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Michael J. Delves

imperial college london

37H指数
104论文数
5.5K被引数
收录论文 63
发表时间
Structure-Guided Optimization of Novel Inhibitors of Plasmodium Lysyl-tRNA Synthetase with Multistage Activity against Malaria Parasites基于结构的优化新型恶性疟原虫赖氨酰-tRNA合成酶抑制剂,其对疟疾寄生虫具有多阶段活性
err2026-06-02
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errBarbara Forte; Fiona Bellany; Peter S. Campbell; Giulia Chemi; Alice Dawson; Mark Anderson; Yaw Aniweh; Anna Y. Burkhard; Anna Caroline Campos Aguiar; Alisje Churchyard; Caitlin A. Cooper; Amália dos Santos Ferreira; Mufuliat Toyin Famodimu; Francis G. Fang; Xiao Hu; Tonnie Huijs; Delphine Baud; Chimed Jansen; María Belén Jiménez Díaz; Roger Bonnert; Susan Boyd; Benigno Crespo-Fernández; Branko Mitasev; Simone Montagna; Sachel Mok; Dinakaran Murugesan; Sunil K. Narwal; Neil R. Norcross; John Okombo; Heekuk Park; Caroline Peet; Dhelio B. Pereira; John M. Post; Janette Reader; Jennifer Riley; David A. Robinson; Raku Shinkyo; Frederick R.C. Simeons; Laura Simpson; Alasdair Smith; Dennis Smith; Josefine Striepen; Carolina B.G. Teles; Rianne van der Laak; Anne-Catrin Uhlemann; Amélie Vantaux; Caroline Wilson; Benoît Witkowski; Gavin Wood; Tomas Yeo; Fabio Zuccotto; Iñigo Angulo-Barturen; Jake Baum; Judith M. Bolscher; Rafael Victorio Carvalho Guido; Lyn-Marié Birkholtz; Michael J. Delves; Laurent Dembele; David A. Fidock; Francisco Javier Gamo; Dennis E. Kyle; Steven P. Maher; Jean Popovici; Chris Walpole; Fabian Gusovsky; Paul A. Willis; Kevin D. Read; Ian H. Gilbert; Beatriz Baragaña
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Targeting Aurora Kinases as Essential Cell-Cycle Regulators to Deliver Multi-Stage Antimalarials Against Plasmodium Falciparum靶向Aurora Kinases这一关键细胞周期调控因子,以递送针对Plasmodium Falciparum的多阶段抗疟药。
err2025-10-23
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errHenrico Langeveld; Keletso Maepa; Marché Maree; Jessica L. Thibaud; Nicolaas Salomane; Rosie Bridgwater; Mufuliat T. Famodimu; Luiz C. Godoy; Charisse Flerida A. Pasaje; Nonlawat Boonyalai; Mariana Laureano de Souza; Justin Fong; Tayla Rabie; Mariëtte van der Watt; Rensu P. Theart; Sonja Ghidelli-Disse; Jacquin C. Niles; Marcus C. S. Lee; Elizabeth A. Winzeler; Michael J. Delves; Kelly Chibale; Kathryn J. Wicht; Lauren B. Coulson; Lyn-Marié Birkholtz
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Optimization and Characterization of the Antimalarial Activity of N-Aryl Acetamides that are Susceptible to Mutations in ROM8 and CSC1ROM8和CSC1易受突变影响的N-芳基乙酰胺类化合物的抗疟活性的优化与表征
err2025-07-18
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errWilliam Nguyen; Coralie Boulet; Madeline G. Dans; Katie Loi; Kate E. Jarman; Claudia B. G. Barnes; Tomas Yeo; Tanaya Sheth; Partha Mukherjee; Arnish Chakraborty; Mufuliat T. Famodimu; Michael J. Delves; Harry Pollard; Colin J. Sutherland; Rachael Coyle; Nicole Sevilleno; Nonlawat Boonyalai; Marcus C. S. Lee; Tayla Rabie; Lyn-Marié Birkholtz; Delphine Baud; Stephen Brand; Mrittika Chowdury; Tania F. de Koning-Ward; David A. Fidock; Paul R. Gilson; Brad E. Sleebs
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Optimization and Characterization of N-Acetamide Indoles as Antimalarials That Target PfATP4N-乙酰胺基吲哚类化合物的优化与表征:靶向PfATP4的抗疟疾药物研究
err2025-04-14
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PREAI
errAwalt, Jon Kyle; Ooi, Zi Kang; Ashton, Trent D.; Mansouri, Mahta; Calic, Petar P. S.; Zhou, Qingmiao; Vasanthan, Santhya; Lee, Serena; Loi, Katie; Jarman, Kate E.; Penington, Jocelyn S.; Qiu, Deyun; Zhang, Xinxin; Lehane, Adele M.; Mao, Emma Y.; Gancheva, Maria R.; Wilson, Danny W.; Giannangelo, Carlo; MacRaild, Christopher A.; Creek, Darren J.; Yeo, Tomas; Sheth, Tanaya; Fidock, David A.; Churchyard, Alisje; Baum, Jake; Famodimu, Mufuliat T.; Delves, Michael J.; Kristan, Mojca; Stewart, Lindsay; Sutherland, Colin J.; Coyle, Rachael; Jagoe, Hannah; Lee, Marcus C. S.; Chowdury, Mrittika; de Koning-Ward, Tania F.; Baud, Delphine; Brand, Stephen; Jackson, Paul F.; Cowman, Alan F.; Dans, Madeline G.; Sleebs, Brad E.
