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Design and Discovery of Substituted 1,3,4-Thiadiazole-1,3,5-Triazine Hybrids as Human Immunodeficiency Virus-1 Non-Nucleoside Reverse Transcriptase Inhibitors with Anti-SARS-CoV-2 and Antibacterial Activities 设计并发现取代的1,3,4-噻二唑-1,3,5-三嗪杂合物作为具有抗SARS-CoV-2和抗菌活性的人类免疫缺陷病毒-1非核苷类反转录酶抑制剂 Singh, Saumya; Srivastava, Kumar Saurabh; Kumawat, Mukesh Kumar; Bhat, Hans Raj; Corona, Angela; Tramontano, Enzo; Mitra, Debashis; Singh, Udaya Pratap 分享 收藏
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Design, Synthesis and Biological Evaluation of 3-Hydrazonoindolin-2-one Derivatives as Novel HIV-1 RNase H Inhibitors 3-肼基酮基吲哚啉-2-酮衍生物的设计、合成及生物评价:作为新型HIV-1 RNase H抑制剂的探索 Zhang, Yiying; Wang, Rao; Bu, Yueyue; Corona, Angela; Dettori, Laura; Tramontano, Enzo; Pannecouque, Christophe; De Clercq, Erik; Meng, Ge; Chen, Fen-Er 分享 收藏
Synthesis and Evaluation of Thiazolidinone-Isatin Hybrids for Selective Inhibition of Cancer-Related Carbonic Anhydrases Onali, Alessia; Sanna, Erica; Lupia, Antonio; Secci, Daniela; Atzeni, Giulia; Demuru, Laura; Angeli, Andrea; Cottiglia, Filippo; Meleddu, Rita; Emmolo, Roberta; Corona, Angela; Maccioni, Elias; Supuran, Claudiu T.; Distinto, Simona 分享 收藏
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Identification of HIV-1 Reverse Transcriptase-Associated Ribonuclease H Inhibitors Based on 2-Hydroxy-1,4-naphthoquinone Mannich Bases Tu, Nhat Quang; Richetta, Clemence; Putzu, Federica; Delelis, Olivier; Ahmed, Khursheed; Masand, Vijay H.; Schobert, Rainer; Tramontano, Enzo; Corona, Angela; Biersack, Bernhard 分享 收藏
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4-(3-Phenylsulfonylindol-2-yl)-1-(pyridin-2-yl)piperazinyl-methanones as Potent Inhibitors of both SARS-CoV-2 and HCoV-OC43 Viruses Puxeddu, Michela; Donalisio, Manuela; Bugert, Joachim Jakob; Corona, Angela; Cocomazzi, Paolo; Milani, Mario; Hucke, Friederike; Arduino, Irene; Esposito, Francesca; Moretti, Paolo; Ortore, Maria Grazia; Nalli, Marianna; Manetto, Simone; Mazzoccanti, Giulia; Bigogno, Chiara; Dondio, Giulio; Scio, Pietro; Coluccia, Antonio; Fracella, Matteo; Antonelli, Guido; Lembo, David; Tramontano, Enzo; Silvestri, Romano; Mastrangelo, Eloise; La Regina, Giuseppe 分享 收藏
New Thiazolidine-4-One Derivatives as SARS-CoV-2 Main Protease Inhibitors Messore, Antonella; Malune, Paolo; Patacchini, Elisa; Madia, Valentina Noemi; Ialongo, Davide; Arpacioglu, Merve; Albano, Aurora; Ruggieri, Giuseppe; Saccoliti, Francesco; Scipione, Luigi; Tramontano, Enzo; Canton, Serena; Corona, Angela; Scognamiglio, Sante; Paulis, Annalaura; Suleiman, Mustapha; Al-Maqtari, Helmi Mohammed; Abid, Fatma Mohamed A.; Kawsar, Sarkar M. A.; Sankaranarayanan, Murugesan; Di Santo, Roberto; Esposito, Francesca; Costi, Roberta 分享 收藏