未登录 An SH3-binding allosteric modulator stabilizes the global conformation of the AML-associated Src-family kinase, Hck SH3-binding变构调节剂稳定AML相关Src家族激酶Hck的整体构象 Selzer, Ari M.; Gerlach, Gabriella; Gonzalez-Areizaga, Giancarlo; Wales, Thomas E.; Cui, Stephanie Y.; Iyer, Prema; Engen, John R.; Camacho, Carlos; Ishima, Rieko; Smithgall, Thomas E. 分享 收藏
Design, Synthesis, and Structure-Activity Relationships of Novel Peptide Derivatives of the Severe Acute Respiratory Syndrome-Coronavirus-2 Spike-Protein that Potently Inhibit Nicotinic Acetylcholine Receptors Hone, Arik J.; Santiago, Ulises; Harvey, Peta J.; Tekarli, Bassel; Gajewiak, Joanna; Craik, David J.; Camacho, Carlos J.; Mcintosh, J. Michael 分享 收藏
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A heterotypic assembly mechanism regulates CHIP E3 ligase activity (vol 41, e109566 , 2022) Das, Aniruddha; Thapa, Pankaj; Santiago, Ulises; Shanmugam, Nilesh; Banasiak, Katarzyna; Dazbrowska, Katarzyna; Nolte, Hendrik; Szulc, Natalia A.; Gathungu, Rose M.; Cysewski, Dominik; Krueeger, Marcus; Dadlez, Michal; Nowotny, Marcin; Camacho, Carlos J.; Hoppe, Thorsten; Pokrzywa, Wojciech 分享 收藏
A peptidomimetic modulator of the CaV2.2 N- type calcium channel for chronic pain Gomez, Kimberly; Santiago, Ulises; Nelson, Tyler S.; Allen, Heather N.; Calderon-Rivera, Aida; Hestehave, Sara; Palma, Erick J. Rodriguez; Zhou, Yuan; Duran, Paz; Loya-Lopez, Santiago; Zhu, Elaine; Kumar, Upasana; Shields, Rory; Koseli, Eda; McKiver, Bryan; Giuvelis, Denise; Zuo, Wanhong; Inyang, Kufreobong E.; Dorame, Angie; Chefdeville, Aude; Ran, Dongzhi; Perez-Miller, Samantha; Lu, Yi; Liu, Xia; Handokon; Arora, Paramjit S.; Patek, Marcel; Moutal, Aubin; Khanna, May; Hu, Huijuan; Laumet, Geoffroy; King, Tamara; Wang, Jing; Damaj, M. Imad; Korczeniewska, Olga A.; Camacho, Carlos J.; Khanna, Rajesh 分享 收藏
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Favorable outcomes of NPM1mut AML patients are due to transcriptional inactivation of FOXM1, presenting a new target to overcome chemoresistance Khan, I.; Kaempf, A.; Raghuwanshi, S.; Chesnokov, M.; Zhang, X.; Wang, Z.; Domling, A.; Tyner, J. W.; Camacho, C.; Gartel, A. L. 分享 收藏
Modulation of the substrate specificity of the kinase PDK1 by distinct conformations of the full- length protein Sacerdoti, Mariana; Gross, Lissy Z. F.; Riley, Andrew M.; Zehnder, Karin; Ghode, Abhijeet; Klinke, Sebastian; Anand, Ganesh Srinivasan; Paris, Kristina; Winkel, Angelika; Herbrand, Amanda K.; Godage, H. Yasmin; Cozier, Gyles E.; Suss, Evelyn; Schulze, Joerg O.; Pastor-Flores, Daniel; Bollini, Mariela; Cappellari, Maria Victoria; Svergun, Dmitri; Graewert, Melissa A.; Aramendia, Pedro F.; Leroux, Alejandro E.; Potter, Barry V. L.; Camacho, Carlos J.; Biondi, Ricardo M. 分享 收藏
Discovery and Biological Characterization of PRMT5:MEP50 Protein-Protein Interaction Inhibitors Asberry, Andrew M.; Cai, Xinpei; Deng, Xuehong; Santiago, Ulises; Liu, Sheng; Sims, Hunter S.; Liang, Weida; Xu, Xueyong; Wan, Jun; Jiang, Wen; Camacho, Carlos J.; Dai, Mingji; Hu, Chang-Deng 分享 收藏