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A potent and selective reaction hijacking inhibitor of Plasmodium falciparum tyrosine tRNA synthetase exhibits single dose oral efficacy in vivo
err2024-12-09
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errXie, Stanley C.; Tai, Chia-Wei; Morton, Craig J.; Ma, Liting; Huang, Shih-Chung; Wittlin, Sergio; Du, Yawei; Hu, Yongbo; Dogovski, Con; Salimimarand, Mina; Griffin, Robert; England, Dylan; de la Cruz, Elisa; Deni, Ioanna; Yeo, Tomas; Burkhard, Anna Y.; Striepen, Josefine; Schindler, Kyra A.; Crespo, Benigno; Gamo, Francisco J.; Khandokar, Yogesh; Hutton, Craig A.; Rabie, Tayla; Birkholtz, Lyn-Marie; Famodimu, Mufuliat T.; Delves, Michael J.; Bolsher, Judith; Koolen, Karin M. J.; van der Laak, Rianne; Aguiar, Anna C. C.; Pereira, Dhelio B.; Guido, Rafael V. C.; Creek, Darren J.; Fidock, David A.; Dick, Lawrence R.; Brand, Stephen L.; Gould, Alexandra E.; Langston, Steven; Griffin, Michael D. W.; Tilley, Leann
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Exploration and characterization of the antimalarial activity of cyclopropyl carboxamides that target the mitochondrial protein, cytochrome b针对线粒体蛋白,细胞色素b的环丙基甲酰胺的抗疟活性的探索和表征
err2024-12-01
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errAwalt, Jon Kyle; Su, Wenyin; Nguyen, William; Loi, Katie; Jarman, Kate E.; Penington, Jocelyn S.; Ramesh, Saishyam; Fairhurst, Kate J.; Yeo, Tomas; Park, Heekuk; Uhlemann, Anne-Catrin; Maity, Bikash Chandra; De, Nirupam; Mukherjee, Partha; Chakraborty, Arnish; Churchyard, Alisje; Famodimu, Mufuliat T.; Delves, Michael J.; Baum, Jake; Mittal, Nimisha; Winzeler, Elizabeth A.; Papenfuss, Anthony T.; Chowdury, Mrittika; de Koning-Ward, Tania F.; Maier, Alexander G.; van Dooren, Giel G.; Baud, Delphine; Brand, Stephen; Fidock, David A.; Jackson, Paul F.; Cowman, Alan F.; Dans, Madeline G.; Sleebs, Brad E.
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Mitochondrial ATP synthesis is essential for efficient gametogenesis in Plasmodium falciparum
err2024-11-16
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errSparkes, Penny C.; Famodimu, Mufuliat Toyin; Alves, Eduardo; Springer, Eric; Przyborski, Jude; Delves, Michael J.
