论文数
8.4K被引数
收录论文 86
发表时间
Tranylcypromine-Based LSD1 Inhibitors as Useful Agents to Reduce Viability of Schistosoma mansoni基于Tranylcypromine的LSD1抑制剂作为降低Schistosoma mansoni存活率的潜在有效药物
err2025-07-02
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errEmanuele Fabbrizi; Gebremedhin Solomon Hailu; A. Ganesan; Rossella Fioravanti; Clemens Zwergel; Chiara Lambona; Sergio Valente; Giulia Fianco; Angela Iuzzolino; Daniela Trisciuoglio; Jonatan Caroli; Andrea Mattevi; Cécile Häberli; Jennifer Keiser; Dante Rotili; Antonello Mai
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Design, Synthesis, and Biological Evaluation of Potent EZH2/LSD1 Dual Inhibitors for Prostate Cancer
err2024-08-28
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PREAI
errLe, Meiling; Lu, Wenhua; Tan, Xiaozhuo; Luo, Bingling; Yu, Tiantian; Sun, Yameng; Guo, Zhirong; Huang, Peng; Zhu, Daqian; Wu, Qiang; Ganesan, A.; Wen, Shijun
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Discovery of 1-Benzhydryl-Piperazine-Based HDAC Inhibitors with Anti-Breast Cancer Activity: Synthesis, Molecular Modeling, In Vitro and In Vivo Biological Evaluation
err2022-11-25
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errOAAI
errRuzic, Dusan; Ellinger, Bernhard; Djokovic, Nemanja; Santibanez, Juan F.; Gul, Sheraz; Beljkas, Milan; Djuric, Ana; Ganesan, Arasu; Pavic, Aleksandar; Srdic-Rajic, Tatjana; Petkovic, Milos; Nikolic, Katarina
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Synthesis of Carboxamide-Containing Tranylcypromine Analogues as LSD1 (KDM1A) Inhibitors Targeting Acute Myeloid Leukemia
err2021-02-03
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errTeresa Borrello, Maria; Benelkebir, Hanae; Lee, Adam; Hin Tam, Chak; Shafat, Manar; Rushworth, Stuart A.; Bowles, Kristian M.; Douglas, Leon; Duriez, Patrick J.; Bailey, Sarah; Crabb, Simon J.; Packham, Graham; Ganesan, A.
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Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in Schistosoma mansoni
err2020-07-01
err6
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errCarneiro, Vitor Coutinho; de Abreu Silva, Isabel Caetano; Amaral, Murilo Sena; Pereira, Adriana S. A.; Silveira, Gilbert Oliveira; Pires, David da Silva; Verjovski-Almeida, Sergio; Dekker, Frank J.; Rotili, Dante; Mai, Antonello; Lopes-Torres, Eduardo Jose; Robaa, Dina; Sippl, Wolfgang; Pierce, Raymond J.; Borrello, M. Teresa; Ganesan, A.; Lancelot, Julien; Thiengo, Silvana; Fernandez, Monica Ammon; Revoredo Vicentino, Amanda Roberta; Mourao, Marina Moraes; Coelho, Fernanda Sales; Fantappie, Marcelo Rosado
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A Decade of Antifungal Leads from Natural Products: 2010-2019
err2019-12-12
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errOAAI
errAldholmi, Mohammed; Marchand, Pascal; Ourliac-Garnier, Isabelle; Le Pape, Patrice; Ganesan, A.
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The timeline of epigenetic drug discovery: from reality to dreams
err2019-12-02
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errGanesan, A.; Arimondo, Paola B.; Rots, Marianne G.; Jeronimo, Carmen; Berdasco, Maria
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β-amino alcohols and their respective 2-phenyl-N-alkyl aziridines as potential DNA minor groove binders
err2018-09-01
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errVaidergorn, Miguel M.; Carneiro, Zumira A.; Lopes, Carla D.; de Albuquerque, Sergio; Reis, Felipe C. C.; Nikolaou, Sofia; e Mello, Juliana F. R.; Genesi, Giovani L.; Trossini, Gustavo H. G.; Ganesan, A.; Emery, Flavio S.
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LSD1 inhibition attenuates androgen receptor V7 splice variant activation in castration resistant prostate cancer models
err2018-05-09
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errda Mota, Sergio Regufe; Bailey, Sarah; Strivens, Rosemary A.; Hayden, Annette L.; Douglas, Leon R.; Duriez, Patrick J.; Borrello, M. Teresa; Benelkebir, Hanae; Ganesan, A.; Packham, Graham; Crabb, Simon J.
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