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Helena I. Boshoff

national institutes of health (nih)

65H指数
266论文数
1.6W被引数
收录论文 136
发表时间
Synthesis of 4-Aminoindole-Containing Cephalosporin Prodrugs and Their Biological Activity against Mycobacterium tuberculosis含4-氨基吲哚基头孢菌素前药的合成及其对结核分枝杆菌的生物活性
err2026-06-09
err0
errOAAI
errSangmi Oh; Helena I. M. Boshoff; Jose Santinni O. Roma; Aidan Boving; Danielle M. Weiner; April Walker; Laura E. Via; Clifton E. Barry III
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PET/CT imaging of tuberculosis lung lesions in marmosets treated with different drug regimens aligns with human clinical outcomes不同药物治疗方案下卷尾猴结核肺病变的PET/CT成像结果与人类临床结局一致
err2026-01-07
err0
PREAI
errTalia Greenstein; Laura E. Via; Mariana Pereira Moraes; Danielle M. Weiner; Emmanuel K. Dayao; April M. Walker; Ayan Abdi; Joel D. Fleegle; Felipe Gomez; Katelyn M. Repoli; Michael J. Woodcock; Helena I. M. Boshoff; Oluwaseun Egbelowo; Kamunkhwala Gausi; Paolo Denti; Firat Kaya; Matthew Zimmerman; Eric L. Miller; Véronique A. Dartois; Clifton E. Barry; Bree B. Aldridge
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Structure-activity relationship study of a new class of 2-amino-3,4-dihydroquinazolines as antitubercular agents
err2026-01-05
err0
errOAAI
errLena Trifonov; Helena I. Boshoff; Jose Santinni O. Roma; Yixuan Fan; He Eun Forbes; Clifton E. Barry; Sangmi Oh
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SuFEx-based antitubercular compound irreversibly inhibits Pks13基于SuFEx的抗结核化合物不可逆地抑制Pks13
errNature
IF48.5
err2025-07-30
err0
PREAI
errInna V. Krieger; Paridhi Sukheja; Baiyuan Yang; Su Tang; Daniel Selle; Ashley Woods; Curtis Engelhart; Pradeep Kumar; Michael B. Harbut; Dongdong Liu; Brendan Tsuda; Bo Qin; Grant A. L. Bare; Gencheng Li; Victor Chi; Julian Gambacurta; Janine Hvizdos; Matthew Reagan; Isabelle L. Jones; Lisa M. Massoudi; Lisa K. Woolhiser; Alessandro Cascioferro; Erica Kundrick; Parul Singh; William Reiley; Thomas R. Ioerger; Dilipkumar Reddy Kandula; Jacob W. McCabe; Taijie Guo; David Alland; Helena I. Boshoff; Dirk Schnappinger; Gregory T. Robertson; Khisi Mdluli; Kyoung-Jin Lee; Jiajia Dong; Shuangwei Li; Peter G. Schultz; Sean B. Joseph; Melissa S. Love; K. Barry Sharpless; H. Michael Petrassi; Arnab K. Chatterjee; James C. Sacchettini; Case W. McNamara
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Fragment-Based Development of Small Molecule Inhibitors Targeting Mycobacterium tuberculosis Cholesterol Metabolism基于片段的针对分枝杆菌胆固醇代谢的小分子抑制剂开发
err2025-07-14
err0
errOAAI
errMadeline E. Kavanagh; Kirsty J. McLean; Sophie H. Gilbert; Cecilia N. Amadi; Matthew Snee; Richard B. Tunnicliffe; Kriti Arora; Helena I. M. Boshoff; Alexander Fanourakis; Maria Jose Rebollo-Lopez; Fatima Ortega; Colin W. Levy; Andrew W. Munro; David Leys; Chris Abell; Anthony G. Coyne
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Thioquinazolinones as Antituberculosis Agents Targeting Phosphopantetheinyl Transferase噻唑并[3,2-a]喹唑啉酮类化合物作为靶向磷脂泛酰巯基乙胺转移酶的抗结核药物
err2025-07-01
err0
PREAI
errAmrita Singh; Logan T. Zwerneman; Kyle Planck; Takushi Kaneko; Andrew J. Perkowski; Christine M. Suh; Alexander Alex; James Bean; Kristin Burns-Huang; David Zhang; Helena I. M. Boshoff; Christine Roubert; Inna Krieger; Mark Gardner; Bastien Cautain; Christopher B. Cooper; Zaid Tanvir; James Sacchettini; Ben S. Gold; Kyu Y. Rhee; Nader Fotouhi; Carl F. Nathan; Jeffrey Aubé
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Sanfetrinem, an oral (3-lactam antibiotic repurposed for the treatment of tuberculosisSanfetrinem,一种用于治疗结核病的口服β-内酰胺类抗生素。
err2025-05-01
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errOAAI
errRamon-Garcia, Santiago; del Rio, Ruben Gonzalez; Arenaz-Callao, Maria Pilar; Boshoff, Helena I.; Rullas, Joaquin; Anca, Sara; Izquierdo, Monica Cacho; de Francisco, Esther Porras; Herran, Esther Perez; Santos-Villarejo, Angel; Mendoza-Losana, Alfonso; Ferrer-Bazaga, Santiago; Thompson, Charles J.; Aguirre, David Barros; Bates, Robert H.