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Tambjamines as Fast-Acting Multistage Antimalarials
err2024-11-11
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PREAI
errKumar, Amrendra; Li, Yuexin; Dodean, Rozalia A.; Roth, Alison; Caridha, Diana; Madejczyk, Michael S.; Jin, Xiannu; Dennis, William E.; Lee, Patricia J.; Pybus, Brandon S.; Martin, Monica; Pannone, Kristina; Dinh, Hieu T.; Blount, Cameron; Chetree, Ravi; Deluca, Jesse; Evans, Martin; Nadeau, Robert; Vuong, Chau; Leed, Susan; Black, Chad; Sousa, Jason; Nolan, Christina; Ceja, Frida G.; Rasmussen, Stephanie A.; Tumwebaze, Patrick K.; Rosenthal, Philip J.; Cooper, Roland A.; Rottmann, Matthias; Orjuela-Sanchez, Pamela; Meister, Stephan; Winzeler, Elizabeth A.; Delves, Michael J.; Matthews, Holly; Baum, Jake; Kirby, Robert W.; Burrows, Jeremy N.; Duffy, James; Peyton, David H.; Reynolds, Kevin A.; Kelly, Jane X.; Kancharla, Papireddy
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Lactam Truncation Yields a Dihydroquinazolinone Scaffold with Potent Antimalarial Activity that Targets PfATP4内酰胺截短产生具有针对PfATP4的有效抗疟活性的二氢喹唑啉酮支架
err2024-10-29
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PREAI
errAshton, Trent D.; Calic, Petar P. S.; Dans, Madeline G.; Ooi, Zi Kang; Zhou, Qingmiao; Loi, Katie; Jarman, Kate E.; Palandri, Josephine; Qiu, Deyun; Lehane, Adele M.; Maity, Bikash; De, Nirupam; Famodimu, Mufuliat T.; Delves, Michael J.; Mao, Emma Y.; Gancheva, Maria R.; Wilson, Danny W.; Chowdury, Mrittika; de Koning-Ward, Tania F.; Baud, Delphine; Brand, Stephen; Jackson, Paul F.; Cowman, Alan F.; Sleebs, Brad E.
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Aryl amino acetamides prevent Plasmodium falciparum ring development via targeting the lipid-transfer protein PfSTART1 (vol 15, 5219, 2024)芳基氨基乙酰胺通过靶向脂质转移蛋白PfSTART1 (vol 15,5219,2024) 防止恶性疟原虫环发育
err2024-09-30
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errDans, Madeline G.; Boulet, Coralie; Watson, Gabrielle M.; Nguyen, William; Dziekan, Jerzy M.; Evelyn, Cindy; Reaksudsan, Kitsanapong; Mehra, Somya; Razook, Zahra; Geoghegan, Niall D.; Mlodzianoski, Michael J.; Goodman, Christopher Dean; Ling, Dawson B.; Jonsdottir, Thorey K.; Tong, Joshua; Famodimu, Mufuliat Toyin; Kristan, Mojca; Pollard, Harry; Stewart, Lindsay B.; Brandner-Garrod, Luke; Sutherland, Colin J.; Delves, Michael J.; Mcfadden, Geoffrey I.; Barry, Alyssa E.; Crabb, Brendan S.; de Koning-Ward, Tania F.; Rogers, Kelly L.; Cowman, Alan F.; Tham, Wai-Hong; Sleebs, Brad E.; Gilson, Paul R.
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A Pan Plasmodium lateral flow recombinase polymerase amplification assay for monitoring malaria parasites in vectors and human populations
err2024-08-30
err1
errOAAI
errHiggins, Matthew; Kristan, Mojca; Collins, Emma L.; Messenger, Louisa A.; Dombrowski, Jamille G.; Vanheer, Leen N.; Nolder, Debbie; Drakeley, Christopher J.; Stone, William; Mahamar, Almahamoudou; Bousema, Teun; Delves, Michael; Bandibabone, Janvier; N'Do, Severin; Bantuzeko, Chimanuka; Zawadi, Bertin; Walker, Thomas; Sutherland, Colin J.; Marinho, Claudio R. F.; Cameron, Mary M.; Clark, Taane G.; Campino, Susana
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Property and Activity Refinement of Dihydroquinazolinone-3-carboxamides as Orally Efficacious Antimalarials that Target PfATP4Dihydroquinazolinone-3-carboxamides作为靶向PfATP4的口服有效抗疟药的性质和活性精制
err2024-08-12
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errAshton, Trent D.; Calic, Petar P. S.; Dans, Madeline G.; Ooi, Zi Kang; Zhou, Qingmiao; Palandri, Josephine; Loi, Katie; Jarman, Kate E.; Qiu, Deyun; Lehane, Adele M.; Maity, Bikash Chandra; De, Nirupam; Giannangelo, Carlo; Macraild, Christopher A.; Creek, Darren J.; Mao, Emma Y.; Gancheva, Maria R.; Wilson, Danny W.; Chowdury, Mrittika; de Koning-Ward, Tania F.; Famodimu, Mufuliat T.; Delves, Michael J.; Pollard, Harry; Sutherland, Colin J.; Baud, Delphine; Brand, Stephen; Jackson, Paul F.; Cowman, Alan F.; Sleebs, Brad E.
