Benjamin D. Cons - Publications, H-index & Citations

Benjamin D. Cons

Astex Pharmaceuticals

9H指数

17论文数

376被引数

收录论文 9

发表时间

Fragment-Based Discovery of a Series of Allosteric-Binding Site Modulators of β-Glucocerebrosidase

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2024-06-27

PREAI

Palmer, Nick; Agnew, Christopher; Benn, Caroline; Buffham, William J.; Castro, Joan N.; Chessari, Gianni; Clark, Mellissa; Cons, Benjamin D.; Coyle, Joseph E.; Dawson, Lee A.; Hamlett, Christopher C. F.; Hodson, Charlotte; Holding, Finn; Johnson, Christopher N.; Liebeschuetz, John W.; Mahajan, Pravin; McCarthy, James M.; Murray, Christopher W.; O'Reilly, Marc; Peakman, Torren; Price, Amanda; Rapti, Magdalini; Reeks, Judith; Schopf, Patrick; St-Denis, Jeffrey D.; Valenzano, Chiara; Wallis, Nicola G.; Walser, Reto; Weir, Heather; Wilsher, Nicola E.; Woodhead, Andrew; Bento, Carla F.; Tisi, Dominic

Alkene 1,3-Difluorination via Transient Oxonium Intermediates

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

IF16.9

2024-06-20

OAAI

Dean, Alice C.; Randle, E. Harvey; Lacey, Andrew J. D.; Giorio, Guilherme A. Marczak; Doobary, Sayad; Cons, Benjamin D.; Lennox, Alastair J. J.

Enabling synthesis in fragment-based drug discovery (FBDD): microscale high-throughput optimisation of the medicinal chemist's toolbox reactions

RSC MEDICINAL CHEMISTRY

IF3.6

2023-01-01

PREAI

Townley, Chloe; Branduardi, Davide; Chessari, Gianni; Cons, Benjamin D.; Griffiths-Jones, Charlotte; Hall, Richard J.; Johnson, Christopher N.; Ochi, Yuji; Whibley, Stuart; Grainger, Rachel

X-ray Screening of an Electrophilic Fragment Library and Application toward the Development of a Novel ERK 1/2 Covalent Inhibitor

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2022-09-14

PREAI

St Denis, Jeffrey D.; Chessari, Gianni; Cleasby, Anne; Cons, Benjamin D.; Cowan, Suzanna; Dalton, Samuel E.; East, Charlotte; Murray, Christopher W.; O'Reilly, Marc; Peakman, Torren; Rapti, Magdalini; Stow, Jessie L.

Fragment-Based Discovery of a Novel, Brain Penetrant, Orally Active HDAC2 Inhibitor

ACS MEDICINAL CHEMISTRY LETTERS

IF4

2022-09-06

OAAI

Tamanini, Emiliano; Miyamura, Shin; Buck, Ildiko M.; Cons, Benjamin D.; Dawson, Lee; East, Charlotte; Futamura, Takashi; Goto, Shintaro; Griffiths-Jones, Charlotte; Hashimoto, Tetsuya; Heightman, Tom D.; Ishikawa, Shunpei; Ito, Hideki; Kaneko, Yosuke; Kawato, Tatsuya; Kondo, Kazumi; Kurihara, Naoki; McCarthy, James M.; Mori, Yukiko; Nagase, Tsuyoshi; Nakaishi, Yuichiro; Reeks, Judith; Sato, Akimasa; Schopf, Patrick; Tai, Kuninori; Tamai, Taichi; Tisi, Dominic; Woolford, Alison J. -A.

Electrostatic Complementarity in Structure-Based Drug Design

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2022-05-05

PREAI

Cons, Benjamin D.; Twigg, David G.; Kumar, Rajendra; Chessari, Gianni

Fragment-based drug discovery and its application to challenging drug targets

STRUCTURE-BASED DRUG DESIGN: INSIGHTS FROM ACADEMIA AND INDUSTRY

IF0

2017-11-08

PREAI

Price, Amanda J.; Howard, Steven; Cons, Benjamin D.