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Developing novel indoles as antitubercular agents and simulated annealing-based analysis of their binding with MmpL3
err2024-12-25
err0
PREAI
errRay, Rajdeep; Das, Stutee; Birangal, Sumit Raosaheb; Boshoff, Helena I.; Roma, Jose Santinni; Lobo, Manisha; Hariharapura, Raghu Chandrashekhar; Shenoy, G. Gautham
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Mtb-Selective 5-Aminomethyl Oxazolidinone Prodrugs: Robust Potency and Potential Liabilities
err2024-04-06
err2
PREAI
errBoshoff, Helena I. M.; Young, Katherine; Ahn, Yong-Mo; Yadav, Veena D.; Crowley, Brendan M.; Yang, Lihu; Su, Jing; Oh, Sangmi; Arora, Kriti; Andrews, Jenna; Manikkam, Michelle; Sutphin, Michelle; Smith, Anthony J.; Weiner, Danielle M.; Piazza, Michaela K.; Fleegle, Joel D.; Gomez, Felipe; Dayao, Emmannual K.; Prideaux, Brendan; Zimmerman, Matthew; Kaya, Firat; Sarathy, Jansy; Tan, Vee Yang; Via, Laura E.; Tschirret-Guth, Richard; Lenaerts, Anne J.; Robertson, Gregory T.; Dartois, Veronique; Olsen, David B.; Barry III, Clifton E.
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The Antitubercular Activities of Natural Products with Fused-Nitrogen-Containing Heterocycles
err2024-02-06
err3
errOAAI
errBoshoff, Helena I.; Malhotra, Neha; Barry III, Clifton E.; Oh, Sangmi
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Inhibition of DXR in the MEP pathway with lipophilic N-alkoxyaryl FR900098 analogs
err2024-01-01
err2
errOAAI
errBague, Darean; Wang, Ruiqin; Hodge, Dana; Mikati, Marwa O.; Roma, Jose S.; Boshoff, Helena I.; Dailey, Allyson L.; Girma, Misgina; Couch, Robin D.; Odom John, Audrey R.; Dowd, Cynthia S.
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Identification and Optimization of Novel Inhibitors of the Polyketide Synthase 13 Thioesterase Domain with Antitubercular Activity
err2023-11-10
err4
errOAAI
errGreen, Simon R.; Wilson, Caroline; Eadsforth, Thomas C.; Punekar, Avinash S.; Tamaki, Fabio K.; Wood, Gavin; Caldwell, Nicola; Forte, Barbara; Norcross, Neil R.; Kiczun, Michael; Post, John M.; Lopez-Roman, Eva Maria; Engelhart, Curtis A.; Lukac, Iva; Zuccotto, Fabio; Epemolu, Ola; Boshoff, Helena I. M.; Schnappinger, Dirk; Walpole, Chris; Gilbert, Ian H.; Read, Kevin D.; Wyatt, Paul G.; Baragana, Beatriz
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Synthesis and Structure-Activity Relationships of a New Class of Oxadiazoles Targeting DprE1 as Antitubercular Agents靶向DprE1的新型恶二唑类抗结核药的合成和构效关系
err2023-08-15
err2
errOAAI
errYadav, Veena D. D.; Boshoff, Helena I. I.; Trifonov, Lena; Roma, Jose Santinni O.; Ioerger, Thomas R. R.; Barry, Clifton E. E.; Oh, Sangmi
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MEPicides: α,β-unsaturated Fosmidomycin N-Acyl Analogs as Efficient Inhibitors of Plasmodium falciparum 1-Deoxy-d-xylulose-5-phosphate reductoisomerase
err2023-06-13
err5
PREAI
errWang, Xu; Edwards, Rachel L.; Ball, Haley S.; Heidel, Kenneth M.; Brothers, Robert C.; Johnson, Claire; Haymond, Amanda; Girma, Misgina; Dailey, Allyson; Roma, Jose Santinni; Boshoff, Helena I.; Osbourn, Damon M.; Meyers, Marvin J.; Couch, Robin D.; Odom John, Audrey R.; Dowd, Cynthia S.
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Chemical approaches to unraveling the biology of mycobacteria
err2023-05-01
err0
errOAAI
errFinin, Peter; Khan, R. M. Naseer; Oh, Sangmi; Boshoff, Helena I. M.; Barry, Clifton E.
