未登录 First-in-class nonsteroidal anti-inflammatory drug and carbonic anhydrase inhibitor hybrid compounds as effective antimycobacterial agents 第一类非甾体抗炎药和碳酸酐酶抑制剂杂合化合物作为有效的抗分枝杆菌剂 Parkkinen, Jenny; Akgul, Ozlem; Berrino, Emanuela; Carta, Fabrizio; Selleri, Silvia; Hammaren, Milka; Aspatwar, Ashok; Bartolucci, Gianluca; Capasso, Clemente; Parikka, Mataleena; Parkkila, Seppo; Supuran, Claudiu T. 分享 收藏
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Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T. 分享 收藏
Green Synthesis of Sulfonamide Derivatives as Human Carbonic Anhydrase Isoforms I, II, IX, XII Inhibitors and Antioxidants: Comprehensive Insights From Biological Evaluation and In-Depth In Silico Analysis 绿色合成磺胺衍生物作为人碳酸酐酶同工酶I、II、IX、XII抑制剂和抗氧化剂：来自生物评价和深入计算机模拟分析的全面见解 Mishra, K. M. Abha; Kumari, Nutan; Carta, Fabrizio; Renzi, Gioele; Singh, Harshdeep; Supuran, Claudiu T.; Sethi, Kalyan K. 分享 收藏
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Unraveling the Potential of Amino-, Acylamino-, and Ureido-Substituted 3H-1,2-Benzoxaphosphepine 2-Oxides toward Nanomolar Inhibitors of Tumor-Associated Carbonic Anhydrases IX and XII 揭示氨基、酰胺氨基和脲基取代的3H-1,2-苯并恶磷杂庚英烷2-氧化物作为肿瘤相关碳酸酐酶IX和XII纳摩尔抑制剂的潜力 Balasova, A; Pustenko, A; Angeli, A; Andreucci, E; Biagioni, A; Nocentini, A; Carta, F; Supuran, CT; Zalubovskis, R 分享 收藏
Discovery of Trypanosoma cruzi Carbonic Anhydrase Inhibitors by a Combination of Ligand- and Structure-Based Virtual Screening 通过结合配体和基于结构的虚拟筛选发现克氏锥虫碳酸酐酶抑制剂 Gori, Denis N. Prada; Barrionuevo, Emilia M.; Alberca, Lucas N.; Sbaraglini, Maria L.; Llanos, Manuel A.; Giovannuzzi, Simone; Carta, Fabrizio; Marchetto, Matias I.; Supuran, Claudiu T.; Soto, Catalina D. Alba; Gavernet, Luciana; Talevi, Alan 分享 收藏
Discover the Power of Lithospermic Acid as Human Carbonic Anhydrase VA and Pancreatic Lipase Inhibitor Through In Silico and In Vitro Studies 通过体内外研究探索 lithospermic acid 作为人碳酸酐酶 VA 和胰腺脂肪酶抑制剂的潜力 Citriniti, Emanuele Liborio; Rocca, Roberta; Costa, Giosue; Sciacca, Claudia; Cardullo, Nunzio; Muccilli, Vera; Karioti, Anastasia; Carta, Fabrizio; Supuran, Claudiu T.; Alcaro, Stefano; Ortuso, Francesco 分享 收藏
In Vitro CO-Releasing and Antioxidant Properties of Sulfonamide-Based CAI-CORMs in a H2O2-Stimulated Human Achilles Tendon-Derived Cell Model 磺胺类cai-corms在H2O2-Stimulated人跟腱来源细胞模型中的体外共释放和抗氧化特性 Berrino, Emanuela; Guglielmi, Paolo; Carta, Fabrizio; Carradori, Simone; Campestre, Cristina; Angeli, Andrea; Arrighi, Francesca; Pontecorvi, Virginia; Chimenti, Paola; Secci, Daniela; Supuran, Claudiu T.; Gallorini, Marialucia 分享 收藏
Design, Synthesis, and In Vitro Evaluation of Aromatic Sulfonamides as Human Carbonic Anhydrase I, II, IX, and XII Inhibitors and Their Antioxidant Activity Mishra, K. M. Abha; Kumari, Nutan; Carta, Fabrizio; Renzi, Gioele; Supuran, Claudiu T.; Sethi, Kalyan K. 分享 收藏
X-ray crystallographic and kinetic studies of biguanide containing aryl sulfonamides as carbonic anhydrase inhibitors Baroni, Chiara; Bozdag, Murat; Renzi, Gioele; De Luca, Viviana; Capasso, Clemente; Bazzicalupi, Carla; Selleri, Silvia; Ferraroni, Marta; Carta, Fabrizio; Supuran, Claudiu T. 分享 收藏
Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms Kilbile, Jaydeo T.; Sapkal, Suryakant B.; Renzi, Gioele; D'Agostino, Ilaria; Boudjelal, Mohamed; Tamboli, Yasinalli; Cutarella, Luigi; Mori, Mattia; Sgambellone, Silvia; Villano, Serafina; Marri, Silvia; Lucarini, Laura; Carradori, Simone; Carta, Fabrizio; Supuran, Claudiu T. 分享 收藏
Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study 抑制铜绿假单胞菌碳酸酐酶，探索环丙沙星对新型抗菌剂的功能化: 深入的多学科研究 Marinacci, Beatrice; D'Agostino, Ilaria; Angeli, Andrea; Carradori, Simone; Melfi, Francesco; Grande, Rossella; Corsiani, Micol; Ferraroni, Marta; Agamennone, Mariangela; Tondo, Anna Rita; Zara, Susi; Puca, Valentina; Pellegrini, Benedetta; Vagaggini, Chiara; Dreassi, Elena; Patrauchan, Marianna A.; Capasso, Clemente; Nicolotti, Orazio; Carta, Fabrizio; Supuran, Claudiu T. 分享 收藏
Superacid-Synthesized Fluorinated Diamines Act as Selective hCA IV Inhibitors Berrino, Emanuela; Michelet, Bastien; Vitse, Kassandra; Nocentini, Alessio; Bartolucci, Gianluca; Martin-Mingot, Agnes; Gratteri, Paola; Carta, Fabrizio; Supuran, Claudiu T.; Thibaudeau, Sebastien 分享 收藏
Lasamide, a Potent Human Carbonic Anhydrase Inhibitor from the Market: Inhibition Profiling and Crystallographic Studies Lasamide，一种来自市场的有效人类碳酸酐酶抑制剂: 抑制分析和晶体学研究 Baroni, Chiara; D'Agostino, Ilaria; Renzi, Gioele; Kilbile, Jaydeo T.; Tamboli, Yasinalli; Ferraroni, Marta; Carradori, Simone; Capasso, Clemente; Carta, Fabrizio; Supuran, Claudiu T. 分享 收藏
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