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收藏Tetrahydropyridine LIMK inhibitors: Structure activity studies and biological characterization
Champire, Anthony; Berabez, Rayan; Braka, Abdennour; Cosson, Aurelie; Corret, Justine; Girardin, Caroline; Serrano, Amandine; Aci-Seche, Samia; Bonnet, Pascal; Josselin, Beatrice; Brindeau, Pierre; Ruchaud, Sandrine; Leguevel, Remy; Chatterjee, Deep; Mathea, Sebastian; Knapp, Stefan; Brion, Regis; Verrecchia, Franck; Vallee, Beatrice; Ple, Karen; Benedetti, Helene; Routier, Sylvain
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收藏Investigation of Ln3+ complexation by a DOTA derivative substituted by an imidazothiadiazole: synthesis, solution structure, luminescence and relaxation properties
Caillet, Emma; Nunes, Lea; Eliseeva, Svetlana V.; Ndiaye, Modou; Isaac, Manon; Pallier, Agnes; Morfin, Jean-Francois; Meudal, Herve; Petoud, Stephane; Routier, Sylvain; Platas-Iglesias, Carlos; Buron, Frederic; Bonnet, Celia S.
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收藏Glycosaminoglycan Mimetics Obtained by Microwave-Assisted Sulfation of Marine Bacterium Sourced Infernan Exopolysaccharide
Colliec-Jouault, Sylvia; Esposito, Fabiana; Ledru, Helene; Sinquin, Corinne; Marchand, Laetitia; Fillaudeau, Arnaud; Routier, Sylvain; Buron, Frederic; Lopin-Bon, Chrystel; Cuenot, Stephane; Bedini, Emiliano; Zykwinska, Agata
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收藏Development and preclinical evaluation of [18F]FBVM as a new potent PET tracer for vesicular acetylcholine transporter
Vercouillie, Johnny; Buron, Frederic; Serriere, Sophie; Rodrigues, Nuno; Gulhan, Zuhal; Chartier, Agnes; Chicheri, Gabrielle; Marzag, Hamid; Oury, Adeline; Percina, Nathalie; Bodard, Sylvie; Ben Othman, Rajah; Busson, Julie; Suzenet, Franck; Guilloteau, Denis; Marchivie, Mathieu; Emond, Patrick; Routier, Sylvain; Chalon, Sylvie
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收藏Selection of Bis-Indolyl Pyridines and Triphenylamines as New Inhibitors of SARS-CoV-2 Cellular Entry by Modulating the Spike Protein/ACE2 Interfaces通过调节Spike蛋白/ACE2界面选择双吲哚吡啶和三苯胺作为SARS-CoV-2细胞进入的新抑制剂
Lapaillerie, Delphine; Charlier, Cathy; Guyonnet-Duperat, Veronique; Murigneux, Emilie; Fernandes, Henrique S.; Martins, Fabio G.; Magalhaes, Rita P.; Vieira, Tatiana F.; Richetta, Clemente; Subra, Frederic; Lebourgeois, Samuel; Charpentier, Charlotte; Descamps, Diane; Visseaux, Benoit; Weigel, Pierre; Favereaux, Alexandre; Beauvineau, Claire; Buron, Frederic; Teulade-Fichou, Marie-Paule; Routier, Sylvain; Gallois-Montbrun, Sarah; Meertens, Laurent; Delelis, Olivier; Sousa, Sergio F.; Parissi, Vincent
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收藏Design and biological evaluation of substituted 5,7-dihydro-6H-indolo[2,3-c]quinolin-6-one as novel selective Haspin inhibitors
Avula, Sreenivas; Peng, Xudan; Lang, Xingfen; Tortorella, Micky; Josselin, Beatrice; Bach, Stephane; Bourg, Stephane; Bonnet, Pascal; Buron, Frederic; Ruchaud, Sandrine; Routier, Sylvain; Neagoie, Cleopatra
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收藏Design, Synthesis and SAR in 2,4,7-Trisubstituted Pyrido[3,2-d]Pyrimidine Series as Novel PI3K/mTOR Inhibitors
Buron, Frederic; Rodrigues, Nuno; Saurat, Thibault; Hiebel, Marie Aude; Bourg, Stephane; Bonnet, Pascal; Nehme, Reine; Morin, Philippe; Percina, Nathalie; Corret, Justine; Vallee, Beatrice; le Guevel, Remy; Jourdan, Marie-Lise; Benedetti, Helene; Routier, Sylvain
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收藏Prodromal neuroinflammatory, cholinergic and metabolite dysfunction detected by PET and MRS in the TgF344-AD transgenic rat model of AD: a collaborative multi-modal study
Chaney, Aisling M.; Lopez-Picon, Francisco R.; Serriere, Sophie; Wang, Rui; Bochicchio, Daniela; Webb, Samuel D.; Vandesquille, Matthias; Harte, Michael K.; Georgiadou, Christina; Lawrence, Catherine; Busson, Julie; Vercouillie, Johnny; Tauber, Clovis; Buron, Frederic; Routier, Sylvain; Reekie, Tristan; Snellman, Anniina; Kassiou, Michael; Rokka, Johanna; Davies, Karen E.; Rinne, Juha O.; Salih, Dervis A.; Edwards, Frances A.; Orton, Llwyd D.; Williams, Stephen R.; Chalon, Sylvie; Boutin, Herve
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收藏Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation
Elie, Jonathan; Feizbakhsh, Omid; Desban, Nathalie; Josselin, Beatrice; Baratte, Blandine; Bescond, Amandine; Duez, Julien; Fant, Xavier; Bach, Stephane; Marie, Dominique; Place, Matthieu; Ben Salah, Sami; Chartier, Agnes; Berteina-Raboin, Sabine; Chaikuad, Apirat; Knapp, Stefan; Carles, Fabrice; Bonnet, Pascal; Buron, Frederic; Routier, Sylvain; Ruchaud, Sandrine
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收藏Bis(het)aryl-1,2,3-triazole quinuclidines as α7 nicotinic acetylcholine receptor ligands: Synthesis, structure affinity relationships, agonism activity, [18F]-radiolabeling and PET study in rats
Ouach, Aziz; Vercouillie, Johnny; Bertrand, Emilie; Rodrigues, Nuno; Pin, Frederic; Serriere, Sophie; Boiaryna, Liliana; Chartier, Agnes; Percina, Nathalie; Tangpong, Pakorn; Gulhan, Zuhal; Mothes, Celine; Deloye, Jean-Bernard; Guilloteau, Denis; Page, Guylene; Suzenet, Franck; Buron, Frederic; Chalon, Sylvie; Routier, Sylvain
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