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A dimer-monomer switch controls CHIP-dependent substrate ubiquitylation and processing Balaji, Vishnu; Mueller, Leonie; Lorenz, Robin; Kevei, Eva; Zhang, William H.; Santiago, Ulises; Gebauer, Jan; Llamas, Ernesto; Vilchez, David; Camacho, Carlos J.; Pokrzywa, Wojciech; Hoppe, Thorsten 分享 收藏
A heterotypic assembly mechanism regulates CHIP E3 ligase activity Das, Aniruddha; Thapa, Pankaj; Santiago, Ulises; Shanmugam, Nilesh; Banasiak, Katarzyna; Dabrowska, Katarzyna; Nolte, Hendrik; Szulc, Natalia A.; Gathungu, Rose M.; Cysewski, Dominik; Krueger, Marcus; Dadlez, Michal; Nowotny, Marcin; Camacho, Carlos J.; Hoppe, Thorsten; Pokrzywa, Wojciech 分享 收藏
A specific inhibitor of ALDH1A3 regulates retinoic acid biosynthesis in glioma stem cells Li, Jianfeng; Garavaglia, Silvia; Ye, Zhaofeng; Moretti, Andrea; Belyaeva, Olga, V; Beiser, Alison; Ibrahim, Md; Wilk, Anna; McClellan, Steve; Klyuyeva, Alla, V; Goggans, Kelli R.; Kedishvili, Natalia Y.; Salter, E. Alan; Wierzbicki, Andrzej; Migaud, Marie E.; Mullett, Steven J.; Yates, Nathan A.; Camacho, Carlos J.; Rizzi, Menico; Sobol, Robert W. 分享 收藏
Chitinase-3-like 1 protein complexes modulate macrophage-mediated immune suppression in glioblastoma Chen, Apeng; Jiang, Yinan; Li, Zhengwei; Wu, Lingxiang; Santiago, Ulises; Zou, Han; Cai, Chunhui; Sharma, Vaibhav; Guan, Yongchang; McCarl, Lauren H.; Ma, Jie; Wu, Yijen L.; Michel, Joshua; Shi, Yi; Konnikova, Liza; Amankulor, Nduka M.; Zinn, Pascal O.; Kohanbash, Gary; Agnihotri, Sameer; Lu, Songjian; Lu, Xinghua; Sun, Dandan; Gittes, George K.; Wang, Qianghu; Xiao, Xiangwei; Yimlamai, Dean; Pollack, Ian F.; Camacho, Carlos J.; Hu, Baoli 分享 收藏
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MAP2 is differentially phosphorylated in schizophrenia, altering its function Grubisha, M. J.; Sun, X.; MacDonald, M. L.; Garver, M.; Sun, Z.; Paris, K. A.; Patel, D. S.; DeGiosio, R. A.; Lewis, D. A.; Yates, N. A.; Camacho, C.; Homanics, G. E.; Ding, Y.; Sweet, R. A. 分享 收藏
Tripeptide IRW Upregulates NAMPT Protein Levels in Cells and Obese C57BL/6J Mice Bhullar, Khushwant S.; Son, Myoungjin; Kerek, Evan; Cromwell, Christopher R.; Wingert, Bentley M.; Wu, Kaiyu; Jovel, Juan; Camacho, Carlos J.; Hubbard, Basil P.; Wu, Jianping 分享 收藏
De novo emergence of adaptive membrane proteins from thymine-rich genomic sequences (vol 11, 781, 2020) 来自富含胸腺嘧啶的基因组序列的适应性膜蛋白的从头出现 (vol 11,781,2020) Vakirlis, Nikolaos; Acar, Omer; Hsu, Brian; Coelho, Nelson Castilho; Van Oss, S. Branden; Wacholder, Aaron; Medetgul-Ernar, Kate; Bowman, Ray W., II; Hines, Cameron P.; Iannotta, John; Parikh, Saurin Bipin; McLysaght, Aoife; Camacho, Carlos J.; O'Donnell, Allyson F.; Ideker, Trey; Carvunis, Anne-Ruxandra 分享 收藏
De novo emergence of adaptive membrane proteins from thymine-rich genomic sequences 来自富含胸腺嘧啶的基因组序列的适应性膜蛋白的从头出现 Vakirlis, Nikolaos; Acar, Omer; Hsu, Brian; Coelho, Nelson Castilho; Van Oss, S. Branden; Wacholder, Aaron; Medetgul-Ernar, Kate; Bowman, Ray W., II; Hines, Cameron P.; Iannotta, John; Parikh, Saurin Bipin; McLysaght, Aoife; Camacho, Carlos J.; O'Donnell, Allyson F.; Ideker, Trey; Carvunis, Anne-Ruxandra 分享 收藏
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