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Structure Based Discovery of Inhibitors of CYP125 and CYP142 from Mycobacterium tuberculosis
err2023-04-12
err4
errOAAI
errKatariya, Mona M.; Snee, Matthew; Tunnicliffe, Richard B.; Kavanagh, Madeline E.; Boshoff, Helena I. M.; Amadi, Cecilia N.; Levy, Colin W.; Munro, Andrew W.; Abell, Chris; Leys, David; Coyne, Anthony G.; McLean, Kirsty J.
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The Myxobacterial Antibiotic Myxovalargin: Biosynthesis, Structural Revision, Total Synthesis, and Molecular Characterization of Ribosomal Inhibition
err2023-01-05
err5
errOAAI
errKoller, Timm O.; Scheid, Ullrich; Koesel, Teresa; Herrmann, Jennifer; Krug, Daniel; Boshoff, Helena I. M.; Beckert, Bertrand; Evans, Joanna C.; Schlemmer, Jan; Sloan, Becky; Weiner, Danielle M.; Via, Laura E.; Moosa, Atica; Ioerger, Thomas R.; Graf, Michael; Zinshteyn, Boris; Abdelshahid, Maha; Nguyen, Fabian; Arenz, Stefan; Gille, Franziska; Siebke, Maik; Seedorf, Tim; Plettenburg, Oliver; Green, Rachel; Warnke, Anna-Luisa; Ullrich, Joachim; Warrass, Ralf; Barry, Clifton E., III; Warner, Digby F.; Mizrahi, Valerie; Kirschning, Andreas; Wilson, Daniel N.; Mueller, Rolf
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Lysyl-tRNA synthetase, a target for urgently needed M. tuberculosis drugs
err2022-10-11
err13
errOAAI
errGreen, Simon R.; Davis, Susan H.; Damerow, Sebastian; Engelhart, Curtis A.; Mathieson, Michael; Baragana, Beatriz; Robinson, David A.; Tamjar, Jevgenia; Dawson, Alice; Tamaki, Fabio K.; Buchanan, Kirsteen, I; Post, John; Dowers, Karen; Shepherd, Sharon M.; Jansen, Chimed; Zuccotto, Fabio; Gilbert, Ian H.; Epemolu, Ola; Riley, Jennifer; Stojanovski, Laste; Osuna-Cabello, Maria; Perez-Herran, Esther; Rebollo, Maria Jose; Lopez, Laura Guijarro; Castro, Patricia Casado; Camino, Isabel; Kim, Heather C.; Bean, James M.; Nahiyaan, Navid; Rhee, Kyu Y.; Wang, Qinglan; Tan, Vee Y.; Boshoff, Helena I. M.; Converse, Paul J.; Li, Si-Yang; Chang, Yong S.; Fotouhi, Nader; Upton, Anna M.; Nuermberger, Eric L.; Schnappinger, Dirk; Read, Kevin D.; Encinas, Lourdes; Bates, Robert H.; Wyatt, Paul G.; Cleghorn, Laura A. T.
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GSK2556286 Is a Novel Antitubercular Drug Candidate Effective In Vivo with the Potential To Shorten Tuberculosis Treatment
err2022-06-21
err28
errOAAI
errNuermberger, Eric L.; Martinez-Martinez, Maria Santos; Sanz, Olalla; Urones, Beatriz; Esquivias, Jorge; Soni, Heena; Tasneen, Rokeya; Tyagi, Sandeep; Li, Si-Yang; Converse, Paul J.; Boshoff, Helena I.; Robertson, Gregory T.; Besra, Gurdyal S.; Abrahams, Katherine A.; Upton, Anna M.; Mdluli, Khisimuzi; Boyle, Gary W.; Turner, Sam; Fotouhi, Nader; Cammack, Nicholas C.; Siles, Juan Miguel; Alonso, Marta; Escribano, Jaime; Lelievre, Joel; Rullas-Trincado, Joaquin; Perez-Herran, Esther; Bates, Robert H.; Maher-Edwards, Gareth; Barros, David; Ballell, Lluis; Jimenez, Elena
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Spiropyrimidinetriones: a Class of DNA Gyrase Inhibitors with Activity against Mycobacterium tuberculosis and without Cross-Resistance to Fluoroquinolones
err2022-04-19
err15
errOAAI
errBasarab, Gregory S.; Ghorpade, Sandeep; Gibhard, Liezl; Mueller, Rudolf; Njoroge, Mathew; Peton, Nashied; Govender, Preshendren; Massoudi, Lisa M.; Robertson, Gregory Thomas; Lenaerts, Anne J.; Boshoff, Helena Ingrid; Joerss, Douglas; Parish, Tanya; Durand-Reville, Thomas F.; Perros, Manos; Singh, Vinayak; Chibale, Kelly
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