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Aryl amino acetamides prevent Plasmodium falciparum ring development via targeting the lipid-transfer protein PfSTART1芳基氨基乙酰胺通过靶向脂质转移蛋白PfSTART1阻止恶性疟原虫环的发展
err2024-06-18
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errDans, Madeline G.; Boulet, Coralie; Watson, Gabrielle M.; Nguyen, William; Dziekan, Jerzy M.; Evelyn, Cindy; Reaksudsan, Kitsanapong; Mehra, Somya; Razook, Zahra; Geoghegan, Niall D.; Mlodzianoski, Michael J.; Goodman, Christopher Dean; Ling, Dawson B.; Jonsdottir, Thorey K.; Tong, Joshua; Famodimu, Mufuliat Toyin; Kristan, Mojca; Pollard, Harry; Stewart, Lindsay B.; Brandner-Garrod, Luke; Sutherland, Colin J.; Delves, Michael J.; Mcfadden, Geoffrey I.; Barry, Alyssa E.; Crabb, Brendan S.; de Koning-Ward, Tania F.; Rogers, Kelly L.; Cowman, Alan F.; Tham, Wai-Hong; Sleebs, Brad E.; Gilson, Paul R.
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Optimisation-based modelling for explainable lead discovery in malaria
err2024-01-01
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errLi, Yutong; Cardoso-Silva, Jonathan; Kelly, John M.; Delves, Michael J.; Furnham, Nicholas; Papageorgiou, Lazaros G.; Tsoka, Sophia
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Machine learning-based phenotypic imaging to characterise the targetable biology of Plasmodium falciparum male gametocytes for the development of transmission-blocking antimalarials
err2023-10-06
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errTsebriy, Oleksiy; Khomiak, Andrii; Miguel-Blanco, Celia; Sparkes, Penny C.; Gioli, Maurizio; Santelli, Marco; Whitley, Edgar; Gamo, Francisco-Javier; Delves, Michael J.
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Bis-6-amidino-benzothiazole Derivative that Cures Experimental Stage 1 African Trypanosomiasis with a Single Dose
err2023-09-18
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errRacane, Livio; Pticek, Lucija; Kostrun, Sanja; Raic-Malic, Silvana; Taylor, Martin Craig; Delves, Michael; Alsford, Sam; Olmo, Francisco; Francisco, Amanda Fortes; Kelly, John M.
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A Pyridyl-Furan Series Developed from the Open Global Health Library Block Red Blood Cell Invasion and Protein Trafficking in Plasmodium falciparum through Potential Inhibition of the Parasite's PI4KIIIB Enzyme
err2023-08-28
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errLing, Dawson B.; Nguyen, William; Looker, Oliver; Razook, Zahra; Mccann, Kirsty; Barry, Alyssa E.; Scheurer, Christian; Wittlin, Sergio; Famodimu, Mufuliat Toyin; Delves, Michael J.; Bullen, Hayley E.; Crabb, Brendan S.; Sleebs, Brad E.; Gilson, Paul R.
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A novel class of sulphonamides potently block malaria transmission by targeting a Plasmodium vacuole membrane protein
err2023-01-30
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errYahiya, Sabrina; Saunders, Charlie N.; Hassan, Sarah; Straschil, Ursula; Fischer, Oliver J.; Rueda-Zubiaurre, Ainoa; Haase, Silvia; Vizcay-Barrena, Gema; Famodimu, Mufuliat Toyin; Jordan, Sarah; Delves, Michael J.; Tate, Edward W.; Barnard, Anna; Fuchter, Matthew J.; Baum, Jake
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Protocols for Plasmodium gametocyte production in vitro: an integrative review and analysis
err2022-12-05
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errOmorou, Roukayatou; Bin Sa'id, Ibrahim; Delves, Michael; Severini, Carlo; Kouakou, Yobouet Ines; Bienvenu, Anne-Lise; Picot, Stephane
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